Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ARFFCGXUOISSHZ
|
6.7 | IC50 | 6 | Yes | |
KLFOAKCPAGOTNG
|
6.7 | IC50 | 4 | Yes | |
NIAIEBGBRXKPAO
|
6.7 | Ki | 7 | — | |
PTYZKNZXNKWTEF
|
6.7 | IC50 | 6 | Yes | |
QFGALMYSDQBVRH
|
6.7 | Ki | 7 | — | |
TUJKFLFRSWBCFZ
|
6.7 | IC50 | 2 | — | |
YTQYMJLEQVXIPD
|
6.7 | Ki | 4 | — | |
CMALBPMZEURNBK
|
6.7 | Ki | 3 | — | |
CMALBPMZEURNBK
|
6.7 | Ki | 4 | Yes | |
VNIVLVJMMLQGNQ
|
6.7 | IC50 | 4 | Yes | |
WHUGMPJJQOVPAC
|
6.7 | IC50 | 4 | Yes | |
IIABJCHWKFZJBK
|
6.7 | Ki | 9 | Yes | |
ONGCECNMBMSPOG
|
6.7 | IC50 | 3 | Yes | |
ROFAQOFULLWONA
|
6.7 | IC50 | 5 | Yes | |
XQJGASWZRFSCKP
|
6.7 | IC50 | 3 | Yes | |
BFJIOGLKGISOKV
|
6.7 | Ki | 8 | — | |
MWKXYRJSVHPPLM
|
6.7 | IC50 | 4 | — | |
QVAVQQVTOJMLHH
|
6.7 | IC50 | 7 | Yes | |
SKLOAVPDSDQCQV
|
6.7 | IC50 | 2 | — | |
TWUOGBAWSSAHQE
|
6.7 | IC50 | 5 | — | |
YYOVZJXOBZVIQK
|
6.7 | IC50 | 3 | — | |
CREFCFAJHQSGNR
|
6.7 | IC50 | 3 | — | |
QPLRROCTSCFWJD
|
6.7 | IC50 | 2 | — | |
SKYVAYDFIWVHPU
|
6.7 | IC50 | 3 | Yes | |
SQQRAMLTIHSAJA
|
6.7 | IC50 | 2 | — | |
VOEOVKSVTSGALB
|
6.7 | IC50 | 6 | Yes | |
FHCIUVTYGHWJQR
|
6.7 | IC50 | 4 | — | |
JSEADFAWCUECMR
|
6.7 | IC50 | 4 | — | |
LFDHAXXLFUSQRL
|
6.7 | IC50 | 5 | Yes | |
RGCUFTVHLLFSQN
|
6.7 | IC50 | 2 | — | |
ZZBMCFITYYSQSJ
|
6.7 | IC50 | 3 | Yes | |
CEVLUPQNDFOYSI
|
6.6 | IC50 | 5 | Yes | |
MGIMQKIBRRRYRM
|
6.6 | IC50 | 4 | Yes | |
TZGXQAYCVFGRLH
|
6.6 | IC50 | 4 | Yes | |
UVZHWHPRZYNZSE
|
6.6 | IC50 | 3 | — | |
XBPHJVRPJAQGKS
|
6.6 | Ki | 3 | — | |
BDCJZZXWIQJYLP
|
6.6 | IC50 | 5 | Yes | |
BGPDKPPPOAJAIA
|
6.6 | IC50 | 2 | — | |
CWSSLFKLYYDKBD
|
6.6 | Ki | 3 | — | |
FODLAGUBVKDEIZ
|
6.6 | IC50 | 5 | Yes | |
JUEZHKLAFJJQNE
|
6.6 | Ki | 3 | — | |
MDDFFAOYZXGICC
|
6.6 | IC50 | 3 | Yes | |
RESDGLIYQGGYGR
|
6.6 | Ki | 3 | — | |
ZYKVSIDVBIFMGD
|
6.6 | IC50 | 3 | Yes | |
DZFFLJXATZFATL
|
6.6 | IC50 | 6 | Yes | |
KXDVOTQQRPPFNY
|
6.6 | IC50 | 3 | — | |
IIABJCHWKFZJBK
|
6.6 | Ki | 9 | Yes | |
JNFDCDGQVIEXPD
|
6.6 | IC50 | 5 | Yes | |
MWPVYUMZDJJEOU
|
6.6 | IC50 | 3 | Yes | |
NLZYFAYMHSXTEW
|
6.6 | IC50 | 3 | — |