Target Details
| UniProt AC | P45984 |
|---|---|
| Gene Symbol | MAPK9 |
| Protein Name | Mitogen-activated protein kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 676
- Clinical molecules 191
- Avg pChEMBL 6.96
KEGG Pathways (75)
- AGE-RAGE signaling pathway in diabetic complications
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Colorectal cancer
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- ErbB signaling pathway
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Huntington disease
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- Pancreatic cancer
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Protein processing in endoplasmic reticulum
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tight junction
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Type II diabetes mellitus
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Active Molecules (676)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YVLVTFFRFJLZON
|
6.4 | IC50 | 2 | — | |
AEYLJTAIDDIOBA
|
6.4 | Ki | 53 | — | |
BSFNGHCTZDCQBF
|
6.4 | Ki | 93 | — | |
HHSVICUMCOBRPT
|
6.4 | Ki | 33 | — | |
IFPPYSWJNWHOLQ
|
6.4 | Ki | 52 | Yes | |
JNXJKTXDSPWNRP
|
6.4 | Ki | 30 | — | |
KTJOPUTZKZLREI
|
6.4 | IC50 | 2 | — | |
OWFLADWRSCINST
|
6.4 | Ki | 30 | — | |
SPYHMOFSJGTUNP
|
6.4 | Ki | 9 | — | |
WVFWTUJEHMVUBG
|
6.4 | Ki | 25 | — | |
WYOMXSAYYXBPMN
|
6.4 | Ki | 24 | — | |
YMSZHISTTIUBDG
|
6.4 | Ki | 7 | — | |
ZGDYBJXDIXVTLV
|
6.4 | Ki | 54 | — | |
ZPXPEKQMLOAPLT
|
6.4 | Ki | 15 | — | |
YKQSOUXCRZONQQ
|
6.4 | IC50 | 3 | Yes | |
RDCWVMUIPUMVKS
|
6.4 | IC50 | 2 | — | |
TUFAYPAXFHVGTH
|
6.4 | IC50 | 3 | — | |
AMAYXMZTQTYOQN
|
6.4 | IC50 | 2 | — | |
OYICHVOOWWQYDE
|
6.4 | IC50 | 2 | — | |
QIQWHUHEIKULHZ
|
6.4 | IC50 | 2 | Yes | |
DXAJWOOLPAIVJG
|
6.4 | Ki | 3 | Yes | |
INUQHONAOUHTRF
|
6.4 | IC50 | 4 | — | |
LTKLQMAKAFTREX
|
6.4 | IC50 | 2 | Yes | |
PBXFZPKEBIEGOE
|
6.4 | IC50 | 3 | — | |
RYCUVZMYBSSMAE
|
6.4 | IC50 | 2 | — | |
UJBJWYNPUOLFIZ
|
6.4 | IC50 | 49 | — | |
KSOFLDHKAGJBFC
|
6.3 | IC50 | 2 | — | |
PKNYJVSQHRVGTB
|
6.3 | IC50 | 2 | — | |
PXJCEFGMIBFUGI
|
6.3 | IC50 | 3 | — | |
QICPQLFMWYQJGX
|
6.3 | IC50 | 5 | — | |
BGGSTZPBQKGLOJ
|
6.3 | IC50 | 3 | Yes | |
HHCBMISMPSAZBF
|
6.3 | IC50 | 23 | — | |
IEZJTLFFNLOEKV
|
6.3 | IC50 | 3 | — | |
ZKMRRJOUWKSONY
|
6.3 | IC50 | 2 | — | |
ZRSKGCIFXQCBBO
|
6.3 | IC50 | 2 | Yes | |
WVXNSAVVKYZVOE
|
6.3 | IC50 | 92 | — | |
NLNVCPSZHKGGDI
|
6.3 | Ki | 2 | — | |
OTVCFDOYUHREFJ
|
6.3 | Ki | 26 | — | |
PCQMERRARZKTPW
|
6.3 | Ki | 68 | — | |
PROLIXHVRCJEFH
|
6.3 | Ki | 46 | — | |
QVMKLKBODZHJDK
|
6.3 | IC50 | 2 | — | |
RKUKAACYUCUJEE
|
6.3 | Ki | 58 | — | |
SFDUUFDVJHFBRB
|
6.3 | IC50 | 4 | — | |
ULSIWAGDPRIVCH
|
6.3 | Ki | 3 | — | |
UPYHVTCMTMZKAX
|
6.3 | Ki | 12 | — | |
ZFBBVSHFSXNGFK
|
6.3 | Ki | 2 | — | |
ZJWZDMQTDMVQQB
|
6.3 | IC50 | 3 | — | |
CYWPFAFZKKJPFQ
|
6.3 | IC50 | 2 | — | |
JTBIKPSVKQZGLW
|
6.3 | IC50 | 3 | Yes | |
LOLPPWBBNUVNQZ
|
6.3 | Kd | 97 | Yes |