Target Details
| UniProt AC | P45452 |
|---|---|
| Gene Symbol | MMP13 |
| Protein Name | Collagenase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,949
- Clinical molecules 1414
- Avg pChEMBL 7.87
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (1,949)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IWQSGINKBSWILJ
|
11.5 | IC50 | 10 | — | |
YNHGVYGMFAREOF
|
11.4 | IC50 | 3 | — | |
LOPZANGJCBIBLO
|
11.2 | IC50 | 4 | — | |
VBMQORMYXJZHKU
|
11.1 | Ki | 2 | — | |
VGAPHGIXAQRVAL
|
10.8 | IC50 | 7 | Yes | |
FGQWFLDBWZDRJJ
|
10.7 | IC50 | 4 | — | |
DACARRUBIAXSBX
|
10.5 | IC50 | 2 | — | |
WIUDGBCTJVXBCM
|
10.5 | IC50 | 7 | — | |
WPZMNBVWWODJJH
|
10.5 | IC50 | 4 | — | |
MLUCCAMJMIYYED
|
10.4 | IC50 | 3 | — | |
NRRIJAHIBBGLNH
|
10.4 | IC50 | 4 | — | |
NTDGKPHATDVYNT
|
10.4 | IC50 | 4 | — | |
ZXGBSFAKYZEOPJ
|
10.4 | IC50 | 4 | — | |
MFOJAATVHNHXKB
|
10.3 | IC50 | 4 | — | |
ZTWMNQMJFNKJFV
|
10.3 | IC50 | 3 | Yes | |
HXZPYZWICHZKRL
|
10.3 | IC50 | 10 | — | |
JGWTVBVOISUVJD
|
10.3 | IC50 | 9 | — | |
BGKNBDGHNBOSGD
|
10.2 | IC50 | 3 | — | |
BGKNBDGHNBOSGD
|
10.2 | IC50 | 3 | — | |
UFKJDXKTPYNZRZ
|
10.2 | IC50 | 4 | — | |
GTZKIGXVCZWIAR
|
10.2 | IC50 | 4 | — | |
LXWCLFCLBYYKME
|
10.2 | IC50 | 4 | — | |
WTEZGXPTIFMTCH
|
10.2 | IC50 | 4 | — | |
XJNFMEAYBQFDAS
|
10.2 | IC50 | 4 | — | |
KLSPLBHGNYWPLX
|
10.1 | IC50 | 3 | — | |
SMKRBNFEFJZHAI
|
10.1 | IC50 | 4 | — | |
YDSGUUACYYBPLW
|
10.1 | IC50 | 4 | — | |
CMKYCYOBCXIZPF
|
10.0 | IC50 | 4 | — | |
DJEDDHGTONHFQL
|
10.0 | IC50 | 2 | — | |
LCYYUMHWMVOGPC
|
10.0 | IC50 | 8 | Yes | |
NBRBWZJMBITNBC
|
10.0 | IC50 | 8 | Yes | |
NUTUARVYQWFZAA
|
10.0 | IC50 | 6 | Yes | |
QKOVHOITGZCHQW
|
10.0 | IC50 | 4 | Yes | |
QVHYJMPAZNGFHN
|
10.0 | Ki | 6 | — | |
SFEPJGMZSMIONR
|
10.0 | IC50 | 7 | Yes | |
SWYRTBQMGJFWDS
|
10.0 | Ki | 3 | — | |
UBBBKPVDKLDZNE
|
10.0 | IC50 | 7 | Yes | |
UCWSKTMFEWSSSI
|
10.0 | IC50 | 4 | — | |
XMUJRKRMNALZLF
|
10.0 | IC50 | 2 | — | |
XQXSQQVRMVVPJW
|
10.0 | IC50 | 8 | Yes | |
YJRJYIQWWPZSTM
|
10.0 | IC50 | 6 | — | |
FMEMUXYNXWETSE
|
10.0 | IC50 | 6 | — | |
GSWRTFGMHRKLKT
|
9.9 | IC50 | 14 | Yes | |
MTRATHZFTCSGDT
|
9.9 | Ki | 6 | Yes | |
HBYRXCFAHCMHAA
|
9.8 | Ki | 9 | Yes | |
CUKATAAPVFYVIL
|
9.8 | IC50 | 9 | — | |
CDQRIIUMNLMHRH
|
9.7 | IC50 | 6 | — | |
WQCXDERWRJMJQA
|
9.7 | IC50 | 6 | — | |
AOPZFYOXZYZEAC
|
9.7 | IC50 | 7 | Yes | |
BDONYXHHXNTUSW
|
9.7 | IC50 | 8 | Yes |