Target Details
| UniProt AC | P45984 |
|---|---|
| Gene Symbol | MAPK9 |
| Protein Name | Mitogen-activated protein kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 676
- Clinical molecules 191
- Avg pChEMBL 6.96
KEGG Pathways (75)
- AGE-RAGE signaling pathway in diabetic complications
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Colorectal cancer
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- ErbB signaling pathway
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Huntington disease
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- Pancreatic cancer
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Protein processing in endoplasmic reticulum
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tight junction
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Type II diabetes mellitus
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Active Molecules (676)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VWIDJTODOGUOHO
|
7.1 | IC50 | 2 | — | |
HJWMLCDGRWWLAQ
|
7.1 | IC50 | 3 | — | |
INESNNFVDPZTKT
|
7.1 | IC50 | 2 | — | |
NSPCSJPGLMJDCZ
|
7.1 | IC50 | 2 | — | |
OVKIYZXGCCAIJG
|
7.1 | Ki | 6 | — | |
RGNHKJWHFIPHIM
|
7.1 | Ki | 66 | — | |
RJZDECGDCKOHBV
|
7.1 | Ki | 70 | — | |
RQVKVJIRFKVPBF
|
7.1 | Ki | 13 | — | |
UDFDIIVNIYWXDM
|
7.1 | Ki | 74 | — | |
VNDWQCSOSCCWIP
|
7.1 | Ki | 39 | Yes | |
DNUIJDUIEIJBJM
|
7.1 | IC50 | 3 | — | |
KXABTDJSBKARGL
|
7.1 | IC50 | 2 | — | |
WQYDASORCSDVNY
|
7.1 | IC50 | 2 | — | |
YPUXXNJBUOZMOQ
|
7.1 | IC50 | 3 | Yes | |
CTQXMPOHMBPPMC
|
7.1 | IC50 | 3 | Yes | |
QVEWXFMWNGGSAH
|
7.1 | IC50 | 3 | Yes | |
BKBYGIARQARTNG
|
7.1 | IC50 | 4 | Yes | |
FVPQKFPGPOAQPF
|
7.1 | IC50 | 3 | — | |
VVVVSXKJECZPRY
|
7.1 | IC50 | 2 | — | |
BRTOSQAESSKFCB
|
7.1 | IC50 | 2 | — | |
HQZRYALYTLZTPR
|
7.1 | IC50 | 2 | — | |
YTPKEJXVUUNXRA
|
7.1 | IC50 | 4 | Yes | |
HGQHCYUSXPTRID
|
7.0 | IC50 | 4 | Yes | |
IHBXLESUKAAQDQ
|
7.0 | IC50 | 3 | Yes | |
XCPPIJCBCWUBNT
|
7.0 | IC50 | 3 | — | |
HDGJMVJJOYGVSR
|
7.0 | IC50 | 3 | Yes | |
CBSFDSPVUSGETR
|
7.0 | IC50 | 2 | — | |
OHUXKIXTONEVBL
|
7.0 | IC50 | 3 | Yes | |
XMMMCYBZGARUKP
|
7.0 | IC50 | 4 | — | |
FVONQZQMUHLATI
|
7.0 | IC50 | 3 | — | |
LZFPDJIWDHUHJG
|
7.0 | IC50 | 3 | — | |
IOZQORJWOUBHKH
|
7.0 | IC50 | 3 | Yes | |
JSQNZBQJTQNCFK
|
7.0 | IC50 | 7 | — | |
YLSFSAKXSQLGSF
|
7.0 | IC50 | 6 | — | |
YMSORXXIQGLXBK
|
7.0 | IC50 | 2 | — | |
YZJYYYWPZRYBLV
|
7.0 | IC50 | 3 | Yes | |
AHMHIFXJPSHHPH
|
7.0 | IC50 | 3 | Yes | |
FXGYCYAFWHJUAS
|
7.0 | Ki | 2 | — | |
HEKAIDKUDLCBRU
|
7.0 | Ki | 20 | — | |
HWNQWUTVZUBWMF
|
7.0 | IC50 | 2 | — | |
LZLQWVSFCFCTJH
|
7.0 | IC50 | 2 | — | |
MGRDWTIBFYFWSG
|
7.0 | IC50 | 2 | — | |
OWRXHGAFWZFFCW
|
7.0 | Ki | 113 | — | |
RTDSHUGNRVXRHN
|
7.0 | Ki | 51 | — | |
SRUYMJRFVGLQDV
|
7.0 | Ki | 37 | — | |
CDCZUMXTSTZOHL
|
7.0 | IC50 | 2 | — | |
DNQLQDZACRVRIW
|
7.0 | IC50 | 2 | — | |
PSUZEBSSYLZYCL
|
7.0 | IC50 | 2 | Yes | |
HSEASLMARZYTKL
|
7.0 | IC50 | 3 | — | |
UFPBREQEYCTWAI
|
7.0 | IC50 | 2 | — |