Target Details
| UniProt AC | P45984 |
|---|---|
| Gene Symbol | MAPK9 |
| Protein Name | Mitogen-activated protein kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 676
- Clinical molecules 191
- Avg pChEMBL 6.96
KEGG Pathways (75)
- AGE-RAGE signaling pathway in diabetic complications
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Alzheimer disease
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Cadherin signaling
- Chagas disease
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Colorectal cancer
- Coronavirus disease - COVID-19
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Endocrine resistance
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- ErbB signaling pathway
- Fc epsilon RI signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- FoxO signaling pathway
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Huntington disease
- IL-17 signaling pathway
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- Insulin signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- Osteoclast differentiation
- Pancreatic cancer
- Parkinson disease
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Pertussis
- Prion disease
- Progesterone-mediated oocyte maturation
- Prolactin signaling pathway
- Protein processing in endoplasmic reticulum
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Relaxin signaling pathway
- Retrograde endocannabinoid signaling
- Salmonella infection
- Shigellosis
- Sphingolipid signaling pathway
- Spinocerebellar ataxia
- T cell receptor signaling pathway
- TNF signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tight junction
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Type II diabetes mellitus
- Wnt signaling pathway
- Yersinia infection
- cAMP signaling pathway
Active Molecules (676)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KFIDJSXUJCJHQB
|
6.5 | IC50 | 6 | — | |
PTPMBQNCXYRTGN
|
6.5 | IC50 | 5 | — | |
CEFDHULRYUTNDO
|
6.5 | IC50 | 2 | Yes | |
DOJMTDCTCJKZNL
|
6.5 | IC50 | 2 | — | |
KGMVZSJAPXYTKH
|
6.5 | IC50 | 23 | — | |
MMMOSWYLESPINL
|
6.5 | IC50 | 2 | Yes | |
PRFQGCBPEYPZAY
|
6.5 | IC50 | 3 | — | |
YGGYBJSDWZSAAU
|
6.5 | IC50 | 5 | — | |
JIVYDIADMNEKCM
|
6.5 | IC50 | 2 | — | |
LNMRSSIMGCDUTP
|
6.5 | Kd | 13 | — | |
XDNOBDTYZKRSTK
|
6.5 | IC50 | 2 | — | |
GQLWKGVBOIYMTN
|
6.5 | Ki | 35 | — | |
IOBVCHJTLVPPBR
|
6.5 | Ki | 39 | — | |
JBRASADWXDKCLJ
|
6.5 | Ki | 22 | — | |
JPTYCOMKVYISJL
|
6.5 | IC50 | 2 | Yes | |
KTBZRPANEUUZDW
|
6.5 | IC50 | 2 | — | |
KUVNSIJSYBSMJX
|
6.5 | Ki | 5 | — | |
LGHBDVLAHHANMX
|
6.5 | Ki | 53 | — | |
LHLBQSAMDHYBJT
|
6.5 | Ki | 3 | — | |
MXJAKLUXZXAYIC
|
6.5 | IC50 | 2 | — | |
OFGKHGRQQKNHAV
|
6.5 | Ki | 5 | — | |
PAMZHNHIZCTSRT
|
6.5 | Ki | 4 | — | |
UIARLYUEJFELEN
|
6.5 | Kd | 289 | Yes | |
WQGDQGAFSDMBLA
|
6.5 | IC50 | 2 | — | |
XJJYJNMNYDNXNO
|
6.5 | Ki | 23 | — | |
YNJWXJNPKHJFBE
|
6.5 | Ki | 2 | — | |
CDHZIFBQYVOWNY
|
6.5 | IC50 | 3 | — | |
MBZXMVKLFZXZRB
|
6.5 | IC50 | 4 | — | |
OFVMIXKKOOXFCD
|
6.5 | IC50 | 2 | Yes | |
XDJCLCLBSGGNKS
|
6.5 | Kd | 21 | — | |
ZYPRSWQPKLBUQM
|
6.5 | IC50 | 3 | Yes | |
BDHQTRQDQKVEIM
|
6.5 | IC50 | 3 | Yes | |
DPTBYUQHDCZBPL
|
6.5 | IC50 | 2 | — | |
MKUCYQPSROSPGD
|
6.5 | IC50 | 4 | Yes | |
XMMMRYGZMVXRBI
|
6.5 | IC50 | 2 | — | |
GTRPPGMPULGRCP
|
6.5 | IC50 | 3 | — | |
DKZYXHCYPUVGAF
|
6.4 | Kd | 112 | — | |
DXTHSIZXMXMTFL
|
6.4 | IC50 | 2 | — | |
LYMPHEWUZFSXGM
|
6.4 | IC50 | 2 | Yes | |
OCGXTBFQADYTFI
|
6.4 | IC50 | 2 | — | |
SPBVUOILOVHJPD
|
6.4 | IC50 | 3 | — | |
SZHHSFHOIDCNLD
|
6.4 | Kd | 6 | — | |
SZHHSFHOIDCNLD
|
6.4 | Kd | 3 | — | |
XURAVYGNAAUXQP
|
6.4 | Kd | 3 | — | |
XLSYZSRXVVCHLS
|
6.4 | Kd | 48 | — | |
XRHSVYXJHZMCCY
|
6.4 | IC50 | 3 | Yes | |
AQGSJPJSRCAJNS
|
6.4 | IC50 | 2 | — | |
UXBBRWNEXINJRZ
|
6.4 | IC50 | 3 | — | |
GUFXTCNPJGZWOZ
|
6.4 | IC50 | 3 | Yes | |
UCPDQFHGSDFSKX
|
6.4 | IC50 | 2 | Yes |