Target Details
| UniProt AC | P45984 |
|---|---|
| Gene Symbol | MAPK9 |
| Protein Name | Mitogen-activated protein kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 676
- Clinical molecules 191
- Avg pChEMBL 6.96
KEGG Pathways (75)
- AGE-RAGE signaling pathway in diabetic complications
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Colorectal cancer
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- ErbB signaling pathway
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Huntington disease
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- Pancreatic cancer
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Protein processing in endoplasmic reticulum
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tight junction
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Type II diabetes mellitus
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Active Molecules (676)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SVIILPGBQTUQPJ
|
7.3 | IC50 | 2 | — | |
WIHAOLDOGQOGIU
|
7.3 | Ki | 5 | — | |
XBAIEEJJCJHBDL
|
7.3 | Ki | 17 | — | |
JQCBHTULSVVPFD
|
7.3 | IC50 | 2 | — | |
ACDQVXJNZDLXFP
|
7.3 | IC50 | 3 | Yes | |
FTIAKTLRFKSDFR
|
7.3 | IC50 | 10 | Yes | |
JOWZBTCWJHFAQE
|
7.3 | IC50 | 4 | — | |
QXNPNLLIZGVUPQ
|
7.3 | IC50 | 3 | Yes | |
XYMGBQVLIQVGBW
|
7.3 | IC50 | 2 | — | |
AWTKTGLFVCACHC
|
7.3 | IC50 | 3 | Yes | |
KVDDBBDCWPLOFR
|
7.2 | IC50 | 3 | — | |
ODPGGGTTYSGTGO
|
7.2 | Kd | 153 | — | |
PDKJQLGOZQXLMW
|
7.2 | IC50 | 2 | — | |
QKJMPSJTHLLZPU
|
7.2 | IC50 | 3 | Yes | |
IPPNJZWFNCNYSG
|
7.2 | IC50 | 3 | — | |
DXTYYUXUIQZDHR
|
7.2 | IC50 | 3 | Yes | |
HWQRBIQRGAZWGS
|
7.2 | IC50 | 3 | Yes | |
VGQNDBIBHCCFKP
|
7.2 | IC50 | 3 | — | |
XQLINAVACFUFEH
|
7.2 | IC50 | 4 | Yes | |
ICDHVAJOGIGIOI
|
7.2 | Ki | 5 | — | |
MGNQNQOSSLCUFP
|
7.2 | Ki | 12 | — | |
AIPARAKSAHWEMY
|
7.2 | IC50 | 2 | — | |
FPOJVFPVFJTSDR
|
7.2 | IC50 | 3 | — | |
AEIKXFACENTHCD
|
7.2 | IC50 | 3 | Yes | |
FJVVBMGXZMJPOI
|
7.2 | IC50 | 3 | — | |
FJVVBMGXZMJPOI
|
7.2 | IC50 | 3 | — | |
GZFOTMBQLVXWAV
|
7.2 | IC50 | 2 | — | |
JGHISYSDWKNXIA
|
7.2 | IC50 | 3 | — | |
KEJPODFMUKBEAK
|
7.2 | IC50 | 3 | Yes | |
MIFPZJRPCSILQA
|
7.2 | IC50 | 3 | — | |
XIUOLJTWTRUVGZ
|
7.2 | IC50 | 2 | — | |
NGOYZSBSNHRWEM
|
7.2 | IC50 | 3 | — | |
OOXCRLOLUWLQCN
|
7.2 | IC50 | 3 | Yes | |
UGKKDOKVLSCRFL
|
7.2 | IC50 | 3 | Yes | |
VFFOCQZCDTURBY
|
7.2 | IC50 | 3 | Yes | |
XVLIRDXMQGPGCW
|
7.2 | IC50 | 4 | Yes | |
GXUIBOOECUSGTA
|
7.2 | IC50 | 2 | Yes | |
IJTANTDZFOCBKK
|
7.2 | IC50 | 3 | Yes | |
RXFQQWFTSGTXMV
|
7.2 | IC50 | 2 | — | |
TWTIIHVYOGLKME
|
7.2 | Ki | 3 | Yes | |
CEFHLBGJHWUOBZ
|
7.2 | Ki | 3 | — | |
MSNLSSCFMUKCNV
|
7.2 | IC50 | 3 | — | |
AJMFKZZQEDNOJZ
|
7.1 | IC50 | 4 | — | |
KDMADGZAPDHVHE
|
7.1 | IC50 | 6 | — | |
LMZRJJTWTQNOEI
|
7.1 | IC50 | 3 | Yes | |
YFZJFPUOKUFWQU
|
7.1 | IC50 | 4 | — | |
ZVDDPXIWKBBCQE
|
7.1 | IC50 | 3 | Yes | |
BEYORXSIIKUPCA
|
7.1 | IC50 | 2 | — | |
SGWLRDAOCLITOM
|
7.1 | IC50 | 7 | — | |
UQQRUYAIZCVJMP
|
7.1 | IC50 | 2 | — |