Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RWOPWLLDIYQNCW
|
7.2 | IC50 | 6 | Yes | |
WQBAMGDQVHWIOJ
|
7.2 | IC50 | 3 | Yes | |
YEVVFVQVGXPEQO
|
7.2 | Ki | 5 | — | |
YOLXRZGSQUXDCT
|
7.2 | IC50 | 3 | — | |
DFWYBNIMFAUWSX
|
7.2 | IC50 | 5 | Yes | |
DJXZXNHJKPAVOT
|
7.2 | IC50 | 2 | — | |
NDCGWDYXJPEWRR
|
7.2 | IC50 | 3 | Yes | |
OUNOAPVJMCBRTF
|
7.2 | IC50 | 2 | — | |
FFHINXVCVWQCSG
|
7.2 | Ki | 6 | — | |
MXFJZXDWWXHXMV
|
7.2 | Ki | 7 | — | |
BGKNBDGHNBOSGD
|
7.2 | IC50 | 5 | Yes | |
CHTZMALPRVCUIK
|
7.2 | IC50 | 4 | — | |
YYBFXMXFWMJGLB
|
7.2 | IC50 | 8 | Yes | |
FJMHXOYGOGYKAU
|
7.2 | IC50 | 3 | Yes | |
HNEDFPGSHTUVKZ
|
7.2 | IC50 | 7 | Yes | |
IFVVAVDCKGJFSK
|
7.2 | IC50 | 3 | Yes | |
NZKKRYAESABOSS
|
7.2 | IC50 | 8 | Yes | |
WVAIZSKMOMDPIT
|
7.2 | IC50 | 6 | Yes | |
ALKUUIDKRJZTBK
|
7.2 | IC50 | 2 | — | |
DVNVXZQJDUVWTB
|
7.2 | IC50 | 3 | Yes | |
FITYZYBFZVGBBP
|
7.2 | IC50 | 4 | — | |
NUUIPCGHCDKNAY
|
7.2 | IC50 | 2 | — | |
RTBMLCLTYAPKIF
|
7.2 | IC50 | 5 | Yes | |
SMRKDKVRUIEVHG
|
7.2 | IC50 | 5 | Yes | |
TVHNMQFVUGWIID
|
7.2 | IC50 | 5 | Yes | |
UVYWXUJXEFVRIM
|
7.2 | IC50 | 3 | Yes | |
XYVVUCAHUUIYFV
|
7.2 | IC50 | 6 | Yes | |
XZWFHJUEAVOHHG
|
7.2 | IC50 | 6 | Yes | |
CXRYZROMBCZZFO
|
7.2 | IC50 | 7 | Yes | |
IFHBUYGFCSEHIF
|
7.2 | IC50 | 6 | Yes | |
IHKCSGLIRGMLDE
|
7.2 | IC50 | 5 | Yes | |
RPOIZUWTBLHTNU
|
7.2 | IC50 | 3 | Yes | |
XMKAMECIIHUBSZ
|
7.2 | IC50 | 5 | Yes | |
XWQYRXPGPDOWAJ
|
7.2 | IC50 | 5 | Yes | |
ZGBAPSHWPBXEKN
|
7.2 | IC50 | 10 | — | |
ZYWQCDFNGKDOSB
|
7.2 | IC50 | 5 | Yes | |
BNKOGVVBAYMLMZ
|
7.2 | IC50 | 6 | Yes | |
BZTZPJQXNWROKR
|
7.2 | IC50 | 4 | — | |
JVBPIOHSXSYBRG
|
7.2 | Ki | 7 | Yes | |
MNJDNDDQYDSDCH
|
7.2 | IC50 | 2 | — | |
STWCTQDLUUVJMC
|
7.2 | Ki | 10 | Yes | |
TWUHFGMOEBVGGW
|
7.2 | IC50 | 3 | Yes | |
DLWHWYIHKZASJX
|
7.2 | IC50 | 2 | — | |
DKLKUPISRVEUAG
|
7.1 | IC50 | 3 | Yes | |
FROMXYGXLCSILK
|
7.1 | IC50 | 3 | — | |
JJHRUUKMPWUYIB
|
7.1 | IC50 | 5 | Yes | |
MVCDTECIYPRJTL
|
7.1 | IC50 | 2 | — | |
UHXPHVQOXYZQPP
|
7.1 | IC50 | 4 | — | |
WYVILPRSBDCCKY
|
7.1 | Ki | 7 | Yes | |
CPUBMGYGVNFLPZ
|
7.1 | IC50 | 8 | Yes |