Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CADOQGNFDXDEHI
|
9.7 | IC50 | 5 | Yes | |
IBRCQOLHLBIVAH
|
9.7 | IC50 | 5 | Yes | |
JATUSZYMCBLDQS
|
9.7 | IC50 | 8 | Yes | |
ORSWNUGKUNQTLF
|
9.7 | IC50 | 7 | Yes | |
OXTBPBSHWBJLJN
|
9.7 | IC50 | 4 | — | |
PCOMQZCYLOTKTN
|
9.7 | IC50 | 5 | Yes | |
PNOYLKIRWUYKLC
|
9.7 | IC50 | 4 | — | |
QDGVTWBFTFHWOG
|
9.7 | IC50 | 8 | Yes | |
SFESNYSPTLYJFZ
|
9.7 | IC50 | 6 | Yes | |
UIGGXLFLAQCMAY
|
9.7 | IC50 | 6 | Yes | |
WVUXCTUJEGJKKV
|
9.7 | IC50 | 5 | Yes | |
XAOJSOMIBKILNZ
|
9.7 | IC50 | 5 | Yes | |
XIOQDQAMCAXVAV
|
9.7 | IC50 | 5 | Yes | |
XXKPJSZGWAMVSD
|
9.7 | Ki | 3 | — | |
YBRVBUDXSMPLGQ
|
9.7 | IC50 | 5 | Yes | |
YDYDCNNQCGFQDL
|
9.7 | Ki | 5 | — | |
YKPYIPVDTNNYCN
|
9.7 | IC50 | 11 | Yes | |
YPRABBTWBDZWGP
|
9.7 | IC50 | 4 | Yes | |
QYCUMAKSYBUWER
|
9.7 | Ki | 6 | — | |
UGWWPGUNBPZMDD
|
9.6 | IC50 | 5 | — | |
NEPHXSICDJEKLG
|
9.6 | IC50 | 6 | — | |
ASZIRMQBBYBMMU
|
9.6 | IC50 | 7 | Yes | |
DZCKADUBMZPQDB
|
9.6 | Ki | 3 | — | |
PGEMRSCSFPLCBF
|
9.6 | IC50 | 8 | Yes | |
SIEIWCDBNIGNIG
|
9.6 | IC50 | 7 | Yes | |
SPEYRVQKGFNUCY
|
9.6 | IC50 | 8 | Yes | |
WVPKYEATTXWJLC
|
9.6 | IC50 | 5 | — | |
VKESMHHXVWGWQQ
|
9.6 | IC50 | 2 | — | |
FOVJQTLLPOZKTJ
|
9.5 | IC50 | 4 | — | |
BKIYUSXBJJEODV
|
9.5 | IC50 | 7 | Yes | |
CFUZFFCLLPGACM
|
9.5 | IC50 | 3 | — | |
FAOIZSVKMZLOCI
|
9.5 | Ki | 2 | — | |
FQPCVUZCOHLRGT
|
9.5 | Ki | 2 | — | |
GDBQQVUOBJAORI
|
9.5 | IC50 | 3 | — | |
JMKHBHJIGFWJPF
|
9.5 | IC50 | 5 | — | |
JRJPXBUCHQFJHU
|
9.5 | IC50 | 6 | Yes | |
NGILBKZKRQUURV
|
9.5 | IC50 | 5 | Yes | |
OCZKLINSAMKTBK
|
9.5 | IC50 | 7 | Yes | |
OMKBGTGZWMRDAZ
|
9.5 | IC50 | 3 | Yes | |
PKAAOTCIUWGSDS
|
9.5 | IC50 | 6 | Yes | |
QJNGNVJSSUXWBO
|
9.5 | IC50 | 8 | Yes | |
STMMWXRQAOVQNP
|
9.5 | IC50 | 5 | Yes | |
TWPPWHMOPIWZMY
|
9.5 | IC50 | 5 | Yes | |
UDYKJHQVNSKFHV
|
9.5 | IC50 | 4 | Yes | |
UXOSVQFKXFZCKF
|
9.5 | IC50 | 3 | Yes | |
VPXAENCQUJDPFF
|
9.5 | IC50 | 4 | — | |
WUGYYDAXBPEKAI
|
9.5 | IC50 | 4 | — | |
XMVQXBAGOTVZDD
|
9.5 | IC50 | 4 | — | |
YBQPTPBTTDQLMD
|
9.5 | IC50 | 4 | — | |
YLRBOIVJMWEGGX
|
9.5 | Ki | 6 | — |