Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QRDYOYPORKWZCP
|
9.2 | IC50 | 6 | Yes | |
QYFKTMNLZHLRIH
|
9.2 | IC50 | 7 | Yes | |
REJAGHRLIZEVSB
|
9.2 | IC50 | 5 | Yes | |
ULDXUWXTVRRUND
|
9.2 | IC50 | 5 | Yes | |
VPDOXKSDXTZFIX
|
9.2 | IC50 | 4 | — | |
WGVFUINCAVSVGT
|
9.2 | IC50 | 6 | Yes | |
YBTXAIOMVIXCOD
|
9.2 | IC50 | 5 | Yes | |
YUFOYANNKICWEX
|
9.2 | IC50 | 4 | Yes | |
SQQHSADBIVCBBM
|
9.1 | IC50 | 4 | Yes | |
ZBRHTUMWSDPCMI
|
9.1 | IC50 | 10 | Yes | |
YZIGEYGKVJNXSU
|
9.1 | IC50 | 4 | Yes | |
BTZXQMHZPVTFBL
|
9.1 | IC50 | 7 | Yes | |
CPBPQYOAJUZJNL
|
9.1 | IC50 | 7 | Yes | |
DZVJLUYVLJYLGY
|
9.1 | IC50 | 5 | Yes | |
JQESDCUCXWEIBZ
|
9.1 | Ki | 2 | — | |
JWKIHGMBZXIUII
|
9.1 | IC50 | 3 | Yes | |
KXEGEKRSCUZQMH
|
9.1 | IC50 | 5 | Yes | |
LOZYBBRAEOAORI
|
9.1 | IC50 | 5 | Yes | |
PECNGMJVFOGIBW
|
9.1 | IC50 | 7 | Yes | |
PUBARVPHTAEUJQ
|
9.1 | IC50 | 5 | Yes | |
RDFQXFRQTOWZEQ
|
9.1 | IC50 | 8 | Yes | |
SEFFUKHXSNXXNA
|
9.1 | IC50 | 2 | — | |
VFDSDRZNXLFCFF
|
9.1 | IC50 | 7 | Yes | |
XSMMFHYHIAOGPC
|
9.1 | IC50 | 5 | Yes | |
YYZDREAOBMTNAP
|
9.1 | IC50 | 6 | Yes | |
ZBOSPOSQGJWURE
|
9.1 | Ki | 5 | — | |
BIHFFXMAAJBXAB
|
9.1 | IC50 | 2 | — | |
BIHSFSZDPRDVEE
|
9.1 | IC50 | 3 | Yes | |
CIECVEXIXKIUIZ
|
9.1 | IC50 | 4 | Yes | |
PLCRCZGBQOTIFV
|
9.1 | IC50 | 3 | Yes | |
RQCXYESMODRPPY
|
9.1 | IC50 | 4 | Yes | |
BUEVFADAMKTXGD
|
9.1 | IC50 | 5 | Yes | |
CYYCSKFJEOSZTF
|
9.1 | IC50 | 9 | Yes | |
DLMROZSTEBHAOO
|
9.1 | IC50 | 4 | Yes | |
FMYMFUHWQBEETO
|
9.1 | IC50 | 5 | Yes | |
HDBHDPIRGZHXCM
|
9.1 | IC50 | 4 | Yes | |
HPIJZAVGIHKGTA
|
9.1 | IC50 | 4 | Yes | |
KMXAXPCBRVZOGA
|
9.1 | IC50 | 7 | — | |
KXZZWRQJKQVMKR
|
9.1 | IC50 | 7 | Yes | |
QCOQJYRPDUMCNP
|
9.1 | IC50 | 5 | Yes | |
SBIQGLZKCCTUIC
|
9.1 | IC50 | 4 | Yes | |
SJTWWQWUAQAYAB
|
9.1 | IC50 | 4 | Yes | |
MEDAEECOIUAMSO
|
9.0 | IC50 | 4 | Yes | |
OCDVFODZPZVZMF
|
9.0 | IC50 | 4 | Yes | |
FKICHBNUXJBKPB
|
9.0 | Ki | 5 | Yes | |
FRIYTZJGYCAFHL
|
9.0 | IC50 | 3 | Yes | |
WJULIBHPWZXMJA
|
9.0 | IC50 | 10 | Yes | |
CMENTMLKKMZGPM
|
9.0 | IC50 | 4 | Yes | |
AKNDZTHCJLFZCF
|
9.0 | IC50 | 9 | Yes | |
ATFPFLNWBZIBTJ
|
9.0 | IC50 | 6 | Yes |