Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GGMOCOYDYRCVAH
|
7.0 | IC50 | 5 | Yes | |
PASQOFLVNKNUQM
|
7.0 | IC50 | 2 | — | |
BBPLRBWLQWBZIO
|
7.0 | IC50 | 5 | — | |
CPWMZTRXCCYTDM
|
7.0 | Ki | 10 | Yes | |
FCYBWLNLMVDLRH
|
7.0 | IC50 | 5 | — | |
FCYBWLNLMVDLRH
|
7.0 | IC50 | 7 | Yes | |
KOVQMCGGWATESY
|
7.0 | Ki | 7 | — | |
OCBYWAVDKLDIDI
|
7.0 | Ki | 5 | Yes | |
VMOSDDURWLNMNG
|
7.0 | IC50 | 8 | Yes | |
GIJWOCNEPGCMND
|
7.0 | IC50 | 4 | Yes | |
SQODILRODCBOCF
|
7.0 | IC50 | 5 | Yes | |
TYSBKRRVVCMKQG
|
7.0 | Ki | 4 | — | |
VVCQPDVATXLSSI
|
7.0 | IC50 | 5 | Yes | |
YTHUQFQHXZIQRV
|
7.0 | IC50 | 2 | — | |
DCRZEJJUPRPPOS
|
7.0 | IC50 | 3 | Yes | |
HANNJPXOWYFOHG
|
7.0 | IC50 | 2 | — | |
HBIQJOZNDMPMAG
|
7.0 | IC50 | 5 | Yes | |
LUHJAOVICRNTRC
|
7.0 | IC50 | 7 | Yes | |
MVEPSFJZKBVDHV
|
7.0 | IC50 | 7 | Yes | |
NFRICHJLQIOONF
|
7.0 | IC50 | 6 | Yes | |
OZAYVSZVQPANBZ
|
7.0 | IC50 | 2 | — | |
PLYGOFXFDNGSQZ
|
7.0 | IC50 | 3 | Yes | |
QGCFRSYWGLGDTC
|
7.0 | IC50 | 3 | Yes | |
QHRUJPVXLYJUEM
|
7.0 | IC50 | 6 | Yes | |
UICCGUSKKDLVIN
|
7.0 | IC50 | 6 | Yes | |
YMFBAKCSKQKFMX
|
7.0 | IC50 | 5 | Yes | |
PLCPLXITTDSMSK
|
7.0 | IC50 | 4 | Yes | |
SUEBJDNLBVTIQP
|
7.0 | Ki | 10 | Yes | |
XZFOATQBCODVSR
|
7.0 | IC50 | 3 | Yes | |
DRCOOMXUPYOBBW
|
7.0 | IC50 | 4 | — | |
LKVAANCBUJLQIE
|
7.0 | IC50 | 4 | Yes | |
NDTTWNHVVUKYIR
|
7.0 | IC50 | 5 | — | |
WUOWVIUWLFFAMY
|
7.0 | IC50 | 2 | — | |
WUVJCBZUUQXYIT
|
7.0 | IC50 | 4 | Yes | |
WYTXTYOLYMMDCW
|
7.0 | IC50 | 3 | Yes | |
FWPVXLYOKAOERT
|
7.0 | IC50 | 8 | Yes | |
KTMMYBDZBIJPLY
|
7.0 | IC50 | 4 | Yes | |
XLNFBXKUCFOQRQ
|
7.0 | IC50 | 4 | — | |
JSOUFOXMENBKFM
|
7.0 | IC50 | 4 | Yes | |
KKGJFHSYGOMRAH
|
7.0 | IC50 | 2 | — | |
GDBNAEMVDGQOCE
|
7.0 | IC50 | 7 | — | |
WRNMBFWQBKEBIX
|
7.0 | IC50 | 4 | Yes | |
JFCGISGLHXBESS
|
6.9 | IC50 | 2 | — | |
KOVQMCGGWATESY
|
6.9 | Ki | 5 | — | |
SBPZKNUSQCPAAY
|
6.9 | IC50 | 3 | Yes | |
XIQNNSMTTLQUTR
|
6.9 | IC50 | 6 | Yes | |
ZIKBROOIDUARGQ
|
6.9 | IC50 | 3 | — | |
GGDBCZZATDMWMQ
|
6.9 | IC50 | 4 | Yes | |
RAOGWYCOADLHPD
|
6.9 | Ki | 2 | — | |
GINBTQGVSPUJLE
|
6.9 | Ki | 9 | Yes |