Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UTVAYVOWTJFEEU
|
7.5 | Ki | 7 | Yes | |
ZWXRGJMHGHMUMB
|
7.5 | Ki | 4 | — | |
IEGOFALJZJPJJD
|
7.5 | IC50 | 4 | Yes | |
ODGSTGNVDAZIJX
|
7.5 | IC50 | 3 | Yes | |
TXFWBKCCZLIBMU
|
7.5 | IC50 | 3 | Yes | |
ZAXFGRVMMQJZLL
|
7.5 | IC50 | 5 | Yes | |
AQWIHDVVCANJLS
|
7.5 | Ki | 3 | — | |
DNPNWGZXJBALIP
|
7.5 | IC50 | 3 | Yes | |
DWAPKTBJQHYHER
|
7.5 | IC50 | 6 | Yes | |
MFTZEUCXFCXINH
|
7.5 | Ki | 6 | — | |
PNAVYQLZJZNXTL
|
7.5 | IC50 | 2 | — | |
SBXVFSKKCXNEDY
|
7.5 | IC50 | 3 | Yes | |
ZOSFRKHRZHSICA
|
7.5 | IC50 | 3 | Yes | |
ZUERCGBCDFBAQX
|
7.5 | IC50 | 3 | Yes | |
HXOLPPZDNXMRHR
|
7.4 | Ki | 4 | — | |
JUPHQCOZPHPYPF
|
7.4 | IC50 | 4 | Yes | |
ONOMIQQPBDQZDA
|
7.4 | Ki | 7 | Yes | |
PFPVZWIKTNGHGO
|
7.4 | Ki | 7 | Yes | |
QPLQAMVXCDXOBY
|
7.4 | IC50 | 5 | — | |
SAJAWNZBKHGJOW
|
7.4 | Ki | 6 | — | |
UFYJMKIWYONTIU
|
7.4 | IC50 | 5 | Yes | |
WKYNDNVMBNENDU
|
7.4 | IC50 | 4 | Yes | |
ZMDMPUVIZFSSCM
|
7.4 | IC50 | 4 | Yes | |
AGRDSOUIPBKOKQ
|
7.4 | IC50 | 4 | Yes | |
LXSYXSGOVAASBA
|
7.4 | IC50 | 6 | Yes | |
RGDPJPMKLABBRX
|
7.4 | Ki | 7 | Yes | |
UQRFKNRXERPSMG
|
7.4 | IC50 | 5 | Yes | |
VKSDFADIGYDZCS
|
7.4 | IC50 | 3 | Yes | |
AOGWJSJATLXUOJ
|
7.4 | IC50 | 6 | Yes | |
HHJKMUMZRIIHIU
|
7.4 | Ki | 10 | Yes | |
LNLWALQGRPVSTA
|
7.4 | IC50 | 3 | Yes | |
UWLVDBFIOGAENY
|
7.4 | IC50 | 2 | — | |
UZVVYDVVOHQVFV
|
7.4 | IC50 | 3 | Yes | |
ZAMIBNJCPAMMPI
|
7.4 | IC50 | 3 | Yes | |
COMDPQPBGQXLMK
|
7.4 | IC50 | 5 | Yes | |
FITQSJBSXMDHOS
|
7.4 | IC50 | 4 | — | |
IPKOKUIXGDZGRK
|
7.4 | IC50 | 4 | — | |
IYEVXJPUTMBOTO
|
7.4 | Ki | 7 | Yes | |
LNPBBURQSUEIHO
|
7.4 | IC50 | 5 | Yes | |
RLDMWDXYWMJUAA
|
7.4 | IC50 | 3 | — | |
WYWAKLNLTJVWAB
|
7.4 | IC50 | 6 | Yes | |
DODLQVHRMPIMNB
|
7.4 | IC50 | 4 | Yes | |
IERBLZLEQYZHMU
|
7.4 | IC50 | 3 | Yes | |
IOEYWFCDGXVEFG
|
7.4 | IC50 | 3 | Yes | |
KOVQMCGGWATESY
|
7.4 | Ki | 7 | — | |
LRVIJTRFTUQDKW
|
7.4 | IC50 | 7 | Yes | |
NZFXVEQIRZMPRQ
|
7.4 | IC50 | 2 | — | |
PTJXSKQZLWNDNB
|
7.4 | IC50 | 5 | Yes | |
PXTTXJDSBQDLQB
|
7.4 | IC50 | 3 | Yes | |
QFAMXNMLWJDJPV
|
7.4 | IC50 | 5 | Yes |