Target Details
| UniProt AC | P45984 |
|---|---|
| Gene Symbol | MAPK9 |
| Protein Name | Mitogen-activated protein kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 676
- Clinical molecules 191
- Avg pChEMBL 6.96
KEGG Pathways (75)
- AGE-RAGE signaling pathway in diabetic complications
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Colorectal cancer
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- ErbB signaling pathway
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Huntington disease
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- Pancreatic cancer
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Protein processing in endoplasmic reticulum
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tight junction
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Type II diabetes mellitus
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Active Molecules (676)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QWBLRTCRXZETHI
|
8.1 | IC50 | 5 | — | |
JSDUDTFXRSCOHV
|
8.1 | IC50 | 4 | Yes | |
KKKRKRMVJRHDMG
|
8.1 | Kd | 14 | — | |
UIRLFLOVKAOFEX
|
8.1 | Ki | 3 | Yes | |
ZOUZXNPDTXVSEH
|
8.1 | IC50 | 3 | Yes | |
KBJSPAOJLUYMQM
|
8.0 | IC50 | 3 | Yes | |
NKUVBRQPLJOWBI
|
8.0 | IC50 | 3 | Yes | |
YEBFCGFMUQJOCV
|
8.0 | IC50 | 3 | Yes | |
YVQKIQSJMFGJEG
|
8.0 | IC50 | 4 | Yes | |
JPSDPJFIFFHAFG
|
8.0 | IC50 | 2 | — | |
MLIRIWBFADTRLZ
|
8.0 | IC50 | 4 | Yes | |
TUZYUHMHEXTLNB
|
8.0 | IC50 | 2 | — | |
XLLHFYYRDKVYSQ
|
8.0 | IC50 | 3 | — | |
BZKOXELLQJFKSQ
|
7.9 | IC50 | 3 | Yes | |
DESXXRVFAOVNTC
|
7.9 | IC50 | 3 | — | |
QJPUIIKZKMYPSK
|
7.9 | IC50 | 3 | — | |
QJPUIIKZKMYPSK
|
7.9 | IC50 | 3 | — | |
SGYOIXNBCYRZBZ
|
7.9 | IC50 | 4 | — | |
KZSUQTFUAGZIRM
|
7.9 | IC50 | 5 | — | |
NFMGZVPRGVERNN
|
7.9 | Ki | 44 | — | |
UCOWZARZLHNDKP
|
7.9 | Ki | 8 | — | |
IRUBRQUHIORGIW
|
7.9 | IC50 | 2 | — | |
JUKUQWGWZSESAV
|
7.9 | Ki | 3 | Yes | |
RDFFZPKZBXFQEF
|
7.9 | IC50 | 3 | Yes | |
SGYOIXNBCYRZBZ
|
7.9 | IC50 | 4 | — | |
KXNZPASCSDMHFQ
|
7.8 | IC50 | 5 | Yes | |
LRVSISWQSCNQKL
|
7.8 | IC50 | 3 | Yes | |
OATHVDKMFZZHHN
|
7.8 | Kd | 9 | — | |
QWBLRTCRXZETHI
|
7.8 | IC50 | 4 | — | |
FVONQZQMUHLATI
|
7.8 | IC50 | 2 | — | |
TXUPRVNNKMSBLZ
|
7.8 | IC50 | 3 | Yes | |
YTPKEJXVUUNXRA
|
7.8 | IC50 | 4 | Yes | |
KDAMBQMCWSCLEM
|
7.8 | IC50 | 4 | — | |
DVEYHFXOGUYFBU
|
7.8 | Kd | 5 | — | |
FLEAYYMORDPWAJ
|
7.8 | Ki | 90 | — | |
JYYLVUFNAHSSFE
|
7.8 | Kd | 9 | — | |
SYLXLRJHNPOSFK
|
7.8 | IC50 | 2 | — | |
VLEFVPMCVJDTHZ
|
7.8 | Ki | 13 | — | |
VSVFDMDYNXAZHL
|
7.8 | IC50 | 4 | — | |
MKHLHLAXBRMALM
|
7.8 | IC50 | 5 | — | |
FILBHLMAZQOSRM
|
7.8 | IC50 | 2 | — | |
IRABIGXKJCMNIG
|
7.8 | IC50 | 3 | Yes | |
JCJAEEODSKNKTC
|
7.8 | IC50 | 6 | Yes | |
SCIILXOOXBQBFM
|
7.8 | Ki | 3 | Yes | |
SSWFFPALFQMQLE
|
7.8 | IC50 | 3 | — | |
VPSYCQPUUYBBBQ
|
7.8 | IC50 | 2 | — | |
BLWZIEOGNLHMEX
|
7.7 | IC50 | 2 | — | |
PTVSTQCTVOIQBP
|
7.7 | IC50 | 3 | — | |
ZZGXJNUHZVCAOW
|
7.7 | IC50 | 3 | Yes | |
GJFCSAPFHAXMSF
|
7.7 | IC50 | 3 | — |