Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SMAMMQUTTZLMCT
|
8.4 | IC50 | 3 | Yes | |
BVVZNDQVRQLIPW
|
8.4 | IC50 | 4 | Yes | |
CBDXJWSRGWXYPR
|
8.4 | IC50 | 5 | Yes | |
CCGWFLCBYDXLBZ
|
8.4 | IC50 | 5 | Yes | |
CLPQPSHMBDAYLR
|
8.4 | IC50 | 6 | Yes | |
FBLQAKOTTHGGBJ
|
8.4 | IC50 | 4 | Yes | |
GCDCQOTVUSLXRJ
|
8.4 | IC50 | 4 | Yes | |
GFDLNQRSUGRRNQ
|
8.4 | IC50 | 6 | Yes | |
GKLOCXVNLLEZMX
|
8.4 | IC50 | 4 | — | |
GTOFARSZXYDPTC
|
8.4 | IC50 | 5 | Yes | |
GTXSRFUZSLTDFX
|
8.4 | IC50 | 5 | — | |
JRKVJTDYMGJJAK
|
8.4 | IC50 | 6 | Yes | |
LNJYGNLGJFKFCM
|
8.4 | IC50 | 5 | Yes | |
MWNWUYJAANVQLN
|
8.4 | IC50 | 6 | Yes | |
NGEXELWTFRTJEQ
|
8.4 | IC50 | 5 | Yes | |
NHIGQLZDIAMPEX
|
8.4 | IC50 | 3 | — | |
NZVNFHULUBKMQI
|
8.4 | IC50 | 4 | Yes | |
OMMFNEZCURCLPN
|
8.4 | IC50 | 6 | Yes | |
PKYBEORBMGUOOP
|
8.4 | IC50 | 4 | Yes | |
PPCHUKYNNDWTFT
|
8.4 | IC50 | 3 | — | |
QOWJHUFMPPFELP
|
8.4 | IC50 | 4 | Yes | |
QXMQRADDQYZCBO
|
8.4 | IC50 | 5 | Yes | |
QYEGLTVXUKXPSD
|
8.4 | IC50 | 4 | Yes | |
RUZDCFCMYATJSO
|
8.4 | IC50 | 5 | Yes | |
VSZRGCMKCYLOIV
|
8.4 | IC50 | 4 | Yes | |
WUQMFARMJJXJMN
|
8.4 | IC50 | 6 | Yes | |
YQCWPKHRHVYSBQ
|
8.4 | IC50 | 6 | Yes | |
YZCLZWVHSZUTMP
|
8.4 | IC50 | 5 | Yes | |
DGZZVIWCMGVHGV
|
8.4 | IC50 | 11 | Yes | |
SLUQTAQKAIYNRS
|
8.4 | IC50 | 3 | Yes | |
VPTHOUBPDJAAER
|
8.4 | IC50 | 6 | Yes | |
YOMXWXIANUYIMH
|
8.4 | IC50 | 10 | Yes | |
RAGDORVOHODYFH
|
8.4 | Ki | 4 | Yes | |
VKFNDAOTTJONML
|
8.4 | IC50 | 9 | Yes | |
YWZUYEWFBPKKSJ
|
8.4 | IC50 | 6 | Yes | |
JJTWKBAUPPWAGL
|
8.4 | IC50 | 4 | Yes | |
QEWCDBOSGBDOOY
|
8.4 | IC50 | 5 | Yes | |
RRETZYBLLSHELY
|
8.4 | IC50 | 6 | Yes | |
RVXGDNRYPJLPKA
|
8.4 | IC50 | 3 | Yes | |
CNVJYZPKUZXAML
|
8.4 | IC50 | 4 | Yes | |
FWJQSGAFJBBJTH
|
8.4 | IC50 | 4 | Yes | |
UJUNISWMIDZDSX
|
8.4 | IC50 | 5 | Yes | |
WBEADJIJDUXNQI
|
8.4 | IC50 | 3 | — | |
XFAVBLSYPFKCGW
|
8.4 | IC50 | 3 | Yes | |
QMHSEIOSCQWTPQ
|
8.3 | IC50 | 6 | Yes | |
VGXYGECPCDQSNI
|
8.3 | IC50 | 6 | Yes | |
WHTRIFCXCJYQKX
|
8.3 | IC50 | 3 | Yes | |
WHTRIFCXCJYQKX
|
8.3 | IC50 | 5 | Yes | |
BFMSCDGDXHTNEA
|
8.3 | IC50 | 3 | Yes | |
NUFBSNVYZRUJSW
|
8.3 | IC50 | 6 | — |