Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CRWSSUTUNYHTON
|
8.8 | IC50 | 2 | — | |
DMIORTQLUPECMV
|
8.8 | IC50 | 3 | Yes | |
FCGHMWYAKRLIIN
|
8.8 | IC50 | 2 | Yes | |
HEKVSVDHQDDIEK
|
8.8 | IC50 | 2 | — | |
HKBXBBXQCDCNLR
|
8.8 | IC50 | 2 | — | |
JHSGRRNCQDDQBC
|
8.8 | IC50 | 9 | — | |
MHIFGXNSNUWQOT
|
8.8 | IC50 | 3 | Yes | |
MIMMUUIYLKITIG
|
8.8 | IC50 | 5 | Yes | |
NJZUERVIVLYZMO
|
8.8 | IC50 | 5 | — | |
OIBWGGKYJHWGPB
|
8.8 | IC50 | 5 | Yes | |
RIJMYCAFDDBRHW
|
8.8 | IC50 | 2 | — | |
SLNHKZUUBJBCKF
|
8.8 | IC50 | 3 | Yes | |
SYNSXJHFJAEBFU
|
8.8 | IC50 | 2 | — | |
UWPHCZNYIWQCKD
|
8.8 | IC50 | 5 | Yes | |
XXOLBMKULOJKQR
|
8.8 | IC50 | 7 | Yes | |
ZFYWVXBCKVCYOL
|
8.8 | IC50 | 7 | Yes | |
QBWALRVIJDSECI
|
8.8 | Ki | 5 | Yes | |
BBMXXNQSDJPWKT
|
8.8 | IC50 | 4 | — | |
BSHJFYSJFLAHQN
|
8.8 | IC50 | 6 | Yes | |
FGQTUBBIXYISNM
|
8.8 | IC50 | 4 | — | |
FTIYYJYCHWIXRZ
|
8.8 | IC50 | 4 | Yes | |
ILDOICSWRSOHSV
|
8.8 | IC50 | 3 | Yes | |
JSYMSOFUKLCCMS
|
8.8 | IC50 | 4 | Yes | |
RDMHVXDIUPIFCJ
|
8.8 | IC50 | 4 | — | |
UMEYNLZNXJZVAP
|
8.8 | Ki | 4 | Yes | |
VCIBNYPUVKINDS
|
8.8 | Ki | 5 | Yes | |
HGHQBSHHIZJUCO
|
8.8 | IC50 | 2 | — | |
IMLFQSRCUZAGNQ
|
8.8 | IC50 | 4 | Yes | |
IYMQHQXCXLDREF
|
8.8 | IC50 | 4 | Yes | |
MASDJPGVHCTFLM
|
8.8 | IC50 | 5 | Yes | |
OICBVOJTVMMIHN
|
8.8 | IC50 | 3 | Yes | |
SNMQJFHUOZBSDS
|
8.8 | Ki | 5 | — | |
UGEYJONPMBOKNN
|
8.8 | IC50 | 7 | Yes | |
ZRAUMSIZBNBIFE
|
8.8 | IC50 | 8 | Yes | |
IAENNQHKVZEBQT
|
8.8 | IC50 | 7 | Yes | |
JRPLACGAMSWTCU
|
8.8 | Ki | 5 | Yes | |
KWEXGQXQATXFLU
|
8.8 | IC50 | 3 | Yes | |
MUWDEQLPHWVPPA
|
8.8 | Ki | 5 | — | |
NDGWYSJFTMSGNY
|
8.8 | IC50 | 6 | Yes | |
RBXJTRGTMYPRKK
|
8.8 | IC50 | 3 | Yes | |
RBZQWZODGBMNHX
|
8.8 | Ki | 6 | Yes | |
SUEBJDNLBVTIQP
|
8.8 | IC50 | 8 | Yes | |
VDUBALDTEGAJSW
|
8.8 | Ki | 7 | Yes | |
XFIZGIIZTOASLY
|
8.8 | IC50 | 4 | Yes | |
YXSJVSGLVWXWOT
|
8.8 | IC50 | 4 | — | |
HJFONKSERLWIGE
|
8.8 | IC50 | 4 | Yes | |
HXAROWWJPCDNRW
|
8.7 | IC50 | 6 | Yes | |
ICFOTHUAZLHTNP
|
8.7 | IC50 | 7 | Yes | |
IFCFGMLOBSUCSN
|
8.7 | IC50 | 5 | Yes | |
KQIFSUSWYMDFOC
|
8.7 | IC50 | 5 | Yes |