Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YXPTXTBBPCLWPQ
|
9.5 | IC50 | 4 | — | |
ZHIRJJYNGRGHQQ
|
9.5 | IC50 | 6 | Yes | |
KBZNOZAJAJRTII
|
9.5 | IC50 | 10 | Yes | |
WKXRIMLOWDOHMN
|
9.5 | Ki | 5 | Yes | |
JJSAEDOMTCNEQL
|
9.5 | IC50 | 2 | — | |
VMWGPLRCSWOQJR
|
9.5 | IC50 | 5 | Yes | |
LFIZWBFUWVSLOR
|
9.4 | Ki | 5 | — | |
MEDAEECOIUAMSO
|
9.4 | IC50 | 4 | Yes | |
HGMNWCDIIMBGAR
|
9.4 | IC50 | 4 | — | |
JIAWWQZPHLPQPH
|
9.4 | IC50 | 3 | Yes | |
AWBXCXPCFJCVSM
|
9.4 | IC50 | 4 | — | |
DABGHULKCXXLEE
|
9.4 | IC50 | 4 | — | |
DCSURGDKZBMZEV
|
9.4 | IC50 | 3 | Yes | |
DIIAIQCOHXBJHI
|
9.4 | IC50 | 6 | Yes | |
FIAWLFURFKPROF
|
9.4 | IC50 | 7 | Yes | |
FOSWRYKPHVPIDJ
|
9.4 | IC50 | 8 | Yes | |
GETDIWSMCUZGCD
|
9.4 | IC50 | 5 | Yes | |
GPLRECXXBJTJRJ
|
9.4 | IC50 | 6 | Yes | |
GXZSIAVJNPWNMR
|
9.4 | IC50 | 7 | Yes | |
HAIGFFSNUYJTQK
|
9.4 | IC50 | 6 | Yes | |
HDTLIPGODNAYEM
|
9.4 | IC50 | 5 | Yes | |
LBNAEOGDUCUPFZ
|
9.4 | IC50 | 4 | — | |
LFOGEPKUSWRLCL
|
9.4 | IC50 | 7 | Yes | |
LXRKTOCLXUHNEM
|
9.4 | IC50 | 6 | Yes | |
NOXYNXIAEWTFQX
|
9.4 | IC50 | 7 | Yes | |
RTBMQALBDMCUCU
|
9.4 | IC50 | 3 | Yes | |
SWRNCXLTVBBIMK
|
9.4 | IC50 | 7 | Yes | |
WBIKMXRYXWFRCE
|
9.4 | IC50 | 4 | Yes | |
WDPVPUZANMBBLA
|
9.4 | Ki | 6 | — | |
WIWASQOQNPNFMY
|
9.4 | IC50 | 5 | Yes | |
WXNWNNKHEJMQOM
|
9.4 | IC50 | 8 | Yes | |
XGMBTNMILCXDFB
|
9.4 | IC50 | 6 | Yes | |
XUDODBAIOYVRJQ
|
9.4 | IC50 | 3 | Yes | |
YBPDYJXZXAPGSU
|
9.4 | IC50 | 6 | Yes | |
YCKAPRALLQTAKS
|
9.4 | IC50 | 6 | Yes | |
ZIMPTCJSUZVWEK
|
9.4 | IC50 | 3 | Yes | |
HFAGTNGCAZYYLZ
|
9.3 | Ki | 13 | Yes | |
KOPIIXVBCHXDHO
|
9.3 | IC50 | 8 | Yes | |
CWYHAUKCGMBLAH
|
9.3 | Ki | 2 | — | |
BEQXRWLSEUIFKP
|
9.3 | Ki | 5 | — | |
CTVWOVYWOFCAMW
|
9.3 | IC50 | 5 | Yes | |
CWBVJJZJNOSACP
|
9.3 | IC50 | 4 | Yes | |
GYETWAWIKBOMPE
|
9.3 | IC50 | 7 | Yes | |
HRESAHCPDRLLRL
|
9.3 | IC50 | 3 | Yes | |
IOLRUMINDIUCLJ
|
9.3 | Ki | 8 | Yes | |
KJQLQEWCQDLQEA
|
9.3 | IC50 | 5 | Yes | |
KYOFVPKPPTUVKK
|
9.3 | IC50 | 8 | Yes | |
MAOGHLYYLNCNCI
|
9.3 | IC50 | 7 | Yes | |
NWFAIXPOXVQZQD
|
9.3 | Ki | 4 | — | |
PFIVDCYVKKFLEU
|
9.3 | IC50 | 5 | Yes |