Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KUDDIXBNWHQPDJ
|
7.7 | IC50 | 5 | Yes | |
LOYIGNDQOZNJNZ
|
7.7 | Ki | 7 | Yes | |
MOHDKNTXJIGORP
|
7.7 | Ki | 7 | Yes | |
RCOBSDNFRJAUBV
|
7.7 | IC50 | 4 | Yes | |
REXXRRWHIZEEBC
|
7.7 | IC50 | 3 | Yes | |
RIICMTINBCLPOY
|
7.7 | Ki | 6 | — | |
ROWNCZWVCCMTQI
|
7.7 | IC50 | 5 | Yes | |
SKADGQGCAOBKKC
|
7.7 | Ki | 7 | Yes | |
YOEUGEBWOYBNPP
|
7.7 | IC50 | 3 | Yes | |
ZOPDCQZNGWSOLM
|
7.7 | IC50 | 5 | Yes | |
GSCKLBZEPMMUCA
|
7.7 | IC50 | 4 | Yes | |
GTRBSPVJGOLISO
|
7.7 | IC50 | 5 | Yes | |
HGCCQMHYESJBML
|
7.7 | Ki | 7 | Yes | |
HLJHTDAQDAFOFS
|
7.7 | Ki | 7 | Yes | |
HUAZIQKZKFNJLA
|
7.7 | IC50 | 6 | — | |
JXCARHJPSZBVFH
|
7.7 | IC50 | 6 | Yes | |
JZIODDCGNMBMLB
|
7.7 | IC50 | 5 | Yes | |
JZJWCJQEWXNHBE
|
7.7 | IC50 | 5 | Yes | |
MALRHJHVJCYQHD
|
7.7 | IC50 | 5 | Yes | |
NEUXHEKNAOUEQU
|
7.7 | Ki | 7 | Yes | |
NZWCKNGEMCPIOP
|
7.7 | IC50 | 2 | — | |
RUILUWMFIHGOHD
|
7.7 | IC50 | 4 | Yes | |
SFHMNFHDIRPFKM
|
7.7 | IC50 | 7 | Yes | |
UNINFAIJOLFFHN
|
7.7 | IC50 | 5 | Yes | |
UXURFMZZZWZYFW
|
7.7 | IC50 | 6 | Yes | |
XWNLDJDYIDRBJI
|
7.7 | IC50 | 2 | — | |
ZCXHDGANXIWOBA
|
7.7 | IC50 | 3 | — | |
XUOKZLGAMXUMSE
|
7.7 | IC50 | 3 | — | |
BCVFMUCILNFXOC
|
7.7 | IC50 | 5 | Yes | |
CTONTIQKTODDRQ
|
7.7 | IC50 | 5 | Yes | |
KVUZGLYOUHGFEF
|
7.7 | IC50 | 5 | Yes | |
PMHIYNQSFXKIMZ
|
7.7 | IC50 | 5 | Yes | |
QTXKDSNGGLBSKK
|
7.7 | Ki | 7 | Yes | |
TUUMURVUDGZZQZ
|
7.7 | IC50 | 6 | Yes | |
UIVFNXLDHQCJRY
|
7.7 | IC50 | 4 | — | |
VJCSPSPTFYXXJB
|
7.7 | IC50 | 6 | Yes | |
WNQMYJZKTYVQPU
|
7.7 | IC50 | 7 | Yes | |
AXBFSSCCVFPFFC
|
7.6 | IC50 | 7 | Yes | |
BHJRCMPVJFWSEN
|
7.6 | IC50 | 2 | — | |
HTUSESRFPXTJLY
|
7.6 | IC50 | 4 | — | |
HXNNABWLGZRTMD
|
7.6 | IC50 | 5 | Yes | |
MGQZHWBYKGXMDX
|
7.6 | IC50 | 5 | Yes | |
NOYXCNRQZBBVGT
|
7.6 | Ki | 7 | Yes | |
PRHFUFABVIQNBK
|
7.6 | IC50 | 3 | Yes | |
RWOLXJOULAGHOB
|
7.6 | IC50 | 5 | Yes | |
UKASSNVNXOWYDK
|
7.6 | IC50 | 4 | — | |
XHPUXKQBUUHEIP
|
7.6 | Ki | 6 | — | |
BGBWSADVPWNBME
|
7.6 | IC50 | 9 | Yes | |
BRECBJOQRORDAF
|
7.6 | IC50 | 3 | Yes | |
FWHAUZNOWRAZOA
|
7.6 | IC50 | 3 | Yes |