Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JOMDWNBZLUPPTA
|
8.0 | IC50 | 3 | Yes | |
KLCHUAUMSZUJEX
|
8.0 | IC50 | 5 | Yes | |
KRUUUOUZTDKUCF
|
8.0 | IC50 | 5 | Yes | |
LMASIGSKSCEZDY
|
8.0 | IC50 | 5 | Yes | |
LYVGWVHFXOYMDJ
|
8.0 | IC50 | 6 | Yes | |
MMJPVSDTLGFIQW
|
8.0 | IC50 | 2 | Yes | |
MZIZOOUSSMSGAV
|
8.0 | IC50 | 5 | Yes | |
NPMTYGOUEKCULB
|
8.0 | IC50 | 5 | Yes | |
NSDMBIOAMTZMED
|
8.0 | IC50 | 5 | Yes | |
PCQHVURJJBFBQG
|
8.0 | Ki | 7 | Yes | |
PHKLGXHLOXCURO
|
8.0 | IC50 | 4 | — | |
RMIHUCKIXBQQLS
|
8.0 | IC50 | 5 | Yes | |
RQEBSVZFRXVOLZ
|
8.0 | IC50 | 5 | Yes | |
RWVGBBDAACKFOR
|
8.0 | IC50 | 3 | Yes | |
SHBOXSNAYNDDGN
|
8.0 | IC50 | 2 | — | |
TWXMFJCBMYOHKC
|
8.0 | IC50 | 3 | Yes | |
UGZOJBSDACNWAB
|
8.0 | Ki | 7 | Yes | |
XBLZKAPRZBJHCZ
|
8.0 | IC50 | 5 | Yes | |
XOYCZHYJWUFTBH
|
8.0 | IC50 | 4 | Yes | |
ZMAQPMCPZORBHF
|
8.0 | IC50 | 5 | Yes | |
ATIAZZHHFGJINP
|
8.0 | IC50 | 3 | Yes | |
XZDDXHHQKBWEQB
|
8.0 | IC50 | 3 | Yes | |
ZUGWYJYJZWGIPG
|
7.9 | IC50 | 2 | — | |
QKYPFBUZQDJQHX
|
7.9 | IC50 | 6 | Yes | |
AARSEFXVCWMMKV
|
7.9 | IC50 | 2 | — | |
AUCTYKZCPSWUEL
|
7.9 | IC50 | 5 | Yes | |
BEZJPBNIFWANDL
|
7.9 | IC50 | 2 | — | |
BKJCTJQMBGJOHN
|
7.9 | IC50 | 5 | Yes | |
FPRHOXXDKHGHSY
|
7.9 | IC50 | 3 | Yes | |
HSJPSXSXQYYJSY
|
7.9 | Ki | 7 | Yes | |
IWTGCCHOUSDKHV
|
7.9 | Ki | 10 | Yes | |
KQEHQRICYJKJLB
|
7.9 | IC50 | 6 | Yes | |
LMKSZZKXCRCXFM
|
7.9 | Ki | 3 | — | |
NKRKWSFHPLAZOP
|
7.9 | IC50 | 7 | Yes | |
PSLXIIKDHBIITK
|
7.9 | IC50 | 3 | Yes | |
RIYWMJMELHHCTR
|
7.9 | IC50 | 2 | — | |
SMUHFCXUZGSRMF
|
7.9 | IC50 | 3 | Yes | |
SQKUIDNBYAHJQB
|
7.9 | IC50 | 5 | — | |
TWQZYQBXMVVVCY
|
7.9 | IC50 | 7 | Yes | |
TWQZYQBXMVVVCY
|
7.9 | IC50 | 7 | Yes | |
TWQZYQBXMVVVCY
|
7.9 | IC50 | 6 | Yes | |
UALGGXUAYUNRBS
|
7.9 | Ki | 7 | Yes | |
UGMRVUAZVAXFHK
|
7.9 | Ki | 8 | Yes | |
UPNGQGNTHSPTJW
|
7.9 | IC50 | 3 | Yes | |
VKCIBOBTIOCYLR
|
7.9 | IC50 | 5 | Yes | |
VMCQYTNLTZJCIG
|
7.9 | IC50 | 5 | Yes | |
WEACEEZKOJLZFG
|
7.9 | Ki | 7 | Yes | |
WLJUNQUGIMIQDZ
|
7.9 | IC50 | 4 | Yes | |
WPXAJFJACNOICK
|
7.9 | Ki | 7 | Yes | |
XUBGKCSUKRWGIB
|
7.9 | IC50 | 3 | Yes |