Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RMUMGJZUGCOZOV
|
7.5 | IC50 | 6 | Yes | |
RTBPRRSADWSXAD
|
7.5 | Ki | 7 | Yes | |
SOPJLCCBZBCHFQ
|
7.5 | IC50 | 3 | Yes | |
URNFYSXQOHQAJN
|
7.5 | IC50 | 3 | Yes | |
WBRQJRYOZZQHQI
|
7.5 | IC50 | 3 | Yes | |
XDSILIXRMZXTNX
|
7.5 | IC50 | 5 | Yes | |
AVQCFDJVRXAPJO
|
7.5 | IC50 | 5 | Yes | |
BLQAAMGUGMNRQN
|
7.5 | IC50 | 6 | Yes | |
CPDXTLZUFAYJLD
|
7.5 | IC50 | 5 | Yes | |
DDSDNLBIGCANQU
|
7.5 | IC50 | 3 | Yes | |
GJICTISPMDMSQH
|
7.5 | IC50 | 4 | Yes | |
GWRXKVPUXYYCMA
|
7.5 | IC50 | 3 | Yes | |
MXZLDTSVPDTTAN
|
7.5 | Ki | 7 | Yes | |
NCROEDXPKVIJMH
|
7.5 | IC50 | 2 | — | |
WNPLPMIXLXNWFU
|
7.5 | IC50 | 3 | Yes | |
SBYCYYMPCYJMTP
|
7.5 | IC50 | 7 | Yes | |
BMJUABISSDGKOA
|
7.5 | Ki | 6 | — | |
CWKUARBGJRTUFB
|
7.5 | IC50 | 3 | Yes | |
FWZHHLOLYIUTJO
|
7.5 | IC50 | 3 | Yes | |
QCVLVTVGVJUODZ
|
7.5 | Ki | 6 | — | |
SILYLRSFWCVUFM
|
7.5 | Ki | 7 | Yes | |
YDCLZJDJJGSFJZ
|
7.5 | Ki | 7 | Yes | |
YJNWDJIIFRGLRO
|
7.5 | Ki | 6 | Yes | |
YLRFPZVTHHHQAF
|
7.5 | IC50 | 4 | Yes | |
GQVFUZHQNCWOMM
|
7.5 | IC50 | 5 | Yes | |
KDJZFDKCOPXERM
|
7.5 | IC50 | 5 | Yes | |
PAICNGFUXUHAMP
|
7.5 | IC50 | 4 | Yes | |
PYXPFZLYNSTHAH
|
7.5 | Ki | 4 | — | |
VAMKUUUJVOOTKN
|
7.5 | IC50 | 5 | Yes | |
WLZISXXOYYGJNT
|
7.5 | Ki | 12 | Yes | |
CYDOQDKDFWIELG
|
7.5 | IC50 | 5 | Yes | |
FVYBFRCALRJYHO
|
7.5 | IC50 | 5 | Yes | |
IPGBSWJQXVYQBT
|
7.5 | IC50 | 3 | Yes | |
ISBRGXFRKARDDV
|
7.5 | IC50 | 5 | Yes | |
IVBBTZQIKSRCPC
|
7.5 | IC50 | 3 | Yes | |
KDBQSPNKNKKPEM
|
7.5 | IC50 | 3 | Yes | |
SPHCUXPEUQITEV
|
7.5 | IC50 | 6 | Yes | |
UXTQFUKVODXBBJ
|
7.5 | IC50 | 3 | Yes | |
YMYDSTVSNKTLJM
|
7.5 | Ki | 7 | Yes | |
FYYONZZUDPFMJO
|
7.5 | IC50 | 5 | Yes | |
ABWKZZSKNBCWLN
|
7.5 | IC50 | 3 | Yes | |
AXDNELHYOHIRLD
|
7.5 | IC50 | 4 | Yes | |
CTEBTZSRXSZTCW
|
7.5 | Ki | 7 | Yes | |
HCEJOINDKHKFPT
|
7.5 | IC50 | 3 | Yes | |
HSFOMBDSDMOJCP
|
7.5 | IC50 | 4 | Yes | |
LWAJTROMLACBIU
|
7.5 | IC50 | 2 | — | |
MWFBMGWABXFCCK
|
7.5 | IC50 | 4 | Yes | |
NHZSRXRDEWWJJS
|
7.5 | Ki | 6 | — | |
PHGLPDURIUEELR
|
7.5 | IC50 | 7 | Yes | |
QZURMXFXKAPVRT
|
7.5 | IC50 | 3 | Yes |