Target Details
| UniProt AC | P45984 |
|---|---|
| Gene Symbol | MAPK9 |
| Protein Name | Mitogen-activated protein kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 676
- Clinical molecules 191
- Avg pChEMBL 6.96
KEGG Pathways (75)
- AGE-RAGE signaling pathway in diabetic complications
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Colorectal cancer
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- ErbB signaling pathway
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Huntington disease
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- Pancreatic cancer
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Protein processing in endoplasmic reticulum
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tight junction
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Type II diabetes mellitus
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Active Molecules (676)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NUEDKDFHLPVYRY
|
6.7 | IC50 | 2 | Yes | |
RCYPVQCPYKNSTG
|
6.7 | IC50 | 7 | — | |
RWVFVOHUWIBKDI
|
6.7 | IC50 | 2 | — | |
XTJZKALDRPVFSN
|
6.7 | IC50 | 5 | — | |
LGICVDGDWJJCIH
|
6.7 | IC50 | 2 | — | |
CCDFASODNLEBEJ
|
6.6 | IC50 | 3 | — | |
JANAZDXNIOBICQ
|
6.6 | IC50 | 5 | — | |
LGICVDGDWJJCIH
|
6.6 | IC50 | 2 | — | |
MXRSDWOBSNRDKJ
|
6.6 | IC50 | 3 | Yes | |
UBQAXNUSTYBVJI
|
6.6 | IC50 | 3 | Yes | |
YYLKKYCXAOBSRM
|
6.6 | Kd | 191 | — | |
DZYPGOHFOPGXTC
|
6.6 | IC50 | 2 | Yes | |
JOOXLOJCABQBSG
|
6.6 | Kd | 139 | — | |
MPVGZUGXCQEXTM
|
6.6 | Kd | 61 | Yes | |
OYXVJMGNNKEOSX
|
6.6 | IC50 | 3 | — | |
QBROFJFJPQJMEQ
|
6.6 | IC50 | 3 | — | |
QLCYBHBQDYLQLC
|
6.6 | IC50 | 2 | — | |
RHLSCLBSPZIGFS
|
6.6 | IC50 | 3 | Yes | |
RLAJOHAIIACFAM
|
6.6 | IC50 | 13 | Yes | |
SVYQRMQQKKCGBE
|
6.6 | IC50 | 2 | Yes | |
JPCGBNVFAUAQSJ
|
6.6 | IC50 | 2 | — | |
KAEBPVNZHCYYSN
|
6.6 | IC50 | 3 | Yes | |
NHSDXYBXQGQSRA
|
6.6 | IC50 | 3 | — | |
FUMCKNCUEAQHCV
|
6.6 | Ki | 103 | — | |
JJGSOVIZOMZMCS
|
6.6 | Ki | 35 | — | |
KKYPRNBBPBRJQX
|
6.6 | Ki | 40 | — | |
LCBNUBGZQBBNPG
|
6.6 | IC50 | 2 | Yes | |
NLUPJKQOKWBWFC
|
6.6 | Ki | 69 | — | |
RPBRKXHDLFDUJN
|
6.6 | IC50 | 2 | — | |
UGZLJUFPCPHHSW
|
6.6 | IC50 | 3 | Yes | |
YPLNLOJZEWIBMR
|
6.6 | IC50 | 2 | — | |
ZGZVRPRSFXRGCF
|
6.6 | Ki | 76 | — | |
HJEPFPDXSFKWQH
|
6.6 | IC50 | 3 | — | |
MXRSDWOBSNRDKJ
|
6.6 | IC50 | 2 | Yes | |
NDIUYMHNCUTVGE
|
6.6 | Ki | 25 | — | |
PBKYQJDUQYHRCL
|
6.6 | IC50 | 2 | — | |
FFPJBQIHDBPVHZ
|
6.6 | IC50 | 3 | Yes | |
FRZMEKOENCSLON
|
6.6 | IC50 | 2 | — | |
GXSSKILQHZMJFZ
|
6.6 | IC50 | 2 | — | |
JMOMBPSAYLGZAN
|
6.6 | IC50 | 2 | — | |
ZBEPMOZEXLGCTF
|
6.6 | IC50 | 3 | — | |
ABBHPRNOFIXTQU
|
6.6 | IC50 | 2 | — | |
QDMXVKKPYBGIAS
|
6.5 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
6.5 | Kd | 231 | Yes | |
VMVANPCSWYULOT
|
6.5 | Kd | 3 | — | |
WWHNHBJMWMVKHQ
|
6.5 | IC50 | 4 | Yes | |
YIVZAUQCWPPATQ
|
6.5 | IC50 | 2 | — | |
WBSWWONMTZEOGS
|
6.5 | Kd | 5 | — | |
XVIMTHVVBGUFCB
|
6.5 | IC50 | 3 | Yes | |
ZUYSNKSNKMMPMB
|
6.5 | IC50 | 2 | — |