Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YSYXAGMNRKARQB
|
6.4 | IC50 | 4 | Yes | |
BBERXYYXGJGELS
|
6.4 | Ki | 4 | — | |
CSVWGAZPMRHMHB
|
6.4 | IC50 | 5 | Yes | |
DVAPUVGZYOTZOY
|
6.4 | IC50 | 4 | Yes | |
HYCYFNRXRRBATO
|
6.4 | IC50 | 3 | — | |
SOPDPCOBVSOXIM
|
6.4 | Ki | 4 | Yes | |
VFEIVMVXXWQZER
|
6.4 | Ki | 2 | — | |
IADFBNIHFKDTRS
|
6.3 | Ki | 2 | — | |
IDHBZDJZPPEMGC
|
6.3 | IC50 | 4 | Yes | |
JNZCXNBTGUHDRZ
|
6.3 | IC50 | 3 | — | |
LKFNHCFYLDRUTH
|
6.3 | IC50 | 4 | Yes | |
WFKAOUORBBLUOE
|
6.3 | IC50 | 2 | — | |
DXRHJEFJSKWMEQ
|
6.3 | IC50 | 2 | — | |
ISAKGERLXJBHSA
|
6.3 | IC50 | 2 | — | |
MOQWSIABFGAXAW
|
6.3 | IC50 | 5 | — | |
OMZKWXAFDODBPH
|
6.3 | IC50 | 2 | — | |
QVNZBDLTUKCPGJ
|
6.3 | IC50 | 10 | — | |
WJUVUTHXZGHZOG
|
6.3 | IC50 | 2 | — | |
CQARAIRTGMAYMZ
|
6.3 | Ki | 8 | — | |
OAXXNDPRBWJXOJ
|
6.3 | IC50 | 4 | Yes | |
WJWOJAKOSRCFKB
|
6.3 | Ki | 9 | Yes | |
AGSXHHFUSDGSSO
|
6.3 | IC50 | 5 | Yes | |
DPNFTGXQMOIHKK
|
6.3 | IC50 | 3 | Yes | |
QFUKIOJKDCKUGI
|
6.3 | IC50 | 3 | Yes | |
QGVCPEQAAKTMNX
|
6.3 | IC50 | 3 | Yes | |
UUTDMYYQOAVOHN
|
6.3 | IC50 | 3 | Yes | |
QYMKPTMAFMKKTC
|
6.3 | IC50 | 5 | Yes | |
SIICAQVADMFEDB
|
6.3 | Ki | 8 | Yes | |
ADDJDJQFPKUMAF
|
6.3 | Ki | 7 | — | |
FIKHJLBGJKASJJ
|
6.3 | IC50 | 2 | — | |
FPJLTHNGOJRXMU
|
6.3 | Ki | 8 | Yes | |
MNAUWMOCDLCGGF
|
6.3 | IC50 | 2 | — | |
PGTJOSSSBWAALE
|
6.3 | Ki | 2 | — | |
SKLOAVPDSDQCQV
|
6.3 | IC50 | 2 | — | |
TXIMSNHHNJBLTN
|
6.3 | IC50 | 3 | Yes | |
ZDYXONOHFKVMSQ
|
6.3 | IC50 | 2 | — | |
LRRAUDSVXJEODP
|
6.3 | Ki | 6 | Yes | |
YUQQWAKBRAEWQZ
|
6.3 | Ki | 2 | — | |
BMPCLJPYXFVWKY
|
6.3 | IC50 | 5 | Yes | |
IXKRFERDVUXQLW
|
6.3 | IC50 | 6 | Yes | |
MUGAWCXYWNGHML
|
6.3 | Ki | 2 | — | |
PMSJHLLBCDOJAE
|
6.3 | IC50 | 5 | Yes | |
RGHANNJVNFHOMO
|
6.3 | IC50 | 3 | Yes | |
AEOWLQGPNGMHBP
|
6.3 | Ki | 8 | — | |
IEYUPLSSJBQATP
|
6.3 | IC50 | 3 | Yes | |
VEAGDTHATZZACO
|
6.3 | IC50 | 2 | — | |
AWJFHAOMPVPERV
|
6.3 | IC50 | 2 | — | |
FRXRVVOCWBNHOQ
|
6.3 | Ki | 3 | — | |
HKKVAUZCGNRBNA
|
6.3 | IC50 | 4 | — | |
JYYLJFGDJRYBNN
|
6.3 | IC50 | 3 | — |