Target Details
| UniProt AC | P45984 |
|---|---|
| Gene Symbol | MAPK9 |
| Protein Name | Mitogen-activated protein kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 676
- Clinical molecules 191
- Avg pChEMBL 6.96
KEGG Pathways (75)
- AGE-RAGE signaling pathway in diabetic complications
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Colorectal cancer
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- ErbB signaling pathway
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Huntington disease
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- Pancreatic cancer
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Protein processing in endoplasmic reticulum
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tight junction
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Type II diabetes mellitus
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Active Molecules (676)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RGWMWOOWHJUGFL
|
7.5 | IC50 | 2 | — | |
WNTHBRVKPVTIQB
|
7.5 | IC50 | 3 | Yes | |
ZBBJZAWEQIRJKZ
|
7.5 | IC50 | 2 | — | |
AHYIIKWTYMCFNB
|
7.5 | IC50 | 3 | — | |
FPVKFPPNOMNINZ
|
7.5 | IC50 | 2 | — | |
SYSMFXCWULAWTA
|
7.4 | IC50 | 3 | Yes | |
UYJNQQDJUOUFQJ
|
7.4 | IC50 | 68 | — | |
XGTBIGDWHOVXDS
|
7.4 | IC50 | 3 | — | |
GZOYOEIHAGHGFM
|
7.4 | IC50 | 6 | — | |
HYNZVOLLNHBFQJ
|
7.4 | IC50 | 4 | Yes | |
IBGLGMOPHJQDJB
|
7.4 | IC50 | 3 | Yes | |
UCRSZQFDYBPHLJ
|
7.4 | IC50 | 3 | Yes | |
UDOITUAULPBVSE
|
7.4 | IC50 | 3 | Yes | |
ZRAANXMCPIIUKV
|
7.4 | IC50 | 2 | — | |
ACPOUJIDANTYHO
|
7.4 | IC50 | 17 | Yes | |
DDDPTRGZLJPPQR
|
7.4 | Ki | 6 | — | |
DICUPAQYEVZWMP
|
7.4 | IC50 | 2 | — | |
GPVFWBNYDOWIIQ
|
7.4 | Ki | 2 | — | |
HJJSEANNATVFNW
|
7.4 | IC50 | 4 | — | |
KRIUNPBAQZGFQA
|
7.4 | IC50 | 76 | — | |
SXBYKNSSEVQWPL
|
7.4 | Ki | 4 | — | |
USOOZXUJZKQXCC
|
7.4 | IC50 | 3 | — | |
WYBGYJNIKOAPQI
|
7.4 | Ki | 4 | — | |
YEHCNYAQEBQCCS
|
7.4 | Ki | 74 | — | |
SZBUKBINUVLFEL
|
7.4 | IC50 | 3 | Yes | |
XCGZBGKVXSQTFT
|
7.4 | IC50 | 3 | Yes | |
ZCCPLJOKGAACRT
|
7.4 | Kd | 599 | — | |
BUCXDWXDBZUFMV
|
7.4 | IC50 | 3 | Yes | |
JCKBTQZTGPJTII
|
7.4 | IC50 | 3 | Yes | |
UNUTTXCETMYXRD
|
7.4 | IC50 | 3 | Yes | |
MYLVKAPPYVXQKQ
|
7.4 | IC50 | 3 | Yes | |
FKBQOEJUXLTCGJ
|
7.4 | IC50 | 3 | — | |
ILTRIOQDZUXVFP
|
7.4 | IC50 | 2 | — | |
YHJXRSXZOCDBEA
|
7.4 | IC50 | 3 | — | |
RJVBVUWFYMRHRI
|
7.3 | IC50 | 4 | Yes | |
JDOKMDILBRSOLL
|
7.3 | IC50 | 3 | Yes | |
NGFCRLVABQTLPT
|
7.3 | IC50 | 3 | Yes | |
VQAHFLPDFJAHTG
|
7.3 | IC50 | 2 | Yes | |
JOAJAXWKPSMMPG
|
7.3 | IC50 | 2 | — | |
KUPWEENZVLBVNM
|
7.3 | IC50 | 3 | Yes | |
NHHQJBCNYHBUSI
|
7.3 | Kd | 220 | — | |
GKDIRDHQIHCEGG
|
7.3 | IC50 | 3 | — | |
HSKWNXWRIGSISU
|
7.3 | IC50 | 2 | — | |
VFDMQZQCLWTEJN
|
7.3 | IC50 | 3 | Yes | |
FGWOKLCRQJXPPQ
|
7.3 | Ki | 14 | — | |
GLVDZCDUMFNCFY
|
7.3 | IC50 | 3 | Yes | |
LZXLRJRSBFKIPI
|
7.3 | IC50 | 2 | — | |
OTQSCDWPCPZRIU
|
7.3 | Ki | 4 | — | |
PTSWSUSIGQQZOO
|
7.3 | Ki | 5 | — | |
STJJPAKEFZQZGB
|
7.3 | IC50 | 3 | — |