Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GXOXVMQTJCQLGA
|
8.0 | IC50 | 3 | Yes | |
OYJHJMVVIQMCQV
|
8.0 | IC50 | 2 | — | |
RQCBSNJRFVZHOS
|
8.0 | IC50 | 10 | Yes | |
HYBHKZKKEGAPOP
|
8.0 | IC50 | 6 | — | |
SJVJJZDVWOYTNM
|
8.0 | IC50 | 3 | Yes | |
ZXSHUUVACBVHFP
|
8.0 | IC50 | 3 | Yes | |
BDWCIDSXORGMEX
|
8.0 | IC50 | 3 | Yes | |
COUUBDFXGTZTPW
|
8.0 | Ki | 5 | Yes | |
DMOIDCGAIGWXGJ
|
8.0 | Ki | 7 | Yes | |
IHPUTEIJIZVYPC
|
8.0 | Ki | 7 | Yes | |
IQFZAFZQQFAEFD
|
8.0 | IC50 | 4 | Yes | |
JLXRKMSJFVPFIG
|
8.0 | IC50 | 4 | — | |
KJOVWWTWOVUHSB
|
8.0 | IC50 | 5 | Yes | |
KOFNJKLYWDTWHZ
|
8.0 | Ki | 7 | Yes | |
LBKCSOUMADYGHM
|
8.0 | IC50 | 6 | Yes | |
NJSAPXUDAYVTFL
|
8.0 | Ki | 7 | Yes | |
OKYUILRERWOFCH
|
8.0 | IC50 | 7 | Yes | |
PEDLXNUHJRCVGF
|
8.0 | IC50 | 3 | Yes | |
PLJKONSYASWBHO
|
8.0 | Ki | 3 | — | |
SESYXDSEOCRODR
|
8.0 | Ki | 7 | Yes | |
UJVIDDIDLMDARE
|
8.0 | IC50 | 4 | Yes | |
ULPVLGUDYQAPPV
|
8.0 | Ki | 7 | Yes | |
UOHZYJYLFKMPMQ
|
8.0 | Ki | 7 | Yes | |
UTERPWJSMDDIGY
|
8.0 | Ki | 8 | Yes | |
VLTOUUSTKONGKC
|
8.0 | Ki | 10 | Yes | |
VYAMAYOVUONCDB
|
8.0 | IC50 | 2 | — | |
WDMMHRSZAREYDM
|
8.0 | IC50 | 2 | — | |
WGTWQHQAJDQPEW
|
8.0 | IC50 | 5 | Yes | |
WICQDDCNCVTFDX
|
8.0 | Ki | 16 | Yes | |
WPYFTDWGMAINBU
|
8.0 | IC50 | 5 | Yes | |
XNKSQYFVFJZMOA
|
8.0 | IC50 | 7 | Yes | |
XYXRFODFDUOQKS
|
8.0 | Ki | 3 | — | |
YJBLORWBSQLNFW
|
8.0 | IC50 | 4 | Yes | |
YTIQSKPYJKROHS
|
8.0 | IC50 | 2 | — | |
YTQYMJLEQVXIPD
|
8.0 | Ki | 4 | — | |
ZZVSRSRVYMQUCW
|
8.0 | IC50 | 6 | Yes | |
OUZMHHWAGJCAFA
|
8.0 | Ki | 8 | — | |
YEKVTHFNPVYQBX
|
8.0 | IC50 | 5 | Yes | |
AYTZJEWKGLEPFF
|
8.0 | IC50 | 4 | — | |
CBLOGBROLDHLEE
|
8.0 | IC50 | 6 | Yes | |
DUCBSHDQTBWWLC
|
8.0 | Ki | 7 | Yes | |
FSVPEOOPDJVOOW
|
8.0 | IC50 | 3 | Yes | |
FTWZRZIOCFAVKU
|
8.0 | IC50 | 5 | Yes | |
FXZROVPZUUATHR
|
8.0 | IC50 | 4 | Yes | |
HESIRWKKCVPIEN
|
8.0 | IC50 | 3 | Yes | |
HIYYLOFJQXHPRU
|
8.0 | IC50 | 5 | Yes | |
HMXFQXRHTFBPFX
|
8.0 | IC50 | 4 | — | |
HVGJVSYGPSRPHL
|
8.0 | IC50 | 5 | Yes | |
ISONEAYXNYSTJQ
|
8.0 | IC50 | 5 | Yes | |
IXEFVZDHNHSUSD
|
8.0 | IC50 | 5 | Yes |