Target Details
| UniProt AC | P45984 |
|---|---|
| Gene Symbol | MAPK9 |
| Protein Name | Mitogen-activated protein kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 676
- Clinical molecules 191
- Avg pChEMBL 6.96
KEGG Pathways (75)
- AGE-RAGE signaling pathway in diabetic complications
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Colorectal cancer
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- ErbB signaling pathway
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Huntington disease
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- Pancreatic cancer
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Protein processing in endoplasmic reticulum
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tight junction
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Type II diabetes mellitus
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Active Molecules (676)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RHFIAUKMKYHHFA
|
6.3 | IC50 | 9 | — | |
HZTYDQRUAWIZRE
|
6.3 | Kd | 40 | Yes | |
NDFIMKGGYOQCBV
|
6.3 | IC50 | 2 | Yes | |
ZNDOZPHFIVKNGZ
|
6.3 | IC50 | 2 | Yes | |
BKUSJXDWGAHZNA
|
6.3 | IC50 | 2 | — | |
QRCYLXLFEDYBSA
|
6.3 | IC50 | 2 | — | |
OBJNFLYHUXWUPF
|
6.3 | IC50 | 17 | — | |
WWFURUYYQWIHRV
|
6.3 | IC50 | 2 | — | |
QUBFVDVWHOIYRD
|
6.2 | IC50 | 2 | — | |
GBKQNVNYZATRQE
|
6.2 | IC50 | 2 | Yes | |
UPOMRTKHZCWMBW
|
6.2 | IC50 | 2 | — | |
ATESPULSOFFUAV
|
6.2 | IC50 | 2 | — | |
BNSPEWBMGVWZFC
|
6.2 | IC50 | 7 | — | |
JTBGYUCLPOTIMW
|
6.2 | IC50 | 2 | — | |
NERJSNYOGGKVRR
|
6.2 | IC50 | 3 | — | |
RVPVTOKNUYGICG
|
6.2 | IC50 | 2 | Yes | |
BTRNKAGATHKDRE
|
6.2 | IC50 | 3 | Yes | |
CLCSSDBGIADDIH
|
6.2 | IC50 | 2 | — | |
IOBZIJYYPWNRQU
|
6.2 | IC50 | 3 | Yes | |
ZJEWMDXOXBQHAB
|
6.2 | IC50 | 2 | — | |
HDRLAVNNWSHSOA
|
6.2 | Ki | 19 | — | |
MCCCQFAOMZMZKE
|
6.2 | Ki | 52 | — | |
MCKPYPWHBUXLEZ
|
6.2 | Ki | 21 | — | |
MNEXDVSJIUQQRH
|
6.2 | IC50 | 6 | — | |
MQRDVGBWWVWMEN
|
6.2 | Ki | 47 | — | |
QXKKPVVOOWBLND
|
6.2 | Ki | 8 | — | |
UUWNXFJBBYAMDT
|
6.2 | Ki | 46 | — | |
WHVFDYQCAMPLMS
|
6.2 | Ki | 20 | Yes | |
ZQUSFAUAYSEREK
|
6.2 | Ki | 7 | — | |
BBPWMHYCJRYYFV
|
6.2 | IC50 | 2 | — | |
LYADGAGFYYXXIO
|
6.2 | IC50 | 82 | — | |
NDINXVZGAZZFMK
|
6.2 | IC50 | 2 | — | |
NIWQPPGSGWOACD
|
6.2 | IC50 | 2 | — | |
OPLYAGXSXQZTGM
|
6.2 | IC50 | 2 | — | |
XLVWDHAXEFKTIB
|
6.2 | IC50 | 2 | — | |
ZYTDQGRQFPNBGA
|
6.2 | IC50 | 2 | — | |
FAUFFPCPZRRZKT
|
6.2 | IC50 | 2 | — | |
ZKESOLNZMJUNTF
|
6.2 | IC50 | 2 | — | |
CWJLAVRXVFHDSJ
|
6.2 | IC50 | 13 | — | |
CXQHYVUVSFXTMY
|
6.2 | Kd | 154 | — | |
QICPQLFMWYQJGX
|
6.2 | IC50 | 5 | — | |
SEJGTFPOEJWEGG
|
6.2 | Kd | 149 | — | |
WXXPHDFRDIYFEP
|
6.2 | IC50 | 2 | — | |
FEQRWFABERLIOV
|
6.2 | IC50 | 3 | — | |
GLLVHHZWPVUNED
|
6.2 | IC50 | 2 | — | |
OHRMONDIKHEVCZ
|
6.2 | IC50 | 2 | — | |
USORQDCKXRFILP
|
6.2 | IC50 | 2 | — | |
MGGUVSLBKUKUGR
|
6.2 | IC50 | 3 | Yes | |
NINIJRDUJSFATI
|
6.2 | IC50 | 3 | Yes | |
SLMJDPXFWRYMLU
|
6.2 | IC50 | 3 | — |