Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QDJTVBZWIYKRMZ
|
8.5 | IC50 | 6 | Yes | |
RHTOEITZKIINCY
|
8.5 | IC50 | 6 | Yes | |
RRSNDPJAXNKWJB
|
8.5 | IC50 | 5 | Yes | |
RSGVYIJLQVPSNJ
|
8.5 | IC50 | 4 | Yes | |
SBPPAFQZTZUQSW
|
8.5 | IC50 | 4 | Yes | |
SEFCVQRMTNTWJO
|
8.5 | IC50 | 6 | Yes | |
UTCUOTDVVXFCLJ
|
8.5 | IC50 | 6 | Yes | |
UTDYWIPXAVCYCE
|
8.5 | IC50 | 5 | Yes | |
WXPUJRINFGPEGC
|
8.5 | IC50 | 3 | Yes | |
XSGJDCITTFQFMZ
|
8.5 | IC50 | 6 | Yes | |
XXNCZTSFXIANIO
|
8.5 | IC50 | 7 | Yes | |
YJKZJSXUMXIJNB
|
8.5 | Ki | 3 | — | |
YJOSMOCGEMCNLK
|
8.5 | IC50 | 6 | Yes | |
ZMVFZGHWXXXQJL
|
8.5 | IC50 | 6 | Yes | |
ZYBCZOFEUHHWME
|
8.5 | IC50 | 6 | Yes | |
BRYABXWERJYEAH
|
8.5 | IC50 | 3 | Yes | |
DRINIAFHXKEERM
|
8.5 | IC50 | 5 | Yes | |
FQEZYKOXVAISOF
|
8.5 | IC50 | 3 | Yes | |
FSSPDFKSDKXWQO
|
8.5 | IC50 | 3 | Yes | |
ICCZTDHQUXGJEO
|
8.5 | IC50 | 3 | Yes | |
JIRXORZYIXSWOB
|
8.5 | IC50 | 11 | Yes | |
BCNQQPWDHJUQFQ
|
8.5 | IC50 | 3 | Yes | |
FKPCCEUCLYUJQA
|
8.5 | IC50 | 6 | Yes | |
OIZMOMFOLNBXHF
|
8.5 | IC50 | 9 | — | |
XOOXBIFEOHDRHE
|
8.5 | IC50 | 6 | Yes | |
XTRLBSLKNQZDBD
|
8.5 | IC50 | 3 | Yes | |
CJTUBZULFXKTAT
|
8.5 | IC50 | 10 | Yes | |
CLXRDURJLYSMHZ
|
8.5 | IC50 | 5 | Yes | |
HUDBGKUNLWLMCD
|
8.5 | IC50 | 2 | — | |
IVPPTWCRAFCOFJ
|
8.5 | IC50 | 5 | — | |
UWCWCXPWHSKCKX
|
8.5 | IC50 | 3 | Yes | |
ZHLANTZRDCBWFM
|
8.5 | IC50 | 6 | Yes | |
ZVKAVYCKILWYEA
|
8.5 | IC50 | 4 | Yes | |
GRSFKJZRDUZQPW
|
8.5 | IC50 | 9 | Yes | |
HHHAELOQIYTSIY
|
8.5 | IC50 | 3 | Yes | |
LOMOBWUKCBVLNJ
|
8.5 | IC50 | 5 | Yes | |
ODOUKZOJMQSYME
|
8.5 | IC50 | 2 | — | |
YUWSFQQPCKKPJG
|
8.5 | IC50 | 9 | Yes | |
FAJZOFHZLDUFEM
|
8.4 | Ki | 6 | Yes | |
KEWGKOQZKWDXBX
|
8.4 | IC50 | 7 | Yes | |
NYACXZAKXKSUHM
|
8.4 | IC50 | 3 | Yes | |
RODBIJLXINIENS
|
8.4 | IC50 | 3 | Yes | |
FVPQYGSYGOKFLW
|
8.4 | Ki | 5 | Yes | |
KNWGEVZOUCQOLE
|
8.4 | IC50 | 3 | Yes | |
ZPNXAVJYHSAOKF
|
8.4 | IC50 | 7 | Yes | |
LRMGKWDRORXPRE
|
8.4 | IC50 | 5 | Yes | |
LZYKHUZBVFGWCA
|
8.4 | IC50 | 3 | Yes | |
MVTUAPMXVXQWFM
|
8.4 | IC50 | 3 | Yes | |
MVTUAPMXVXQWFM
|
8.4 | IC50 | 5 | Yes | |
FBLGEUMPZQFQFF
|
8.4 | IC50 | 2 | — |