Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
VBQDZZHUUPHQGQ 8.0 IC50 11
JYBXLCIZWPNCMU 8.0 IC50 11
LIWBYJGLHCGRCM 8.0 Ki 8
PSXPQUNJMZAIKK 8.0 Ki 2
RPPABJHZNYUIDN 8.0 Ki 2
XJDTUPZAYLTURR 8.0 IC50 2
HLOGNWFNJMJTFF 8.0 Ki 2
HMCIAPJBFDNMOO 8.0 Ki 2
ZRUCSUZKLOXDQK 8.0 IC50 2
ACPHUHSYZGYUCK 8.0 Ki 5
PQACGZHZKXPWQM 8.0 Ki 2
SPTQZFUOJBUHQA 8.0 IC50 5
FBTSLPXYWKHFJN 8.0 Ki 5
OHKODMIWVVUDGL 8.0 Ki 4
YRJXIUNIRVSCPU 8.0 Ki 2
CRXFCGUGNWJSEY 7.9 Ki 5
HFZDMKMXPGRKCK 7.9 Ki 2
IZXOINQUSUGYPF 7.9 Ki 4
JLHNNIALZUDMPM 7.9 IC50 4
SCQZRFDFSKEVKQ 7.9 Ki 4
SNPPWIUOZRMYNY 7.9 IC50 5
VGFNJHVYMJKBLY 7.9 Ki 2
YERXBIUSFBYSAG 7.9 Ki 2
GFWIBMSUBMVIDR 7.9 IC50 2
JPRGWWSALFMHMG 7.9 Ki 2
FRPOHHKGFSZXFJ 7.9 Ki 2
JYUTVPNZUICOSN 7.9 Ki 4
NZYPTMVAFUKKKD 7.9 Ki 2
VEDPMPOSMIIBBR 7.9 Ki 2
XVFBZAKFUWQJMY 7.9 Ki 2
ZIFKLIOWIKMCIM 7.9 Ki 2
ZJSCNDMSVCKOLZ 7.9 Ki 2
ZMEGTXPZASMCHV 7.9 Ki 3
FIIBHEYGLZGMCK 7.8 Ki 5
PSXPQUNJMZAIKK 7.8 Ki 2
QAOGJKYLKKJSNB 7.8 Ki 2
RQOGEOGXPQQGHI 7.8 Ki 2
SSDSOAIBEZINDQ 7.8 Ki 2
BKXZRLFPGYWHTM 7.8 IC50 7
KZTLNPPLLLJLHU 7.8 Ki 7
GIDJZDYNVHMFAH 7.8 IC50 9
JYUTVPNZUICOSN 7.8 Ki 3
LPUSMQXNPXCRTA 7.8 IC50 2
PEAGCBDUMAQJJR 7.8 IC50 2
BJLKZFUZNNATGZ 7.8 IC50 7
FTYHMMVUGBYQCJ 7.8 IC50 2
FTYHMMVUGBYQCJ 7.8 IC50 2
IBKIPEZDVFQTJT 7.8 Ki 5
PKRPUUWZLBLPCX 7.8 IC50 2
XLPXWVVFGRJJCY 7.8 Ki 2
2D structure