Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PAXQYYVHPNBESJ
|
6.3 | IC50 | 4 | — | |
PWKVCJUBXCXPFI
|
6.3 | IC50 | 2 | — | |
QRWJUWNAJTZLAE
|
6.3 | IC50 | 5 | Yes | |
VKKROTIIKHOVOQ
|
6.3 | IC50 | 2 | — | |
ZQKXCFSWZGWAET
|
6.3 | IC50 | 3 | — | |
BLDFRIYOIZRRJI
|
6.2 | Ki | 4 | — | |
JMWVTDZGNUFBMO
|
6.2 | Ki | 4 | — | |
KEHDBOGRIVHUBV
|
6.2 | Ki | 6 | — | |
RUVHVYMIMBVNKN
|
6.2 | Ki | 5 | — | |
HECFJRXDSZZJLW
|
6.2 | IC50 | 3 | Yes | |
JAPLGNWCNXCEJT
|
6.2 | IC50 | 5 | Yes | |
JSZJOMOAWAHHBK
|
6.2 | IC50 | 3 | Yes | |
MYFWCGILTGDUAM
|
6.2 | Ki | 8 | Yes | |
UKLIIGXGTPSYBF
|
6.2 | IC50 | 4 | Yes | |
IHSDOJRAORURAS
|
6.2 | IC50 | 5 | Yes | |
QQGKYSPTORHWNZ
|
6.2 | Ki | 6 | — | |
AVFCHUYQSZAIFE
|
6.2 | Ki | 4 | — | |
GXINZIOTECAGST
|
6.2 | IC50 | 3 | Yes | |
KDDWLGBIYXTPJG
|
6.2 | Ki | 5 | — | |
LWNWGJXWKYGLPU
|
6.2 | IC50 | 5 | Yes | |
MRYXWLVKWYVRPC
|
6.2 | IC50 | 4 | Yes | |
QNVRWDPZVVAENF
|
6.2 | Ki | 4 | Yes | |
VWOQXPBXOWHZCH
|
6.2 | IC50 | 6 | Yes | |
YSRLIHTZJHEXLM
|
6.2 | IC50 | 2 | — | |
PDKBAEDNMKVROV
|
6.2 | Ki | 8 | Yes | |
ATLFNGKZSBVKHI
|
6.2 | IC50 | 3 | — | |
GOLLITFKIKKRMV
|
6.2 | Ki | 2 | — | |
KRVMUJILUZQWCW
|
6.2 | IC50 | 2 | — | |
QRQKVQCDKFEWSW
|
6.2 | IC50 | 4 | — | |
BRXGWWVUCIZYMM
|
6.2 | IC50 | 4 | — | |
BRXGWWVUCIZYMM
|
6.2 | IC50 | 5 | Yes | |
LEDMBBYIVRLZAS
|
6.2 | Ki | 9 | Yes | |
LYRSIRCJLISGFP
|
6.2 | IC50 | 4 | — | |
VHCRBJFCQRNNFG
|
6.2 | IC50 | 4 | Yes | |
VIPIKALUTUDDKU
|
6.2 | Ki | 2 | — | |
AENHIDVKFOYIJJ
|
6.2 | Ki | 4 | Yes | |
LLZNOGUPMFYFGU
|
6.2 | IC50 | 3 | — | |
PYSVMZGECWVLOT
|
6.2 | IC50 | 4 | Yes | |
RWKJBOMUESGCBO
|
6.2 | Ki | 4 | Yes | |
JIIMVBXHLBKVOM
|
6.2 | IC50 | 6 | Yes | |
RBTRVKIWYJFOJW
|
6.2 | IC50 | 2 | — | |
KGICPKKIUBLFER
|
6.2 | Ki | 4 | — | |
MMIHYNVQXYWTFM
|
6.2 | Ki | 4 | — | |
MMIHYNVQXYWTFM
|
6.2 | Ki | 4 | — | |
NVJUVGMOOGFJLZ
|
6.2 | Ki | 5 | Yes | |
QOWBVKQSFCSJAK
|
6.2 | IC50 | 5 | — | |
XJRRXPFUJFHHGA
|
6.2 | IC50 | 3 | — | |
YWXFICBFTYVHJU
|
6.2 | Ki | 4 | — | |
MKEVHBFZBURDHJ
|
6.2 | IC50 | 2 | — | |
NEOOWKPSCAQYPI
|
6.2 | IC50 | 4 | Yes |