Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MKAIHDAGQJQAHA
|
6.9 | IC50 | 5 | Yes | |
QFTWPDUNHCKGKX
|
6.9 | IC50 | 6 | Yes | |
SMWVRODLVRVTBW
|
6.9 | IC50 | 2 | — | |
QROXNPLBULDOSL
|
6.9 | IC50 | 4 | Yes | |
WXMUXNHNFVCNMU
|
6.9 | IC50 | 5 | — | |
KDSNJNDUIRTNNR
|
6.9 | IC50 | 2 | — | |
KDSNJNDUIRTNNR
|
6.9 | IC50 | 4 | Yes | |
WQCYWYOJQMZTMB
|
6.9 | IC50 | 4 | — | |
YSMSZPWEAVKTEN
|
6.9 | IC50 | 4 | Yes | |
ZCJYXMGAZICHPN
|
6.9 | IC50 | 3 | Yes | |
AXIUEWMOHLWPSR
|
6.9 | IC50 | 5 | Yes | |
BJBJSCJDKGVTKQ
|
6.9 | IC50 | 2 | — | |
INGMGORXRMQEAG
|
6.9 | IC50 | 3 | Yes | |
IYSKDTAJMOMROJ
|
6.9 | IC50 | 4 | Yes | |
LEMPBGCFFWGHBZ
|
6.9 | IC50 | 4 | — | |
RXYVRCSDLULANF
|
6.9 | IC50 | 2 | — | |
VOESHNWTIDIZCL
|
6.9 | Ki | 10 | Yes | |
WOIMZSMDPIJLFO
|
6.9 | Ki | 9 | Yes | |
FKTHQTYGTOEBAW
|
6.9 | Ki | 7 | — | |
IHWAKJKUYYZNCF
|
6.9 | IC50 | 6 | Yes | |
ZXQRCQILIYTPOF
|
6.9 | IC50 | 3 | Yes | |
APKBGNTVZCZTJL
|
6.9 | IC50 | 3 | — | |
BUELAJMDFCPTAV
|
6.9 | IC50 | 4 | — | |
RCCBHNFHHCGOQM
|
6.9 | IC50 | 4 | Yes | |
UZCHBPQXZPPPNZ
|
6.9 | IC50 | 2 | — | |
XLKQIIIKETWLMI
|
6.9 | Ki | 8 | — | |
XOBSNYRLSVUYKY
|
6.9 | IC50 | 2 | — | |
XRIJPQABKMSHIA
|
6.9 | IC50 | 3 | Yes | |
KMLOBHZAEFITDB
|
6.9 | IC50 | 4 | — | |
NRADMZCIASMSFG
|
6.9 | IC50 | 5 | Yes | |
VZKDMHBTNFCZIW
|
6.9 | IC50 | 4 | Yes | |
AXPBXFSDSKBQDG
|
6.8 | IC50 | 5 | Yes | |
FQZUGHBEAWJYRZ
|
6.8 | IC50 | 3 | Yes | |
JXHAGXRDZALSLG
|
6.8 | Ki | 9 | Yes | |
LUTKRKPVCCDDOR
|
6.8 | IC50 | 3 | Yes | |
LVVFBDASYOIWFN
|
6.8 | IC50 | 4 | Yes | |
MLRVULAXCZJAAN
|
6.8 | IC50 | 5 | Yes | |
NKGBFKCCSGHHPF
|
6.8 | IC50 | 2 | — | |
PYGZWPVJQNBFNS
|
6.8 | IC50 | 6 | Yes | |
ZEEUPEFKULHDHM
|
6.8 | IC50 | 2 | Yes | |
BTZMVJPRQAIPRP
|
6.8 | IC50 | 5 | Yes | |
GCCFOYRWIAVTCA
|
6.8 | IC50 | 3 | Yes | |
MAARMQUENBUSOG
|
6.8 | IC50 | 2 | — | |
UFEAOVWYWYBIFX
|
6.8 | IC50 | 4 | Yes | |
ZSZSGGNFCMWYDF
|
6.8 | IC50 | 3 | Yes | |
MLJSRWALBCZDCB
|
6.8 | IC50 | 3 | Yes | |
WTCSNHGGDSKNJP
|
6.8 | IC50 | 2 | — | |
WUJPOLIUEWWSHN
|
6.8 | IC50 | 2 | — | |
XAISFEMYYICOMZ
|
6.8 | IC50 | 4 | Yes | |
FHAJCDXKKGQJQW
|
6.8 | IC50 | 5 | Yes |