Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TXRXSTLBPVIGRX
|
8.2 | IC50 | 3 | — | |
OFXJMYWLEABUGO
|
8.2 | IC50 | 3 | Yes | |
QMJIUHKQZQSTQO
|
8.2 | IC50 | 3 | Yes | |
ASSONXJFMGBTAQ
|
8.2 | IC50 | 3 | Yes | |
ATNNMKHWMHMLHP
|
8.2 | Ki | 7 | Yes | |
BADHAWRYSSJDAG
|
8.2 | IC50 | 4 | Yes | |
CFEKPCYWRLBSBI
|
8.2 | IC50 | 6 | Yes | |
CXRZYJPQMZBWAW
|
8.2 | IC50 | 5 | Yes | |
DOZFSSIRRROWRF
|
8.2 | Ki | 3 | — | |
FMQWWPFJFLUCHZ
|
8.2 | IC50 | 6 | Yes | |
FPHXOEUJYCDFQF
|
8.2 | IC50 | 4 | Yes | |
GDXZUNJRYLVZAT
|
8.2 | IC50 | 4 | — | |
GWQPVXKPORBEIM
|
8.2 | IC50 | 5 | Yes | |
HEYGZWVOCCBCPY
|
8.2 | IC50 | 6 | Yes | |
HNXQLWUITFQYPE
|
8.2 | Ki | 10 | Yes | |
JAVKQWAQQAGPFN
|
8.2 | IC50 | 5 | Yes | |
JKMQHCXIFJQOMJ
|
8.2 | IC50 | 3 | Yes | |
LGJLWDFGIABLSI
|
8.2 | IC50 | 3 | — | |
LTTRJMCJTUBEGF
|
8.2 | IC50 | 4 | — | |
MDWFJTBWOFNAQX
|
8.2 | IC50 | 7 | Yes | |
PPTJZFSGDMWVFF
|
8.2 | IC50 | 5 | Yes | |
ROMGJVVZNVJOPW
|
8.2 | Ki | 10 | Yes | |
SHMJSERYBLZGBT
|
8.2 | IC50 | 3 | Yes | |
SNYKGOMEURTYMK
|
8.2 | Ki | 10 | Yes | |
VRUQYJXYEALKCT
|
8.2 | IC50 | 6 | Yes | |
VURZBHKGMIEEFK
|
8.2 | Ki | 7 | Yes | |
WJPFHUMULGZBAI
|
8.2 | IC50 | 4 | Yes | |
ZACZGYFEWPTMFL
|
8.2 | IC50 | 2 | — | |
ZGSTVUAZFACDLH
|
8.2 | IC50 | 7 | — | |
ZQENIBLYGGLKSO
|
8.2 | IC50 | 5 | Yes | |
AQVWDVBVCMNHDC
|
8.2 | IC50 | 5 | Yes | |
JWILGVWCZHAXFQ
|
8.2 | IC50 | 3 | Yes | |
RVBSKRBWGPIJIS
|
8.2 | IC50 | 3 | Yes | |
SAXMIJMROZDLCS
|
8.2 | IC50 | 3 | Yes | |
ZHXMXRVBOZWQPF
|
8.2 | IC50 | 5 | Yes | |
FECFHXJGVVXRMZ
|
8.2 | IC50 | 3 | Yes | |
FQRZOEBSTPAQBJ
|
8.2 | IC50 | 4 | — | |
ITQUODOQSFVYAA
|
8.2 | IC50 | 3 | Yes | |
MVPVFNYLHBJBHV
|
8.2 | IC50 | 5 | Yes | |
NSOWFDNMRUSVGR
|
8.2 | IC50 | 3 | Yes | |
QWBFNTUMBVGNBO
|
8.2 | IC50 | 3 | Yes | |
SQWPYMHLYZKCEN
|
8.2 | IC50 | 3 | — | |
AOBTZEZFLADCMR
|
8.2 | IC50 | 3 | Yes | |
DGNSDTQNQWONIY
|
8.2 | IC50 | 3 | Yes | |
FQMDDNHJAAIYKQ
|
8.2 | IC50 | 3 | Yes | |
WIAJGSYMEDWMGP
|
8.2 | IC50 | 5 | Yes | |
LFOGEPKUSWRLCL
|
8.2 | IC50 | 7 | Yes | |
SQWPYMHLYZKCEN
|
8.2 | IC50 | 3 | — | |
AWDZLFOJMUGNPS
|
8.2 | IC50 | 6 | Yes | |
BYFPJSOGSJVRJE
|
8.2 | IC50 | 5 | Yes |