Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
ILQGLXGUCRBEIV 7.6 Ki 2
QYFZGNQKVGYCKF 7.6 IC50 4
QYLKSFXBRALDIS 7.6 IC50 9
SESASZSELWFBAR 7.6 Ki 2
YAUZNKLMKRQDAM 7.6 Ki 7
NXIPMBQVNTWEEX 7.6 Ki 2
IEVJOUFGBRDCNE 7.6 Ki 2
JYUTVPNZUICOSN 7.6 Ki 2
QEMXHQIAXOOASZ 7.6 Ki 2
SMBPQHQVCQWZFD 7.6 Ki 2
JUOSGGQXEBBCJB 7.6 Ki 2
VLLKJTHFWNJPCE 7.6 IC50 9
WXFJHDPNAFRAND 7.6 Ki 2
FVFPYWYYJOGROX 7.6 IC50 4
PLQXXAVXCSTSDP 7.6 Ki 2
YRTJBUGCGGXTRV 7.6 IC50 5
LMURERRHDMDFGM 7.6 Ki 2
OWGALOIRPXUFMD 7.6 Ki 2
UBFYWPOOPLWTOY 7.6 Ki 2
YRVIKLBSVVNSHF 7.6 Ki 2
FEXICIZLMMJVEY 7.6 Ki 2
NSFPLWWBWPKKGV 7.6 Ki 2
VYJRBHHHDMICNS 7.6 IC50 4
DYIAIEHOHKXIMP 7.5 Ki 2
KPHRNXIFUJLFNL 7.5 Ki 5
PBDGFSBXTPVLEL 7.5 Ki 2
VPTXDMQKJHWYPV 7.5 IC50 4
MXUDEADPGZWZCH 7.5 IC50 9
MYKUKUCHPMASKF 7.5 Ki 2
MYKUKUCHPMASKF 7.5 Ki 3
QTFANGXLYPOILI 7.5 Ki 2
XHANNERZOZVNJM 7.5 Ki 2
GRIIGTWDNLOPDT 7.5 Ki 2
GTUIQNHJSXQMKW 7.5 Ki 3
LOWDJVQAZMFOLZ 7.5 IC50 10
SXXVFTHHNPFWFL 7.5 Ki 2
WJSJLTQPBJXQOW 7.5 Ki 4
YFCWBKBNFCDPDF 7.5 Ki 2
BTRMENQCGLMYLK 7.5 Ki 4
ZMRXSORFBXMBCB 7.5 IC50 8
BIERIKWXCCJADR 7.5 Ki 2
CNECFZVDGRAPIN 7.5 IC50 2
JBABGZDZOMSKLX 7.5 IC50 8
PFEJBPNFLAFPKN 7.5 IC50 10
RHQJWLPJMQCJOF 7.5 Ki 2
UIRMNVOEQMAKFM 7.5 IC50 7
XOXNEDDHVCBSGK 7.5 Ki 3
ZDKWIWBHZBARRN 7.5 IC50 2
ZKFJPGLUUMQAFH 7.5 Ki 2
IELBAACIVCODPI 7.5 IC50 8
2D structure