Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CIOUXWQXQFITHV
|
8.2 | IC50 | 3 | — | |
CLTINYAXRIROMY
|
8.2 | IC50 | 5 | Yes | |
DCWUWJBJOHDJGB
|
8.2 | IC50 | 5 | Yes | |
DHMHJSLNCAYKRH
|
8.2 | IC50 | 5 | Yes | |
FJXZBLKBEVSCAB
|
8.2 | IC50 | 4 | Yes | |
FTFANCIOHXJKDG
|
8.2 | IC50 | 4 | Yes | |
GFUITADOEPNRML
|
8.2 | IC50 | 8 | Yes | |
GKHRDWHFKKUYAX
|
8.2 | Ki | 9 | — | |
GZQRNXJPJXICJZ
|
8.2 | IC50 | 4 | Yes | |
HKAXLEJIOVCYCD
|
8.2 | IC50 | 5 | Yes | |
ICSWIBNMQZLUKX
|
8.2 | IC50 | 3 | Yes | |
IVXFVTBAZBQGPK
|
8.2 | IC50 | 5 | Yes | |
LHUIUEQQDGBKCU
|
8.2 | IC50 | 5 | Yes | |
MIKGRMSWGTVOSA
|
8.2 | IC50 | 4 | — | |
NDHPESZMBIVDPO
|
8.2 | IC50 | 2 | — | |
NNUQGANTDABHBL
|
8.2 | IC50 | 3 | Yes | |
PYJCXRBSZSSHDD
|
8.2 | IC50 | 3 | Yes | |
QXMXXJUEHWZLCA
|
8.2 | IC50 | 3 | Yes | |
RCGPSTRFXVIUQB
|
8.2 | Ki | 7 | Yes | |
RPOHBDSRTDJNFN
|
8.2 | IC50 | 5 | Yes | |
SMZPWUUYPYYHIV
|
8.2 | IC50 | 5 | Yes | |
SQWPYMHLYZKCEN
|
8.2 | IC50 | 3 | — | |
SVUOUTRIPGSFHF
|
8.2 | IC50 | 5 | Yes | |
TUIHSDQRXNNCLL
|
8.2 | IC50 | 6 | Yes | |
USIMDPVZFWUXPH
|
8.2 | IC50 | 6 | Yes | |
UWHPJOBPMXNVII
|
8.2 | IC50 | 5 | Yes | |
VDJRMQXPNKTLQA
|
8.2 | IC50 | 5 | Yes | |
VVZTYGQJDUUATC
|
8.2 | IC50 | 7 | Yes | |
WFQFQAQNCYHBTC
|
8.2 | IC50 | 8 | Yes | |
WHHAEBOHMHRZGW
|
8.2 | IC50 | 4 | — | |
XAUUSUAZNMIGRK
|
8.2 | IC50 | 6 | Yes | |
XJFYJIMKKGZKGX
|
8.2 | IC50 | 6 | Yes | |
ZMAYDSCNOCAOHA
|
8.2 | IC50 | 5 | Yes | |
ZQORGANDVNQVJF
|
8.2 | Ki | 6 | Yes | |
CDYLCTGLLNQEQF
|
8.1 | IC50 | 5 | Yes | |
RPWGPXSVYLHGRZ
|
8.1 | IC50 | 7 | Yes | |
RTYBJAJUHLHGKX
|
8.1 | IC50 | 3 | — | |
ZAQHFZCMMMYWLV
|
8.1 | IC50 | 3 | Yes | |
BPNDGQNQHSBNOE
|
8.1 | IC50 | 7 | Yes | |
MEGFCBVTRXVKDO
|
8.1 | IC50 | 6 | Yes | |
HAWUDCIVXQTNAF
|
8.1 | IC50 | 3 | Yes | |
HYKTXCHYRXFJMV
|
8.1 | IC50 | 3 | Yes | |
JUCUDUBNTIXZOX
|
8.1 | IC50 | 3 | Yes | |
RTYBJAJUHLHGKX
|
8.1 | IC50 | 3 | — | |
YSLNEVXKZVORTK
|
8.1 | IC50 | 4 | Yes | |
YZKBLJHHYZDROJ
|
8.1 | IC50 | 4 | Yes | |
AANXPIMDONQTQF
|
8.1 | IC50 | 5 | Yes | |
AINJYWXKBKRQSX
|
8.1 | IC50 | 6 | Yes | |
AKTPDJLIUXRMDA
|
8.1 | IC50 | 5 | Yes | |
AYPPVQRNMZPQMU
|
8.1 | IC50 | 6 | Yes |