Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QGVCPEQAAKTMNX
|
6.6 | IC50 | 3 | Yes | |
ZVQKPPCVSXIXMD
|
6.6 | IC50 | 5 | — | |
FGPWEPZCTGVLNA
|
6.6 | IC50 | 5 | Yes | |
LNMKFTOPZCDAED
|
6.6 | IC50 | 4 | Yes | |
UVGAWIJNBYCHSP
|
6.6 | Ki | 7 | — | |
VXYUSBYRYYLNHT
|
6.6 | Ki | 4 | — | |
AWLKOGZBGNQOBA
|
6.6 | IC50 | 5 | Yes | |
FRFSAUPOCJTACG
|
6.6 | IC50 | 3 | Yes | |
HGICQEUHJFERNR
|
6.6 | IC50 | 4 | Yes | |
KFGJNQLPIZMSFB
|
6.6 | IC50 | 5 | Yes | |
OREDIHYKGISTDR
|
6.6 | IC50 | 6 | Yes | |
QPSBVVFMTSFAJY
|
6.6 | IC50 | 5 | Yes | |
UVGAWIJNBYCHSP
|
6.6 | Ki | 9 | Yes | |
WRDNQNGMPREKKZ
|
6.6 | IC50 | 4 | Yes | |
CCTDBXLXFNHDIL
|
6.6 | IC50 | 2 | — | |
FFHXMPKAWWFPSX
|
6.6 | IC50 | 3 | Yes | |
IZRGHLXXFQNRMD
|
6.6 | IC50 | 2 | — | |
VMTJQZUZINLEKC
|
6.6 | IC50 | 5 | Yes | |
KNBKYJWSHYOTTH
|
6.6 | IC50 | 2 | — | |
LAXIFXUCVNKYRQ
|
6.6 | IC50 | 5 | Yes | |
MTIXYSCCUVKNDA
|
6.6 | IC50 | 3 | — | |
AVXZGSSHGFLSMF
|
6.5 | IC50 | 3 | — | |
BCBPGVLRMIXMDN
|
6.5 | IC50 | 4 | Yes | |
DIUYYSMPEUKBTJ
|
6.5 | IC50 | 2 | — | |
IQGHPUPMOUUHPP
|
6.5 | IC50 | 2 | Yes | |
MIENZPZOHXCZQM
|
6.5 | IC50 | 7 | — | |
OZKMQEXIBBMJLW
|
6.5 | IC50 | 3 | — | |
QRQKVQCDKFEWSW
|
6.5 | IC50 | 2 | — | |
VKBVPNSUAROFRU
|
6.5 | IC50 | 3 | — | |
WOYRYBDDOIPDIG
|
6.5 | IC50 | 3 | — | |
BDCJZZXWIQJYLP
|
6.5 | IC50 | 5 | Yes | |
BRHXKZALFBLRIF
|
6.5 | IC50 | 5 | Yes | |
OCVZODLPTGAJKD
|
6.5 | IC50 | 3 | Yes | |
ROPVZXZEHJGNGB
|
6.5 | IC50 | 3 | — | |
FSFVECJWHSGENK
|
6.5 | IC50 | 6 | Yes | |
FUXYTSOUUZCQPA
|
6.5 | IC50 | 7 | — | |
LYGIRBLDUCXHDY
|
6.5 | IC50 | 4 | Yes | |
FTRCUXMVUJZMHT
|
6.5 | IC50 | 7 | Yes | |
LEDMBBYIVRLZAS
|
6.5 | Ki | 9 | Yes | |
LQLNFJVHRIWFTO
|
6.5 | IC50 | 3 | Yes | |
NXFDHNJDXVCAMS
|
6.5 | IC50 | 2 | — | |
ROFAQOFULLWONA
|
6.5 | IC50 | 2 | Yes | |
VMMAOHBHWSKMLW
|
6.5 | IC50 | 4 | Yes | |
ACXIBBRPTTWRDM
|
6.5 | Ki | 2 | — | |
KEEWWGMUNANVLU
|
6.5 | IC50 | 5 | Yes | |
NUKWNBCRJJDVNF
|
6.5 | IC50 | 3 | — | |
PBCSMBZCRUWUMR
|
6.5 | IC50 | 2 | — | |
PBCSMBZCRUWUMR
|
6.5 | IC50 | 2 | — | |
LDDKAYGLGQWILO
|
6.5 | IC50 | 6 | — | |
PDKBAEDNMKVROV
|
6.5 | Ki | 9 | Yes |