Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LSURBVCXYPJWOW
|
8.7 | IC50 | 3 | Yes | |
SJJAJPMVTRAZSX
|
8.7 | IC50 | 5 | Yes | |
UUVAUHUMINHXNV
|
8.7 | IC50 | 2 | — | |
CRPDTHYTIJXWLZ
|
8.7 | IC50 | 7 | Yes | |
IRPQGYYABIPNQJ
|
8.7 | IC50 | 3 | Yes | |
JCCRVIZMNYULMQ
|
8.7 | IC50 | 6 | Yes | |
JZZAWBZYLOHRQP
|
8.7 | IC50 | 2 | — | |
MRZSOAZZNSUPLS
|
8.7 | IC50 | 3 | — | |
MRZSOAZZNSUPLS
|
8.7 | IC50 | 5 | Yes | |
QKYPFBUZQDJQHX
|
8.7 | IC50 | 5 | Yes | |
SOPBVJMMDDZVHQ
|
8.7 | IC50 | 3 | — | |
SYYRIPAKWJBIOW
|
8.7 | IC50 | 8 | Yes | |
BLCLPMFYNMXITO
|
8.7 | IC50 | 5 | Yes | |
CWVWYGJTCDBSIW
|
8.7 | IC50 | 6 | Yes | |
CXFQYPXLXLPGNM
|
8.7 | IC50 | 5 | Yes | |
DDHYHOSBNZTEDO
|
8.7 | IC50 | 5 | Yes | |
DUZIIVUARYJPTE
|
8.7 | IC50 | 4 | Yes | |
FMPSZEWYBZCYDN
|
8.7 | IC50 | 6 | Yes | |
FUPNXXAGJGHNFI
|
8.7 | IC50 | 3 | — | |
GMRJGTBNERTZIB
|
8.7 | IC50 | 5 | Yes | |
GNNAXEPAOIUDTH
|
8.7 | IC50 | 6 | Yes | |
HHLQXXSIVVEBOY
|
8.7 | IC50 | 5 | Yes | |
HJPPIRCRVNMSQH
|
8.7 | IC50 | 4 | — | |
HKQQBEWUPLWAAA
|
8.7 | IC50 | 5 | Yes | |
HUTRBECWDORHKF
|
8.7 | IC50 | 4 | Yes | |
HWRVCRDVLWYPOY
|
8.7 | IC50 | 6 | Yes | |
HYZDHISHDZBYBQ
|
8.7 | IC50 | 6 | Yes | |
IOUQKHPLPLPITI
|
8.7 | IC50 | 5 | Yes | |
JBVXKMHBLNDBBV
|
8.7 | IC50 | 6 | Yes | |
KLYIBVBIKFMTRO
|
8.7 | IC50 | 6 | Yes | |
LCQNQVIUMDNDJS
|
8.7 | IC50 | 6 | Yes | |
LKSVLIAQUIGTTF
|
8.7 | IC50 | 6 | Yes | |
NIUQIJFMBOIHLA
|
8.7 | IC50 | 6 | Yes | |
NLPICQLAIKGJBE
|
8.7 | IC50 | 5 | Yes | |
NPFGSGCFKYSLPI
|
8.7 | IC50 | 6 | Yes | |
NQPIHEUUYRAYII
|
8.7 | IC50 | 8 | Yes | |
NRCQPJPKKZDRND
|
8.7 | Ki | 6 | Yes | |
NVQGQIYFJRAZLX
|
8.7 | Ki | 6 | Yes | |
NXRASPQMAAGLPZ
|
8.7 | IC50 | 6 | Yes | |
NZSGHPOSLLMCJS
|
8.7 | IC50 | 6 | Yes | |
OCSMOTCMPXTDND
|
8.7 | IC50 | 14 | Yes | |
PAAGUAHWPSXIJP
|
8.7 | IC50 | 6 | Yes | |
PILJHIOYYOZKRU
|
8.7 | IC50 | 3 | — | |
PLYLMXDSDZFWLJ
|
8.7 | IC50 | 6 | Yes | |
QHERSXDLUJOMHD
|
8.7 | Ki | 5 | — | |
RMZUAMXVNUZHBB
|
8.7 | IC50 | 6 | Yes | |
TVRLHUWRJSTBAB
|
8.7 | IC50 | 6 | Yes | |
TZYCKWCFYXFTIR
|
8.7 | IC50 | 5 | Yes | |
UGLOKYALFGIDPP
|
8.7 | IC50 | 4 | Yes | |
UGMUJIKGJCCUOY
|
8.7 | IC50 | 6 | Yes |