Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HJFONKSERLWIGE
|
8.6 | IC50 | 3 | Yes | |
HOSYCMQDQLQXLY
|
8.6 | IC50 | 2 | — | |
WWNOVCQMRIZSRV
|
8.6 | IC50 | 8 | Yes | |
XJMDDZUUIUEEJH
|
8.6 | Ki | 5 | — | |
JGGFVHVZVBWBKF
|
8.6 | Ki | 4 | Yes | |
NHBOIMAIUCLQKQ
|
8.6 | IC50 | 4 | Yes | |
OTYJRWAMIOUIHN
|
8.6 | IC50 | 4 | Yes | |
QQDWEVONJRXVDB
|
8.6 | Ki | 6 | Yes | |
RMKNDVDQYWXAON
|
8.6 | IC50 | 7 | Yes | |
SXSIQUOYBXOPSS
|
8.6 | IC50 | 7 | Yes | |
GUHYZHHGWPARCR
|
8.6 | IC50 | 6 | Yes | |
IYWLZQLIFMUDCK
|
8.6 | IC50 | 5 | Yes | |
JAKYATQFPKVBNE
|
8.6 | IC50 | 5 | Yes | |
KHZOOCSTBFXVQU
|
8.6 | IC50 | 3 | Yes | |
LQRPHHDGTPYXHT
|
8.6 | IC50 | 5 | Yes | |
MAGDFYDBVAIRMV
|
8.6 | IC50 | 3 | — | |
CCVGKLVIMFBNBM
|
8.5 | IC50 | 5 | Yes | |
JNCKLKQBIMZPBF
|
8.5 | IC50 | 4 | Yes | |
JOOOUNMUHMUOJH
|
8.5 | IC50 | 3 | Yes | |
YNIHTMMJQXUNPE
|
8.5 | Ki | 7 | Yes | |
AFHDVSQBDWGAQU
|
8.5 | IC50 | 5 | Yes | |
AJUUQAWYLUYLDD
|
8.5 | IC50 | 6 | Yes | |
APXZBXMVEOBZDS
|
8.5 | IC50 | 2 | — | |
AWRGYKCXXWRYTJ
|
8.5 | IC50 | 4 | — | |
BDPAGEAOFNRCNJ
|
8.5 | IC50 | 4 | — | |
BGWGORXFGYPUAF
|
8.5 | IC50 | 5 | Yes | |
BLYHHTXBRXLLOI
|
8.5 | IC50 | 7 | Yes | |
CBFHYDZLOMACOM
|
8.5 | IC50 | 6 | Yes | |
CVZIHNYAZLXRRS
|
8.5 | IC50 | 10 | Yes | |
CVZIHNYAZLXRRS
|
8.5 | IC50 | 6 | Yes | |
DDFFKEPNXVTRCY
|
8.5 | IC50 | 4 | Yes | |
GBGAKFWYCGVPHY
|
8.5 | IC50 | 7 | Yes | |
GFUITADOEPNRML
|
8.5 | Ki | 6 | — | |
GFUITADOEPNRML
|
8.5 | Ki | 11 | Yes | |
GXFNBOPPVZGKBI
|
8.5 | IC50 | 3 | Yes | |
HDOJQDDADGGFGH
|
8.5 | IC50 | 6 | Yes | |
JIYWMQDJGOAJMD
|
8.5 | IC50 | 6 | Yes | |
KGVROUUAKSRCEI
|
8.5 | IC50 | 6 | Yes | |
KQYGUXCNMQFLRN
|
8.5 | IC50 | 5 | Yes | |
KSLUOGMHCJCRLQ
|
8.5 | IC50 | 6 | Yes | |
KWWNNPAPYSJGQH
|
8.5 | IC50 | 6 | Yes | |
MQDWBVIPJPRWIJ
|
8.5 | IC50 | 6 | Yes | |
MRJCPNBIHXIUFQ
|
8.5 | IC50 | 3 | Yes | |
MWYSQPGMUZLIHV
|
8.5 | Ki | 6 | Yes | |
NBBPYGNNDFCNNP
|
8.5 | IC50 | 5 | Yes | |
NVAYQDCPVGCOHV
|
8.5 | Ki | 5 | Yes | |
OJLWCTMBGWSVFC
|
8.5 | IC50 | 6 | Yes | |
PRBMKJZQAUSBQV
|
8.5 | IC50 | 6 | Yes | |
PRCRNUDMWULKSO
|
8.5 | IC50 | 7 | Yes | |
QAFRSDWNZLQCBN
|
8.5 | IC50 | 6 | Yes |