Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UFJYSWCFYDZPKS
|
6.2 | IC50 | 4 | Yes | |
KDEHHSHGVKUYEZ
|
6.1 | IC50 | 3 | — | |
LKRHPZIUVGMVCY
|
6.1 | IC50 | 5 | Yes | |
WTWNYQALQSSSPL
|
6.1 | IC50 | 4 | Yes | |
BYQIIKCYPGKHOY
|
6.1 | Ki | 5 | Yes | |
DFRHCKHXGKQVLI
|
6.1 | IC50 | 3 | Yes | |
FUYXUEFCWRUMHG
|
6.1 | IC50 | 4 | — | |
GVUFJCREUUFMPP
|
6.1 | IC50 | 3 | Yes | |
JDBUKSMCZPXYJU
|
6.1 | IC50 | 4 | — | |
MBVFAXQWLSRZPW
|
6.1 | Ki | 2 | — | |
MCBALNMZVCCHAP
|
6.1 | Ki | 4 | Yes | |
QDMJDGKLXWJUSU
|
6.1 | Ki | 2 | — | |
HGILVKJBXAXGDH
|
6.1 | IC50 | 3 | Yes | |
VLNVWKDSFQRXHZ
|
6.1 | IC50 | 5 | Yes | |
GIEQMQWMJSYCKB
|
6.1 | Ki | 5 | — | |
IRVGVLJCCVMVAY
|
6.1 | IC50 | 5 | Yes | |
ZQFMPAUDTOJXIB
|
6.1 | Ki | 8 | Yes | |
AKWUAHDLDRSRDC
|
6.1 | IC50 | 6 | Yes | |
FHZGYMLWCVBBPM
|
6.1 | IC50 | 4 | Yes | |
JPIVNFSAQUANEQ
|
6.1 | IC50 | 2 | — | |
KVMYRTIGLLQRFY
|
6.1 | Ki | 4 | Yes | |
JFRAGUOIAHJTOM
|
6.1 | IC50 | 3 | Yes | |
JQJWNYAMOJOHCE
|
6.1 | IC50 | 4 | Yes | |
XQTUJUSPSCMEOC
|
6.1 | IC50 | 4 | Yes | |
RXFCFGLSOUOCEA
|
6.1 | IC50 | 4 | Yes | |
ILNPRELUGQHUMU
|
6.1 | IC50 | 3 | Yes | |
KXFPWCKTSXRQIS
|
6.1 | IC50 | 4 | — | |
JYGPMNNMAQCQMG
|
6.0 | Ki | 4 | — | |
RBRFAUFMZOIMMS
|
6.0 | IC50 | 2 | — | |
RBRFAUFMZOIMMS
|
6.0 | IC50 | 3 | — | |
RMDGEXDQWGEALM
|
6.0 | IC50 | 3 | Yes | |
WEJRAOYHTAOVFY
|
6.0 | Ki | 3 | Yes | |
XDKNQAWYSUZUDU
|
6.0 | IC50 | 3 | Yes | |
ZURDTDSRPUWYTO
|
6.0 | IC50 | 2 | — | |
JRSOKCXTAIQJPK
|
6.0 | IC50 | 4 | Yes | |
LBVBVIKJOWWVJX
|
6.0 | IC50 | 4 | — | |
NYSZVCQWENKRKM
|
6.0 | IC50 | 5 | Yes | |
UUDTVMMARAFNKG
|
6.0 | Ki | 4 | — | |
YMAXKJGQKQACFZ
|
6.0 | IC50 | 5 | Yes | |
KLUBFNJJJWONQA
|
6.0 | IC50 | 4 | Yes | |
LSGQQGGAWBOKIB
|
6.0 | IC50 | 4 | Yes | |
NWEMVUGYMZFTLT
|
6.0 | Ki | 2 | — | |
OOQSIBQKXZCHOC
|
6.0 | IC50 | 3 | — | |
KQTIZOWWQVTBNZ
|
6.0 | IC50 | 5 | Yes | |
QHEIMJONTDDZIV
|
6.0 | IC50 | 5 | — | |
QSVVRYPBRVSBDL
|
6.0 | IC50 | 2 | — | |
HPPQTJSDCSGPAX
|
6.0 | IC50 | 2 | — | |
RYUNWXPVOIGBCD
|
6.0 | IC50 | 4 | Yes | |
YTDQNSGULXQVKB
|
6.0 | IC50 | 3 | Yes |