Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JGJZJJQMNAKKDG
|
7.6 | Ki | 7 | Yes | |
KMBQQDDLWIEVKL
|
7.6 | IC50 | 4 | Yes | |
KVLYVSHQXNTARE
|
7.6 | IC50 | 4 | Yes | |
LEWMAZXEBPMBSY
|
7.6 | Ki | 8 | Yes | |
MTSOZTJGECJILJ
|
7.6 | IC50 | 6 | Yes | |
NZUPMMOEPOVBQE
|
7.6 | Ki | 5 | — | |
QFPRVWUEWDLNPU
|
7.6 | Ki | 7 | Yes | |
RGJXGQMBVWRXCQ
|
7.6 | IC50 | 5 | Yes | |
SDNJCCVGVQBNKQ
|
7.6 | IC50 | 2 | — | |
SFWRCXWXHAIKBP
|
7.6 | IC50 | 5 | Yes | |
UPPWLWGJBCEKOO
|
7.6 | IC50 | 3 | Yes | |
VEUYFZWVWBJLBT
|
7.6 | IC50 | 6 | Yes | |
XNLVNQQMTWGGIM
|
7.6 | IC50 | 5 | Yes | |
XUHCFLAIQCGOLL
|
7.6 | IC50 | 3 | Yes | |
ZPFSKFCSVXPMBD
|
7.6 | Ki | 6 | Yes | |
DJZNIZCARKSSDE
|
7.6 | IC50 | 9 | Yes | |
DMMXGBRKSOTFSC
|
7.6 | IC50 | 3 | Yes | |
DWGIEOGNSCZDJK
|
7.6 | IC50 | 3 | — | |
JSQUVSOHRBZSNW
|
7.6 | IC50 | 5 | Yes | |
KUNPRZXRPKRXHM
|
7.6 | IC50 | 4 | Yes | |
KURIXYQCCHLXJD
|
7.6 | IC50 | 3 | Yes | |
LIYRHLZYJZBQCM
|
7.6 | IC50 | 3 | Yes | |
QJQSFVGRKOULTN
|
7.6 | IC50 | 3 | Yes | |
TVMGXYGVVFPAHO
|
7.6 | IC50 | 3 | Yes | |
VMTQLXIANRICIV
|
7.6 | IC50 | 2 | — | |
VSLVJIBOSDQNRC
|
7.6 | Ki | 2 | — | |
CTCOBJWAVVPWJG
|
7.6 | IC50 | 5 | Yes | |
OKJQKYSMNUJIEF
|
7.6 | IC50 | 2 | — | |
JFQFSHSHMHJPSW
|
7.6 | IC50 | 5 | Yes | |
KHCVBQLHKXPRJT
|
7.6 | IC50 | 4 | Yes | |
QGGLZVYZDFRHHX
|
7.6 | IC50 | 3 | Yes | |
SEOIKBYFTLCBTF
|
7.6 | IC50 | 6 | Yes | |
YWAPUIQWVUXRRW
|
7.6 | IC50 | 4 | Yes | |
ZLOBLTFULLQWKZ
|
7.6 | IC50 | 6 | Yes | |
DOPZAFIJEYWGQT
|
7.6 | IC50 | 4 | Yes | |
HOXYEQZQHOZJQN
|
7.6 | IC50 | 3 | Yes | |
LZVLSPCMSRJJKT
|
7.6 | IC50 | 3 | Yes | |
QCHHXEMLMRDLDA
|
7.6 | IC50 | 6 | Yes | |
QCLOBJCDRHHNCL
|
7.6 | Ki | 10 | Yes | |
QOOGIVWLICWQOB
|
7.6 | IC50 | 5 | Yes | |
RRUNLAIBQVECGY
|
7.6 | IC50 | 5 | Yes | |
VLGURNLPQGCFIS
|
7.6 | IC50 | 4 | Yes | |
WQCOVODIHQDZNG
|
7.6 | IC50 | 5 | Yes | |
ZXVWNUSVQOQAIY
|
7.6 | Ki | 5 | — | |
HWZVYNMATDDRGV
|
7.6 | IC50 | 4 | Yes | |
BHCRZOUPEFVWHZ
|
7.5 | IC50 | 3 | Yes | |
BTCYLUBBXQARQV
|
7.5 | Ki | 7 | — | |
FNCXJJHZBHAVJZ
|
7.5 | IC50 | 2 | — | |
FSJPBIIVCZKHRS
|
7.5 | IC50 | 2 | — | |
IMCGJWBSANDEHB
|
7.5 | IC50 | 3 | Yes |