Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
GDXUHGVVRIPSQZ 7.8 Ki 5
NMIYWOZAHQVTIW 7.8 Ki 2
BMWDQBTXNBGORC 7.8 IC50 8
INYNWEUTASDACG 7.8 Ki 5
KWVYCGMBGRYVQH 7.8 Ki 4
WJSJLTQPBJXQOW 7.8 Ki 4
CREYMMOMGYLCND 7.8 Ki 2
OGHPAVPNKPGGDV 7.8 Ki 2
OWGROKMAKCBXPP 7.8 Ki 2
GITHBFKKVBHLFE 7.8 Ki 2
KEDWUBLQPZPFSQ 7.8 Ki 2
YMXSEXVSDUSENY 7.8 Ki 2
HFIMLFRJUJSWHZ 7.7 Ki 2
HGSHFGWWOPXUPH 7.7 IC50 2
XRIVGYHVHPSIIW 7.7 Ki 5
YMHTVJRMNCYCNZ 7.7 Ki 2
KXAAIPFSUGPVMQ 7.7 Ki 5
KXAAIPFSUGPVMQ 7.7 Ki 2
OPSFQCOCUXZPDB 7.7 Ki 4
OWQGYUFKEMELBK 7.7 Ki 2
YDGOUEKZXBLUDG 7.7 IC50 8
ZKFFJBXJJFDBJM 7.7 IC50 8
ZPZKWVOWBPNQFC 7.7 IC50 2
YPUPVMYOUBYNAY 7.7 IC50 2
IPCBFNXNVLCHMF 7.7 Ki 2
KZGXXLRPBQODHL 7.7 Ki 2
KZGXXLRPBQODHL 7.7 Ki 2
MRSAIDFRTZWWBE 7.7 Ki 2
MTYYINDDZCLHDE 7.7 Ki 2
QDIMTFLILFWWDN 7.7 IC50 2
QWEBUPURHNWVEK 7.7 IC50 5
SYTFEYDNYKQRMV 7.7 Ki 2
VBHJNDXDBMNCHU 7.7 IC50 2
YDLFIHZHGDGEQV 7.7 Ki 2
CCGVLNAUEKVICK 7.7 IC50 8
FOBOXOHWDKQRAH 7.7 IC50 4
MZCXDLPGCAZQJL 7.7 Ki 2
NBNDFLJNAYAZMD 7.7 IC50 4
NNKLMOMWOOXRDH 7.7 Ki 2
RNOBTWYQAWEZHH 7.7 Ki 4
RSEXFRQQJHVYPG 7.7 IC50 4
SITVIGRZUIUBEV 7.7 IC50 2
WYTGRFGLIURWGC 7.7 Ki 2
HMSUQCBFNZLLMB 7.7 IC50 2
IGHCCJIYQAMMPL 7.7 Ki 2
INYNWEUTASDACG 7.7 Ki 5
XOEJXZGEXAMGIL 7.7 Ki 4
IDNNDKWFPXHHMF 7.7 Ki 2
JYHOJSHACNBFKD 7.7 IC50 2
HDLZINNMWOTETA 7.6 Ki 2
2D structure