Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CSPDSJARPZQPMQ
|
7.8 | Ki | 7 | Yes | |
DPDYQDPIBOABCX
|
7.8 | IC50 | 3 | Yes | |
DYSNZNGQZPYHHP
|
7.8 | Ki | 7 | Yes | |
HHSADBHNZPOTTJ
|
7.8 | Ki | 7 | Yes | |
TUUMURVUDGZZQZ
|
7.8 | IC50 | 3 | — | |
AYZMSYVMXDNCPT
|
7.7 | IC50 | 2 | — | |
BBQIWKGIQNPWJU
|
7.7 | IC50 | 3 | Yes | |
FLIOXLIZONFFSH
|
7.7 | IC50 | 3 | — | |
FROMXYGXLCSILK
|
7.7 | IC50 | 3 | — | |
HBDUXNUNXGZOCK
|
7.7 | IC50 | 4 | — | |
KNOYHJOPRUTPSQ
|
7.7 | Ki | 7 | — | |
LAGAITXTFHYXGS
|
7.7 | IC50 | 5 | Yes | |
MIWJQVMHJSFHGV
|
7.7 | IC50 | 5 | Yes | |
OEHVKBKRRIUTOR
|
7.7 | Ki | 6 | Yes | |
PPTRNTHJEHNDDP
|
7.7 | IC50 | 4 | Yes | |
PZMQNEDVJSDLAW
|
7.7 | Ki | 6 | — | |
UGRPRGWEEBXORM
|
7.7 | IC50 | 3 | — | |
WHSJFJHSWYAKDM
|
7.7 | IC50 | 3 | Yes | |
WMBVCTBFQRRSBU
|
7.7 | IC50 | 4 | Yes | |
XSEREZCRIQFANN
|
7.7 | IC50 | 3 | Yes | |
YHSMTPXGPORQER
|
7.7 | IC50 | 3 | Yes | |
ZPNXAVJYHSAOKF
|
7.7 | IC50 | 7 | Yes | |
DKTYDWAJILHINP
|
7.7 | IC50 | 3 | Yes | |
HMJIPPQTLJLPNE
|
7.7 | IC50 | 3 | Yes | |
IJIWBJJLSPLOBZ
|
7.7 | IC50 | 2 | — | |
IPNPHTJFPPPVQA
|
7.7 | IC50 | 6 | Yes | |
ITMFWUAKJPURIP
|
7.7 | Ki | 6 | Yes | |
JXZUMXBHWMKALL
|
7.7 | Ki | 3 | — | |
MHGISLAIZQKUNW
|
7.7 | Ki | 7 | Yes | |
MHYRZRJQEBSULL
|
7.7 | Ki | 6 | Yes | |
NAUAIDYHJRWZDQ
|
7.7 | IC50 | 3 | Yes | |
PZJJOMPTIHBGHO
|
7.7 | IC50 | 8 | Yes | |
RPNGFLLEKVAIHJ
|
7.7 | IC50 | 4 | Yes | |
SVDCGRYSXBTBBO
|
7.7 | IC50 | 3 | Yes | |
UCKDGXYIQSPPDL
|
7.7 | IC50 | 5 | Yes | |
UIODHSBHBXTRBO
|
7.7 | IC50 | 3 | Yes | |
UNQHIMAGAUGZGX
|
7.7 | IC50 | 5 | Yes | |
XVUIGVGFVWRFJO
|
7.7 | Ki | 8 | Yes | |
YWWJREBSMRNZGO
|
7.7 | IC50 | 3 | Yes | |
ZVJILQAAQQNBOP
|
7.7 | IC50 | 6 | — | |
BLVTYAOGMSRRPZ
|
7.7 | IC50 | 3 | Yes | |
CQIQKDQFHVTTKM
|
7.7 | IC50 | 5 | Yes | |
CQIQKDQFHVTTKM
|
7.7 | IC50 | 5 | Yes | |
CZYVJSTWDMVAFM
|
7.7 | IC50 | 6 | Yes | |
DZOZBHZWCFMSKH
|
7.7 | IC50 | 4 | Yes | |
GTRSMAWFAMXNCF
|
7.7 | IC50 | 6 | Yes | |
GWEITLSXCOXESW
|
7.7 | IC50 | 7 | Yes | |
IRBWGGQXMBAYQL
|
7.7 | IC50 | 7 | Yes | |
JQGYJNKTRDAQCV
|
7.7 | IC50 | 5 | Yes | |
JRCGNOYYZQLNTH
|
7.7 | Ki | 11 | Yes |