Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VSJBIWYXNLUPIE
|
7.4 | Ki | 10 | Yes | |
WBHJOSGWNQHLCM
|
7.4 | IC50 | 3 | Yes | |
WXFYHQKQOWMEDX
|
7.4 | IC50 | 3 | Yes | |
YLYMDJMYRSEUOA
|
7.4 | IC50 | 7 | Yes | |
ZBTKKYFIZQHNDQ
|
7.4 | IC50 | 7 | Yes | |
ZVAKMIZOMSWYGQ
|
7.4 | IC50 | 7 | Yes | |
AQKDLUIAUGFUEC
|
7.4 | Ki | 7 | Yes | |
GHKVZKUXCOXDAW
|
7.4 | IC50 | 6 | Yes | |
ZQBRASLBYJYZLM
|
7.4 | IC50 | 5 | Yes | |
DBYYJEGRUPLGLD
|
7.4 | Ki | 7 | Yes | |
FDKIFIWQKFBOTH
|
7.4 | IC50 | 5 | Yes | |
KFTWEWMQNRZZNL
|
7.4 | IC50 | 5 | Yes | |
OUIRYNJKZCTIHG
|
7.4 | IC50 | 5 | Yes | |
QTUCHEGSWFEUBW
|
7.4 | Ki | 3 | — | |
TWTZRHWHKRIAHT
|
7.4 | IC50 | 3 | Yes | |
AJXYMDJBIXFLCO
|
7.4 | IC50 | 6 | Yes | |
HLPVNHUQEVIWBT
|
7.4 | IC50 | 3 | Yes | |
HQIAPHYTAVZNQW
|
7.4 | IC50 | 3 | Yes | |
INVXSBCIDABVMG
|
7.4 | IC50 | 5 | Yes | |
IQNGGJYKFADFHE
|
7.4 | IC50 | 4 | — | |
IQNGGJYKFADFHE
|
7.4 | IC50 | 6 | Yes | |
KAWCOVYOZMDLKQ
|
7.4 | IC50 | 4 | Yes | |
NPZDPBHMFYXBRP
|
7.4 | IC50 | 4 | Yes | |
IKJQAKILPMDYQE
|
7.4 | IC50 | 4 | Yes | |
RBRSAOMOZVVQSQ
|
7.4 | IC50 | 4 | Yes | |
WKTQKJFJPJOVNX
|
7.4 | IC50 | 3 | Yes | |
WPGRSZLFNFYSPR
|
7.4 | IC50 | 4 | — | |
ZAVWWISQYKVWCT
|
7.4 | IC50 | 6 | Yes | |
AUIKJLRMPLDORG
|
7.3 | Ki | 10 | Yes | |
BTDOGCFKKXBYKB
|
7.3 | IC50 | 3 | Yes | |
FTUOECQUSPMQQZ
|
7.3 | Ki | 7 | Yes | |
FBDOWURNGYMLPJ
|
7.3 | Ki | 7 | — | |
FWPVXLYOKAOERT
|
7.3 | IC50 | 4 | — | |
IVDMXEGLZLKBRS
|
7.3 | IC50 | 5 | Yes | |
KHCZZISCPQRODX
|
7.3 | Ki | 6 | Yes | |
QDUBONLFDSIPOU
|
7.3 | IC50 | 2 | — | |
KRJQQXQOPZJOSC
|
7.3 | IC50 | 5 | Yes | |
MJYIMHGWKZRGTK
|
7.3 | IC50 | 2 | — | |
WGPIMMRNIAYWBT
|
7.3 | IC50 | 5 | Yes | |
XFKRGURHEZYQDK
|
7.3 | IC50 | 5 | Yes | |
BUSXTPHZLBAFDD
|
7.3 | IC50 | 5 | Yes | |
HSQOMGXZKXTHEM
|
7.3 | IC50 | 5 | Yes | |
PTONAIKVYGVBIS
|
7.3 | IC50 | 5 | Yes | |
CWDYQHCEZVYJNX
|
7.3 | Ki | 3 | — | |
HFRJPVNBQJAJIX
|
7.3 | IC50 | 4 | Yes | |
OFRXWZGHEVNQHU
|
7.3 | Ki | 6 | — | |
PTUCPHGSAFOJAU
|
7.3 | Ki | 9 | — | |
PTUCPHGSAFOJAU
|
7.3 | Ki | 7 | — | |
YCIYENASUWAOBH
|
7.3 | IC50 | 5 | Yes | |
BBYYDINTRXZVIU
|
7.3 | IC50 | 3 | Yes |