Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RBTIHKNARDNLNU
|
7.1 | IC50 | 5 | Yes | |
QJKGJGURDPRKGW
|
7.1 | IC50 | 4 | Yes | |
QVIMBPCQZGHONM
|
7.1 | IC50 | 6 | Yes | |
CQGUKDZSAPDCJL
|
7.1 | IC50 | 5 | Yes | |
FIPYOKGRSDJCAR
|
7.1 | IC50 | 9 | Yes | |
IQUZJJXEDANMJD
|
7.1 | Ki | 4 | — | |
JCUTWTFOYUXMPS
|
7.1 | Ki | 10 | Yes | |
PRQWPDFKJBVNKQ
|
7.1 | IC50 | 6 | Yes | |
AAVVXYJNWGIBPT
|
7.1 | IC50 | 4 | Yes | |
BOXAYSWQFMJSDX
|
7.1 | IC50 | 6 | Yes | |
BVTIVQKMMMOOTF
|
7.1 | IC50 | 3 | Yes | |
CSAFQHHGNGUQOL
|
7.1 | Ki | 10 | Yes | |
FEOIBPWKGPFSTB
|
7.1 | IC50 | 3 | Yes | |
HJAQLIVSMXUHPV
|
7.1 | Ki | 10 | Yes | |
HVWVSAVLGKOEBY
|
7.1 | IC50 | 3 | Yes | |
IIUXBHAJTPNCIR
|
7.1 | Ki | 6 | — | |
KRGBAILWDVNOCW
|
7.1 | IC50 | 6 | Yes | |
NMPAJDNRYQXHBH
|
7.1 | IC50 | 3 | Yes | |
OEPLGUBYTRYCJX
|
7.1 | IC50 | 7 | Yes | |
OPYOHFRGHGDNSJ
|
7.1 | Ki | 7 | Yes | |
RMPYEISUTHEMLW
|
7.1 | IC50 | 3 | Yes | |
TUUMURVUDGZZQZ
|
7.1 | IC50 | 6 | Yes | |
CKYKLNXMCJIGPN
|
7.1 | Ki | 6 | — | |
TYZVGHNHMXVHTN
|
7.1 | Ki | 5 | — | |
XFLXFAKGEAQTOI
|
7.1 | IC50 | 4 | Yes | |
CNEKWCSJAXATCC
|
7.1 | IC50 | 6 | Yes | |
CYIOQNVVHKTYRH
|
7.1 | IC50 | 5 | Yes | |
ITWGWXCEGHFMHT
|
7.1 | IC50 | 10 | Yes | |
PTUCPHGSAFOJAU
|
7.1 | Ki | 9 | Yes | |
RLUGMDBAWBLDJQ
|
7.1 | IC50 | 5 | Yes | |
YUYXLIRWRFFNDS
|
7.1 | IC50 | 5 | Yes | |
YXQWYGVDVQBPGA
|
7.1 | IC50 | 4 | — | |
ZEZNNQDUSMNIDE
|
7.1 | IC50 | 5 | Yes | |
GHZXWVPNZMUKBT
|
7.1 | IC50 | 5 | Yes | |
HOSIVTBRRYYOOH
|
7.1 | Ki | 7 | Yes | |
JEALYKJUQQXXBO
|
7.1 | IC50 | 5 | Yes | |
PYKDJHBKQBUYDN
|
7.1 | IC50 | 2 | — | |
UZMHOPNYRMEVNJ
|
7.1 | IC50 | 5 | Yes | |
VMOSDDURWLNMNG
|
7.1 | IC50 | 5 | Yes | |
APJIPTNFOKEMIQ
|
7.1 | IC50 | 5 | Yes | |
DPDQSBRVGYFIHD
|
7.1 | IC50 | 4 | Yes | |
YNTZVOSILJPSFZ
|
7.1 | IC50 | 2 | — | |
CKCBYWFMRXPHJM
|
7.0 | Ki | 4 | — | |
JGDVFBCMNUSQQW
|
7.0 | IC50 | 5 | Yes | |
MOVLHCHTKCWLQE
|
7.0 | IC50 | 3 | Yes | |
UEGUSCZBRJCYEP
|
7.0 | IC50 | 2 | — | |
KJDPTHLLJDQIMT
|
7.0 | IC50 | 5 | Yes | |
QDHXNZRPVLUOML
|
7.0 | Ki | 6 | — | |
BGJNPKHDPBUJSP
|
7.0 | IC50 | 4 | — | |
CZWJAEJHLBICAX
|
7.0 | IC50 | 3 | — |