Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BSIZUMJRKYHEBR
|
8.1 | IC50 | 15 | Yes | |
CDVYEYANHXGLCX
|
8.1 | Ki | 10 | Yes | |
FCGVXISUYVDDPU
|
8.1 | IC50 | 7 | Yes | |
GHHVNOZFZMDYFQ
|
8.1 | Ki | 7 | Yes | |
GJOCABIDMCKCEG
|
8.1 | IC50 | 6 | Yes | |
GOLRDGXHDIYHCN
|
8.1 | IC50 | 6 | Yes | |
HEJQAFMDGAOYSZ
|
8.1 | IC50 | 4 | Yes | |
IOQOIXCSRBBCDP
|
8.1 | IC50 | 3 | Yes | |
JKWHUKMFJPDCMY
|
8.1 | IC50 | 5 | Yes | |
KLRCKSDGEDNMNL
|
8.1 | IC50 | 4 | Yes | |
KNFQAZOHJDVGHS
|
8.1 | Ki | 5 | — | |
KSGNBXMXFPLVKJ
|
8.1 | IC50 | 3 | Yes | |
LJNWPYWHBAYDNO
|
8.1 | IC50 | 5 | Yes | |
LWZOHIDILGLXGF
|
8.1 | IC50 | 5 | Yes | |
MAVDNGWEBZTACC
|
8.1 | IC50 | 9 | Yes | |
MRBPTYYVXXZQBB
|
8.1 | IC50 | 5 | Yes | |
QAEKGVKCHDBGEN
|
8.1 | IC50 | 3 | Yes | |
RCSWIFOOANTXTQ
|
8.1 | IC50 | 3 | Yes | |
RKPWDSLUQARCLB
|
8.1 | IC50 | 5 | Yes | |
RMMYIAVIROFVLC
|
8.1 | IC50 | 4 | Yes | |
ZRDGYJAMDSHROJ
|
8.1 | IC50 | 7 | Yes | |
ZTVJLUOPMWIKSV
|
8.1 | IC50 | 6 | Yes | |
NVZOQOOLHGCJGV
|
8.1 | IC50 | 3 | Yes | |
UKBSDNIYHDAZDN
|
8.1 | IC50 | 3 | Yes | |
VAQVSMUJBPTVIS
|
8.1 | IC50 | 7 | Yes | |
YDCCHZDGDMSTQT
|
8.1 | IC50 | 5 | — | |
NVQQPOVAPJFBOD
|
8.1 | IC50 | 2 | — | |
BEKYMPWGANBKBK
|
8.1 | Ki | 7 | Yes | |
DOFYUNJDVUXVMB
|
8.1 | IC50 | 5 | Yes | |
DWBZTKJXPJGGSU
|
8.1 | IC50 | 6 | Yes | |
ISXZSJVTKFNYSR
|
8.1 | IC50 | 3 | Yes | |
JMTSRJRSBJJBGP
|
8.1 | IC50 | 6 | Yes | |
JMWYGNIQHYKDCH
|
8.1 | Ki | 7 | Yes | |
KASLMAICRUMQME
|
8.1 | IC50 | 5 | Yes | |
LEIFVUOVYOUZFH
|
8.1 | IC50 | 5 | Yes | |
RSMQCSLXBNSQJJ
|
8.1 | Ki | 7 | Yes | |
SHTYCRVVDNRZDY
|
8.1 | IC50 | 5 | Yes | |
WVNVANHURONWTG
|
8.1 | IC50 | 5 | Yes | |
XFCISDUWYSMJOU
|
8.1 | IC50 | 3 | Yes | |
XRGWUGBXRHDGDG
|
8.1 | IC50 | 6 | Yes | |
YPLGVMIJHPJLRA
|
8.1 | IC50 | 6 | Yes | |
YRUNEWMUGNJMAR
|
8.1 | Ki | 7 | Yes | |
YTTGWCXMRQNZJI
|
8.1 | IC50 | 5 | Yes | |
ZBIYSEFCPUXCRC
|
8.1 | IC50 | 5 | Yes | |
IGOVNBYALNSOHR
|
8.0 | IC50 | 3 | — | |
OJGIWNSVHKBBDS
|
8.0 | IC50 | 3 | Yes | |
YTCCTPYUECNUFO
|
8.0 | IC50 | 7 | Yes | |
BOXSOXSFZRZIAF
|
8.0 | IC50 | 3 | Yes | |
FFBVONWPZBISIM
|
8.0 | IC50 | 2 | — | |
ASLUWSDEBRNVJV
|
8.0 | IC50 | 6 | Yes |