Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GLFZNNLEMNMSQE
|
6.8 | IC50 | 3 | Yes | |
KISNQJUMQDMWMF
|
6.8 | IC50 | 3 | — | |
KOKCTGWRLDNNGZ
|
6.8 | IC50 | 3 | Yes | |
RBRFAUFMZOIMMS
|
6.8 | IC50 | 3 | — | |
WJFKRCVNGHZYFA
|
6.8 | IC50 | 5 | Yes | |
MESQXIKYNYUZRV
|
6.8 | IC50 | 4 | Yes | |
MNQFMKHWJNOSIX
|
6.8 | IC50 | 5 | Yes | |
NPWNPFHGYNOBOO
|
6.8 | IC50 | 7 | Yes | |
PDBHRMUGMOPNOC
|
6.8 | IC50 | 5 | Yes | |
VGMJDHAFWAQDDY
|
6.8 | IC50 | 4 | Yes | |
WDDBBBHPBMFFCX
|
6.8 | IC50 | 4 | — | |
DNWSNDYODYMMSH
|
6.8 | IC50 | 3 | — | |
WGRMVARLTSCXRH
|
6.8 | IC50 | 3 | Yes | |
YTQYMJLEQVXIPD
|
6.8 | Ki | 4 | — | |
AWEAPFWTHDDCFJ
|
6.8 | IC50 | 3 | Yes | |
FJRQWHSKVHCEKG
|
6.8 | IC50 | 4 | Yes | |
MBHDDZHFZICCLX
|
6.8 | IC50 | 4 | — | |
UVAFSUYDCCCUTO
|
6.8 | IC50 | 5 | Yes | |
XATUMTIXUAJCSA
|
6.8 | IC50 | 4 | — | |
XGGNDAOPHPLHFW
|
6.8 | IC50 | 4 | — | |
GFRCZBUEHADXTC
|
6.8 | IC50 | 3 | Yes | |
ZHMXASGBGYZMST
|
6.8 | IC50 | 3 | Yes | |
UQNGOLQNCCYWJR
|
6.8 | IC50 | 5 | Yes | |
FVDPKGPPYGTKTO
|
6.8 | IC50 | 2 | — | |
UYVXUYVAIIWBSW
|
6.8 | Ki | 3 | — | |
GISWZMJMNJMSEO
|
6.8 | IC50 | 4 | — | |
JWGZOXAEXNYYHO
|
6.8 | IC50 | 3 | Yes | |
KJUQRHGKOLRTFD
|
6.8 | IC50 | 3 | Yes | |
KSOLTKWEALJMDR
|
6.8 | IC50 | 5 | Yes | |
BGUXTVRZPYKBBN
|
6.7 | IC50 | 5 | Yes | |
CGAZROFVKJRMSR
|
6.7 | IC50 | 3 | Yes | |
JJTWETADXAELLS
|
6.7 | Ki | 9 | Yes | |
JXHAGXRDZALSLG
|
6.7 | Ki | 9 | Yes | |
KATBPZLMXQIZLF
|
6.7 | IC50 | 4 | Yes | |
MCYLJYADJGYSSU
|
6.7 | IC50 | 2 | — | |
NAMZXOAZPHMVHE
|
6.7 | IC50 | 3 | Yes | |
UBHBDSABSVVUTP
|
6.7 | IC50 | 4 | — | |
VFDHTLCJQNLYTR
|
6.7 | IC50 | 2 | — | |
DNUKGGCABDLAEO
|
6.7 | IC50 | 4 | Yes | |
FFGHBWJVBSUBKN
|
6.7 | IC50 | 2 | — | |
XRLMAIWPTHLVKY
|
6.7 | IC50 | 5 | Yes | |
ZUJXLCINYDKZGV
|
6.7 | IC50 | 4 | Yes | |
BIJSDGADEZEMHH
|
6.7 | IC50 | 2 | — | |
CNPRJTXDIHRZPF
|
6.7 | Ki | 4 | — | |
IASRCCATUJITDX
|
6.7 | IC50 | 4 | Yes | |
RDCLFTKMELYUEI
|
6.7 | IC50 | 2 | Yes | |
XORCBTCEBZUVES
|
6.7 | IC50 | 5 | Yes | |
DUPLEMOAJXTDKP
|
6.7 | IC50 | 4 | Yes | |
FNRFZJFDQHKMHF
|
6.7 | IC50 | 5 | Yes | |
FWGPCZGIMGDSOM
|
6.7 | IC50 | 5 | Yes |