Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VBPVZEMPZISXMF
|
9.0 | IC50 | 5 | Yes | |
VCKCQHDSLLCTDH
|
9.0 | IC50 | 6 | Yes | |
VCKIKUWRRCAZBI
|
9.0 | IC50 | 6 | Yes | |
WWVKBGIBCFSFOJ
|
9.0 | IC50 | 5 | Yes | |
WZTNVCMELDPHHH
|
9.0 | IC50 | 6 | Yes | |
XOVSRAFNJNQNRK
|
9.0 | IC50 | 4 | Yes | |
XQRSTZJAXGSSTI
|
9.0 | IC50 | 4 | Yes | |
XXCBSIYZQACPFC
|
9.0 | IC50 | 5 | Yes | |
YGXMCNARAMUPPX
|
9.0 | IC50 | 7 | Yes | |
YMQBLRHAACUVFH
|
9.0 | IC50 | 6 | Yes | |
YNSHKUPPIHHCNP
|
9.0 | IC50 | 6 | Yes | |
ZBDXZEGIXHCDMC
|
9.0 | IC50 | 5 | Yes | |
ZORDGSDKVXISJV
|
9.0 | IC50 | 6 | Yes | |
ZTJUBPXNBSLSGL
|
9.0 | IC50 | 6 | Yes | |
ZWHGUGYVAMXPJZ
|
9.0 | IC50 | 5 | Yes | |
ZZEIPXVXVCUKGA
|
9.0 | IC50 | 6 | Yes | |
DSBXKNRWNDALKK
|
9.0 | IC50 | 4 | Yes | |
JGTIIKHYSZFICL
|
9.0 | IC50 | 5 | Yes | |
LIBJLMBRYDKFLR
|
9.0 | IC50 | 2 | — | |
MMOBDSFVSOBMOV
|
9.0 | IC50 | 7 | Yes | |
PNVLBMRGQMDPBJ
|
9.0 | IC50 | 5 | Yes | |
PUHDBKGWNNZTBP
|
9.0 | IC50 | 8 | Yes | |
RVKPGECPCLBLDB
|
9.0 | IC50 | 10 | Yes | |
YEBHJCQWJHLMTP
|
9.0 | IC50 | 4 | Yes | |
CYZMUIMLRBJSRO
|
8.9 | IC50 | 4 | Yes | |
DZCGIZPIPKWUIX
|
8.9 | IC50 | 7 | Yes | |
DZVDZJSJBKHJOK
|
8.9 | IC50 | 5 | Yes | |
MRSUSKBPRPSZTK
|
8.9 | IC50 | 2 | — | |
NOCFVGZKPITVEY
|
8.9 | IC50 | 5 | Yes | |
NWYAUZLEGMZWIR
|
8.9 | IC50 | 2 | — | |
QVCXUWWKONKLBL
|
8.9 | Ki | 6 | Yes | |
SNWCXQPNOQQJPW
|
8.9 | IC50 | 4 | Yes | |
UAFRGDNTZQMZFA
|
8.9 | Ki | 5 | Yes | |
ZXORTEVXPYNWIB
|
8.9 | IC50 | 5 | Yes | |
ALKUUIDKRJZTBK
|
8.9 | IC50 | 2 | — | |
AHBFOOOWLVWQFO
|
8.9 | IC50 | 6 | Yes | |
AOPSFGSGYVNAEJ
|
8.9 | IC50 | 5 | Yes | |
BHBGOKVZFAQJAD
|
8.9 | IC50 | 5 | Yes | |
DNGGPLKVDUPXFN
|
8.9 | IC50 | 5 | — | |
DNGGPLKVDUPXFN
|
8.9 | IC50 | 7 | Yes | |
FUOOTOLTPDFGCS
|
8.9 | IC50 | 3 | Yes | |
REZSPXZZCJTZIK
|
8.9 | IC50 | 8 | Yes | |
URNPXFKEVDQWTO
|
8.9 | IC50 | 3 | Yes | |
VJHXJEDXSPNSEK
|
8.9 | IC50 | 3 | Yes | |
VUANPBMJTLCNSC
|
8.9 | IC50 | 6 | Yes | |
VXZXTODNXJFRKF
|
8.9 | IC50 | 3 | Yes | |
XSWDEIOVOAQSMZ
|
8.9 | IC50 | 7 | Yes | |
XVZWTHXPJUVJAU
|
8.9 | IC50 | 6 | Yes | |
YZIGEYGKVJNXSU
|
8.9 | IC50 | 3 | Yes | |
BGEFVHSKSARWDE
|
8.8 | IC50 | 3 | Yes |