Target Details
UniProt ACP46098
Gene SymbolHTR3A
Protein Name5-hydroxytryptamine receptor 3A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 382
  • Clinical molecules 7
  • Avg pChEMBL 7.39
Top Co-occurrence Targets
Active Molecules (382)
InChIKey pChEMBL Type Targets Clinical
ZPEDRMCLQWINAG 8.8 Ki 5
LZFIKFXIHTZOJR 8.8 Ki 2
QZNZJWLUNDXZQA 8.8 Ki 5
HBDLBTSITBUDIR 8.8 Ki 2
BUXACHZAYWAZJL 8.7 Ki 7
ZVJIBTNUNUXAIO 8.7 Ki 5
JAPSHKUKFHJHQZ 8.7 IC50 5
RBZYOKIYUDKYOZ 8.7 IC50 5
XRXDAJYKGWNHTQ 8.7 Ki 13 Yes
XUKROCVZGZNGSI 8.7 Ki 2
AASFRXJJHSMTFI 8.6 IC50 5
PEDIKBSWZVFPLW 8.6 IC50 5
HSLUKGWVBNRWNC 8.6 IC50 5
ZGUGXTYWGBQHSU 8.6 Ki 5
PDWZKMOQJPHUIY 8.6 Ki 5
DNVBBWNTRFFIHW 8.6 Ki 2
TXCYUSKWBHUVEP 8.6 IC50 2
VCADIWSEVTZZOR 8.6 Ki 3
ZNRGQMMCGHDTEI 8.6 Ki 9
HOMWNUXPSJQSSU 8.5 Ki 6
ICKPJMDBIACNSE 8.5 Ki 3
LWQLZCWBSPLMBP 8.5 Ki 3
NNRSVGLUJAPMQD 8.5 Ki 5
GZSKEXSLDPEFPT 8.5 Kd 5
CKUTYLGHNWXIJF 8.5 Ki 5
FELGMEQIXOGIFQ 8.5 Ki 10
BLLXLUVDRGHQHD 8.5 IC50 5
APTTVZDGFWGGHT 8.4 Kd 5
MPZDFMTUBDIVPH 8.4 IC50 5
OYASVWZGKNBLSA 8.3 IC50 5
HNDAZSYDBSRFST 8.3 Ki 2
KYIGOCCCBXRHNJ 8.3 IC50 43
BSNKYWSMUAGMDO 8.3 IC50 2
CKXVQPZQTVVCCB 8.3 Kd 5
DNQOMGGYJRBLOX 8.3 Kd 5
PXNBOFBSFXZTES 8.3 Ki 5
RMKNXTZRZSDIHT 8.3 IC50 5
ACKJXXOVSOCBPX 8.2 Ki 3
DXPJJGVPGVKFPQ 8.2 IC50 5
YQUHQGUROPITGF 8.2 Ki 5
WFQOETMVYMINSA 8.2 IC50 4
XLVVGMWYXBVUJZ 8.2 Ki 5
ACSDLURGGYXLSE 8.2 IC50 5
GLWWAUFFFXRHOL 8.2 Ki 2
VXYGXEFRVWLJIR 8.2 IC50 5
MNJNPLVXBISNSX 8.2 IC50 5
LJMASYWVOMQDML 8.2 IC50 5
IONCWLLKDMISKP 8.1 Ki 2
KVDHVTQKKLVMJD 8.1 Ki 5
ZKSNSGVNASDNFY 8.1 Ki 5
2D structure