Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PTGMPWHDIULCAR
|
9.3 | IC50 | 6 | Yes | |
REZSPXZZCJTZIK
|
9.3 | IC50 | 6 | — | |
TUYLXABAVZEOSZ
|
9.3 | IC50 | 4 | — | |
TZQQXIZDSZWWPC
|
9.3 | IC50 | 6 | Yes | |
WFVYENBQHIIIQE
|
9.3 | IC50 | 7 | Yes | |
XFBRPTYLOIFAQR
|
9.3 | IC50 | 8 | Yes | |
XJMLKUIRAXOATH
|
9.3 | IC50 | 7 | Yes | |
XKUVMLDMSDMUFF
|
9.3 | IC50 | 3 | — | |
ROSNVSQTEGHUKU
|
9.3 | IC50 | 12 | Yes | |
SHSBTGZNXOPCNV
|
9.3 | IC50 | 4 | Yes | |
RLDSXGKXSYXTOQ
|
9.3 | IC50 | 3 | Yes | |
PRJCFROAJDAXAD
|
9.3 | Ki | 8 | Yes | |
IEJULHWWGPPJNO
|
9.2 | IC50 | 4 | Yes | |
UJKKQEHHLXCTJE
|
9.2 | IC50 | 6 | — | |
MFNVPUYZKNRAKT
|
9.2 | IC50 | 4 | — | |
SPBFQBQZZSCDQE
|
9.2 | Ki | 2 | — | |
ADDYZQRMSCIHFH
|
9.2 | IC50 | 4 | — | |
DLLCDWXNWWRIFJ
|
9.2 | IC50 | 4 | Yes | |
HYJOVEQOBWVFPG
|
9.2 | IC50 | 5 | Yes | |
ITDDXQSXMTUIFM
|
9.2 | IC50 | 7 | Yes | |
JKRVXAWKSWVVCV
|
9.2 | IC50 | 7 | Yes | |
KLWUGXOQJJWEBZ
|
9.2 | Ki | 5 | — | |
LIQFLIXIOKMDTJ
|
9.2 | Ki | 7 | Yes | |
LMIHEFSBOIGKDH
|
9.2 | IC50 | 8 | Yes | |
OOUAVDQEGOBVOR
|
9.2 | IC50 | 3 | Yes | |
OXLIYFANWBIKMH
|
9.2 | IC50 | 3 | Yes | |
PDYICDUZWJCQQF
|
9.2 | IC50 | 4 | — | |
QURZZKPWFKUXBF
|
9.2 | IC50 | 5 | Yes | |
UFKFLDDRYBWLPH
|
9.2 | IC50 | 5 | Yes | |
XRSYNYGEEYTXJV
|
9.2 | IC50 | 2 | — | |
TUUOOTOFTLPOMW
|
9.2 | IC50 | 3 | Yes | |
YHEMJEYZYLVDRO
|
9.2 | IC50 | 3 | Yes | |
BTMSEVQRJBBBAY
|
9.2 | IC50 | 3 | — | |
OGAPQRGMHIGAGP
|
9.2 | IC50 | 4 | Yes | |
SOOSDOUTIZJYOW
|
9.2 | IC50 | 4 | Yes | |
SOOSDOUTIZJYOW
|
9.2 | IC50 | 2 | — | |
BNPWNBBKUMLEJM
|
9.2 | Ki | 5 | Yes | |
JNMYIRAUFFFDQS
|
9.2 | IC50 | 4 | Yes | |
MMCUCOOPEAHRPL
|
9.2 | Ki | 6 | Yes | |
NKHJMAWHLPBSOA
|
9.2 | Ki | 5 | — | |
QHHHTEGVVKPDKH
|
9.2 | IC50 | 6 | — | |
PSLRKUXEVFQKIV
|
9.2 | IC50 | 2 | — | |
BSGLIFPGYIIUAJ
|
9.2 | IC50 | 7 | Yes | |
FNEPKOHTWFANAW
|
9.2 | IC50 | 4 | Yes | |
HMXFQXRHTFBPFX
|
9.2 | IC50 | 4 | — | |
LFOGEPKUSWRLCL
|
9.2 | IC50 | 7 | Yes | |
LGVIBWRSRHZDQG
|
9.2 | IC50 | 6 | Yes | |
LUCWASGSJPPQEE
|
9.2 | IC50 | 3 | — | |
OQWMKRBWGAJEGE
|
9.2 | IC50 | 4 | Yes | |
QCRPOQONCVCBFI
|
9.2 | IC50 | 4 | Yes |