Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CYVZQRKPMGDNKM
|
7.8 | IC50 | 4 | Yes | |
FPHZWTIGUNTHAS
|
7.8 | IC50 | 3 | — | |
HIWQTXDWQYKMGH
|
7.8 | Ki | 7 | Yes | |
HZTQDRLCDGHQSA
|
7.8 | IC50 | 5 | Yes | |
IXHBDLPZTUSLFD
|
7.8 | Ki | 5 | — | |
JENVXNLJMJTTNA
|
7.8 | IC50 | 3 | Yes | |
SPZLSWDAZSYJAK
|
7.8 | IC50 | 2 | — | |
UGBFTDFVLBACAS
|
7.8 | Ki | 7 | Yes | |
UJKQHAYQMMMAEL
|
7.8 | Ki | 7 | Yes | |
WNLZTTHHHYZJMB
|
7.8 | IC50 | 9 | Yes | |
YTELTZFLAYFFDQ
|
7.8 | IC50 | 3 | Yes | |
YTQZUTBYXGOMDQ
|
7.8 | IC50 | 2 | Yes | |
ZVFJPOKDCLPATG
|
7.8 | IC50 | 4 | Yes | |
BCOFTFDFNHXYGF
|
7.8 | IC50 | 5 | Yes | |
DFPDFXUEOXPMIV
|
7.8 | Ki | 7 | Yes | |
FOTKISDMFBTXGP
|
7.8 | IC50 | 3 | — | |
GJOCABIDMCKCEG
|
7.8 | IC50 | 5 | Yes | |
JQVXQUOPUHBHAD
|
7.8 | IC50 | 5 | Yes | |
JTLSDSKNFBJVAB
|
7.8 | IC50 | 3 | Yes | |
MZISFPSOTJFTTJ
|
7.8 | Ki | 7 | Yes | |
NAVKLAFIVRMQMW
|
7.8 | IC50 | 5 | Yes | |
NYEXRVCCRODWLT
|
7.8 | IC50 | 5 | Yes | |
SSFOEYVZLXDDTG
|
7.8 | IC50 | 7 | Yes | |
UMBHCIONUFCHIP
|
7.8 | IC50 | 5 | Yes | |
VIZCCTVYPJKZBP
|
7.8 | IC50 | 3 | — | |
YDDMVPLLJTZTQL
|
7.8 | Ki | 7 | Yes | |
YHTDLXCRQOJRHH
|
7.8 | IC50 | 5 | Yes | |
YTQYMJLEQVXIPD
|
7.8 | Ki | 4 | — | |
ZGWIOFHKEXLJPC
|
7.8 | IC50 | 5 | Yes | |
MDMQULYGCYNXQN
|
7.8 | Ki | 6 | — | |
ZQUJAHCTHDEZMJ
|
7.8 | Ki | 6 | — | |
APKANDPILBIUDO
|
7.8 | IC50 | 5 | Yes | |
AXHCVGDTGFVLIU
|
7.8 | IC50 | 5 | Yes | |
BGDARAHTNRWTGV
|
7.8 | IC50 | 6 | Yes | |
DQDPBMDGDOPPLK
|
7.8 | Ki | 7 | Yes | |
HZWSSUJZEMEIID
|
7.8 | IC50 | 5 | Yes | |
IINBMMZSLVIMTL
|
7.8 | IC50 | 5 | Yes | |
KJFHTZIVTSKATM
|
7.8 | IC50 | 5 | Yes | |
LMSMOBVZXAUSAU
|
7.8 | IC50 | 4 | Yes | |
QMJIUHKQZQSTQO
|
7.8 | IC50 | 3 | Yes | |
WLZQVNRDQZYTID
|
7.8 | Ki | 6 | — | |
WYWVSRVZNIIISU
|
7.8 | IC50 | 7 | Yes | |
XCCIACQOXSWRJQ
|
7.8 | Ki | 7 | Yes | |
YPTZORUBNMNKDA
|
7.8 | IC50 | 2 | — | |
ZGSTVUAZFACDLH
|
7.8 | Ki | 8 | Yes | |
ZJVORNZEDYXDGJ
|
7.8 | IC50 | 4 | — | |
ZSRPSCNAFVEYRR
|
7.8 | IC50 | 4 | Yes | |
ZWHIVWLHYJCFFA
|
7.8 | IC50 | 5 | Yes | |
UTSFQPTVPZNJJH
|
7.8 | IC50 | 7 | Yes | |
BITXXJKMASUYME
|
7.8 | Ki | 7 | Yes |