Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QRDJMZMVDBUNNQ
|
6.5 | IC50 | 5 | Yes | |
ZGEUEQMPAIUHSM
|
6.5 | IC50 | 3 | Yes | |
CXPHOOFGGKZGTC
|
6.5 | Ki | 5 | — | |
OEXQBZKLEMTXMU
|
6.5 | Ki | 3 | — | |
PTUSTBHDXAVNPJ
|
6.5 | IC50 | 5 | Yes | |
YLPGDDBCDVVMDA
|
6.5 | IC50 | 4 | Yes | |
FIBCANQMNSDCGQ
|
6.5 | IC50 | 4 | — | |
PEOWGCZHIMSTFM
|
6.5 | IC50 | 2 | — | |
NPTUUUXCZCQNQS
|
6.5 | IC50 | 5 | — | |
RMJFXTVVOBTABN
|
6.5 | IC50 | 3 | Yes | |
XNDAUZRSIAEAAR
|
6.5 | Ki | 6 | — | |
AWDSUFIHUSMPAR
|
6.5 | IC50 | 3 | Yes | |
BWHNAQMOABQLDB
|
6.5 | IC50 | 4 | Yes | |
OURSUJYXZLSVCS
|
6.5 | IC50 | 5 | — | |
RPWIXTPWMSUQKW
|
6.5 | IC50 | 4 | Yes | |
KIMPOJXDFKFBTL
|
6.5 | IC50 | 2 | — | |
LOOGWNWWNBNMRC
|
6.5 | IC50 | 4 | Yes | |
MDOGBVLWCBWUMC
|
6.5 | IC50 | 5 | Yes | |
DKBDATWDEJHFQS
|
6.4 | IC50 | 2 | — | |
DUPWUQYVKWCUOG
|
6.4 | Ki | 7 | — | |
FFCQFLOKIRUZOS
|
6.4 | IC50 | 3 | — | |
KAUWQENTXQTKQG
|
6.4 | Ki | 4 | — | |
MFBQXIJAOSFCJR
|
6.4 | IC50 | 3 | Yes | |
PPLPLBVUEJOBPI
|
6.4 | IC50 | 4 | — | |
RJKVRZJNTANTQB
|
6.4 | IC50 | 2 | — | |
PKQOURGVZCVPOK
|
6.4 | IC50 | 2 | — | |
QNMBQUIJYLNNSV
|
6.4 | IC50 | 3 | — | |
UDTXDKDGZMYOBK
|
6.4 | IC50 | 5 | Yes | |
WKYYIJNBJSICFM
|
6.4 | IC50 | 5 | — | |
WOIMZSMDPIJLFO
|
6.4 | Ki | 7 | Yes | |
FGEXLQKMIJWUIY
|
6.4 | IC50 | 5 | Yes | |
KHHNQNYSKXXUCV
|
6.4 | Ki | 2 | — | |
UHWQCCAGEXNQTH
|
6.4 | IC50 | 3 | Yes | |
VACPECYZKUSTIV
|
6.4 | Ki | 2 | — | |
ZMQVXCLMHVVMKI
|
6.4 | IC50 | 2 | — | |
CXZHJWRHSTZNHB
|
6.4 | IC50 | 4 | Yes | |
IDKKXCKXGPPWMS
|
6.4 | IC50 | 5 | Yes | |
UEOYACNTKVVWRI
|
6.4 | Ki | 6 | Yes | |
VZHMZJYVSCWQIX
|
6.4 | IC50 | 5 | — | |
XXBXRJDBCMCGGD
|
6.4 | IC50 | 3 | — | |
LRYRCUJGWNCKPO
|
6.4 | IC50 | 5 | Yes | |
MVRHXCGLUWVMKH
|
6.4 | IC50 | 7 | Yes | |
OTDAXJIWZBAIMD
|
6.4 | IC50 | 2 | — | |
AGLYKFTUNLOGBT
|
6.4 | IC50 | 5 | Yes | |
BENVRUSKAIOVEH
|
6.4 | IC50 | 2 | — | |
IUPDLWWZWJCNBN
|
6.4 | IC50 | 2 | — | |
LJJFKNOMQHHBEW
|
6.4 | IC50 | 4 | Yes | |
UROHLDAMBMAOKL
|
6.4 | IC50 | 5 | Yes | |
NLIWJNDBQYUCSF
|
6.4 | Ki | 4 | — | |
QCBWOUQUDIILOW
|
6.4 | IC50 | 5 | Yes |