Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AUWOIDNULNLPBA
|
9.0 | IC50 | 5 | Yes | |
AXTUTMYETKQSJS
|
9.0 | IC50 | 6 | Yes | |
BIHFHTLMZBLJAX
|
9.0 | IC50 | 4 | Yes | |
BLXHYKZAZZIQOC
|
9.0 | Ki | 3 | — | |
CAPSVCHNNRHIDK
|
9.0 | IC50 | 6 | Yes | |
CBKKHHSQVZVIBM
|
9.0 | IC50 | 6 | Yes | |
CBMKHOZXSARYNG
|
9.0 | IC50 | 6 | Yes | |
DHCMKRCHROJJHB
|
9.0 | IC50 | 3 | Yes | |
DTPBPOWGEIFZGM
|
9.0 | IC50 | 5 | Yes | |
FLIOXLIZONFFSH
|
9.0 | IC50 | 5 | Yes | |
FNURWSLLBXZLRC
|
9.0 | IC50 | 7 | Yes | |
FPSMXPGSVWPWCG
|
9.0 | IC50 | 8 | — | |
GKDAXRUOVHMLSA
|
9.0 | IC50 | 6 | Yes | |
GQEYBNSJJQDDLY
|
9.0 | IC50 | 5 | Yes | |
HGCZRPPCNXJXAB
|
9.0 | IC50 | 7 | Yes | |
HZELUBQHAZKZKC
|
9.0 | IC50 | 5 | Yes | |
IGDBRYFDPWPBAI
|
9.0 | IC50 | 3 | Yes | |
IIBGHLQTRXDEKI
|
9.0 | IC50 | 7 | Yes | |
IMKDKHQDFFLOKK
|
9.0 | IC50 | 13 | Yes | |
IVGHGMHNUBCTDC
|
9.0 | Ki | 6 | Yes | |
JDOCJRYXQAWUOO
|
9.0 | IC50 | 7 | Yes | |
JXMJSOSLBMBYGM
|
9.0 | IC50 | 4 | — | |
JZHHNBACJYFNCE
|
9.0 | IC50 | 4 | — | |
JZKQUJKQSKTEON
|
9.0 | IC50 | 6 | Yes | |
KLSLMSQYLRDFGN
|
9.0 | IC50 | 5 | Yes | |
KMLHPTCEMLILLL
|
9.0 | IC50 | 4 | Yes | |
KUEURUPTKRCKAQ
|
9.0 | IC50 | 6 | Yes | |
LTVIJEFEZVFIST
|
9.0 | IC50 | 14 | Yes | |
MKKSGKUWQUXKAQ
|
9.0 | IC50 | 6 | Yes | |
NAXMTMYDSBOGMZ
|
9.0 | IC50 | 5 | Yes | |
NVQUYHFBHXGQLL
|
9.0 | IC50 | 6 | Yes | |
NXCSXUBVRRHHLE
|
9.0 | IC50 | 4 | — | |
OLEYZXUQGOKVKT
|
9.0 | IC50 | 7 | Yes | |
OOCSYABQMHKMLM
|
9.0 | IC50 | 6 | Yes | |
OUPAYUKAUNZSER
|
9.0 | IC50 | 4 | Yes | |
PCSKPZLQCNGMCY
|
9.0 | IC50 | 6 | Yes | |
PECBDMOWKLTTSB
|
9.0 | IC50 | 4 | — | |
PQPJWKCPMXIWMW
|
9.0 | IC50 | 6 | Yes | |
QYZPDCGWIJYZMN
|
9.0 | IC50 | 8 | Yes | |
RAOAFDPXSFVLJD
|
9.0 | IC50 | 6 | Yes | |
RYRSPABEKSPRKC
|
9.0 | IC50 | 7 | Yes | |
RZDQDYGREGZPAT
|
9.0 | IC50 | 5 | Yes | |
SESDSMKBCYCQSU
|
9.0 | IC50 | 6 | Yes | |
SKVZRQFKXKDXCW
|
9.0 | IC50 | 5 | Yes | |
SRPXVKQVZQEPFT
|
9.0 | IC50 | 5 | Yes | |
SSVAOOCBANMUMS
|
9.0 | IC50 | 5 | Yes | |
UIMOJSHBVUUXAE
|
9.0 | Ki | 3 | — | |
UKLIIGXGTPSYBF
|
9.0 | IC50 | 8 | Yes | |
ULILDPSFFUSXJH
|
9.0 | IC50 | 9 | Yes | |
ULILDPSFFUSXJH
|
9.0 | IC50 | 7 | — |