Target Details
| UniProt AC | P45984 |
|---|---|
| Gene Symbol | MAPK9 |
| Protein Name | Mitogen-activated protein kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 676
- Clinical molecules 191
- Avg pChEMBL 6.96
KEGG Pathways (75)
- AGE-RAGE signaling pathway in diabetic complications
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Colorectal cancer
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- ErbB signaling pathway
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Huntington disease
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- Pancreatic cancer
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Protein processing in endoplasmic reticulum
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tight junction
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Type II diabetes mellitus
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Active Molecules (676)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RVSKJUNTDGBSSS
|
6.8 | Ki | 25 | — | |
VTTJSUDCCDBRRF
|
6.8 | IC50 | 3 | Yes | |
WIRUYYYAAJOIKO
|
6.8 | Ki | 4 | — | |
YYZKQTUYOUJSCB
|
6.8 | IC50 | 2 | — | |
ZEAYLBFKDUMFPX
|
6.8 | IC50 | 3 | — | |
FXBNFLKLXHFULB
|
6.8 | IC50 | 3 | Yes | |
QHGCJZAERWMAPE
|
6.8 | IC50 | 2 | — | |
SRTMONQYBOXBGE
|
6.8 | IC50 | 3 | Yes | |
STNCBMGTCZRJPA
|
6.8 | IC50 | 2 | — | |
DVRSTRMZTAPMKO
|
6.8 | IC50 | 10 | Yes | |
QMCGWRVMZPNHKW
|
6.8 | IC50 | 5 | — | |
MUNGYPZWBYEXFS
|
6.8 | IC50 | 2 | — | |
UWYRBEMRLWEHSY
|
6.8 | IC50 | 2 | — | |
WUFVFWHZRSJNAV
|
6.8 | IC50 | 4 | Yes | |
YMIHNRVATUXFGL
|
6.8 | IC50 | 2 | — | |
BXZQZGKOTDCAKN
|
6.7 | IC50 | 3 | — | |
DAJHYBRFYWDMMM
|
6.7 | IC50 | 2 | Yes | |
DWLWDAIUYUOIEU
|
6.7 | IC50 | 2 | — | |
GOUYNVPPUCUZSS
|
6.7 | IC50 | 6 | — | |
INYGRZCFSWSMOQ
|
6.7 | IC50 | 2 | — | |
FOAAMZPWLWPKOE
|
6.7 | IC50 | 3 | — | |
OIJDKSLOXVWFRV
|
6.7 | IC50 | 3 | Yes | |
PXOJJCCSYAVCPK
|
6.7 | IC50 | 3 | Yes | |
ATAFJTOBINKREW
|
6.7 | IC50 | 2 | — | |
HHAPAAFKKUAWAI
|
6.7 | IC50 | 5 | — | |
MAOSUPNJVJGJEU
|
6.7 | IC50 | 5 | — | |
MKHUGLZLKVCOGF
|
6.7 | IC50 | 2 | — | |
PHDVAWAUKMHEJM
|
6.7 | IC50 | 3 | Yes | |
PLJKGPIWOOUPAJ
|
6.7 | IC50 | 3 | — | |
BBJVUPIDQPSQJP
|
6.7 | IC50 | 2 | — | |
CZJALLIMKKSCNX
|
6.7 | IC50 | 2 | — | |
FFQQZBOORWKWDZ
|
6.7 | Ki | 3 | — | |
JEHSPMHADICABR
|
6.7 | IC50 | 3 | — | |
LQRBZQWMQBTWDI
|
6.7 | Ki | 3 | — | |
OHMPXDCOVKOOAN
|
6.7 | IC50 | 4 | — | |
PEEMSUJXJVLHFP
|
6.7 | Ki | 4 | — | |
QCOULMVHIHJKFY
|
6.7 | Ki | 14 | — | |
SBFPHSVZEXSHTL
|
6.7 | Ki | 62 | — | |
UTMRCMCLMBDPNW
|
6.7 | Ki | 10 | — | |
VYOMWAWIBCGOKB
|
6.7 | IC50 | 4 | — | |
BLKGCBHORBGPFK
|
6.7 | IC50 | 2 | Yes | |
FVOMNFNIDIQPDL
|
6.7 | IC50 | 3 | — | |
IMARJVJNXLXPIX
|
6.7 | IC50 | 3 | — | |
IXHWMGAFLNPNII
|
6.7 | IC50 | 6 | — | |
KORISVSXBGATCA
|
6.7 | IC50 | 2 | — | |
QHKYPYXTTXKZST
|
6.7 | Kd | 28 | — | |
NXXOMTBHZVIUJY
|
6.7 | IC50 | 2 | — | |
AVLYNJZZQYEFEA
|
6.7 | IC50 | 8 | Yes | |
CGUOXTCHDHXWRO
|
6.7 | IC50 | 2 | — | |
HENCYENWBZRSLR
|
6.7 | IC50 | 3 | — |