Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
MVQIWKVEEIZQLL 8.3 IC50 5
ZHQDDVCHGDJTCT 8.3 Ki 2
NMIIKXFGCKOYRV 8.2 IC50 5
JCOOLTXCASTQDG 8.2 Ki 2
RHYPCHMNNLGAHN 8.2 Ki 2
YIMFXBPXUPTIEJ 8.2 Ki 7
VXQLPXYMYHKASH 8.2 Ki 5
AFIZEQKQIKDZQH 8.2 Ki 2
FEIJFKLKIQDCEV 8.2 Ki 2
KMZCUSKKQFNPIY 8.2 Ki 5
ODWWODYTMVKWGE 8.2 Ki 5
XJUAPPAIWQVLER 8.2 Ki 2
KKVSVXVHHIOCHW 8.2 Ki 4
LUECZUZBDUKVMO 8.2 Ki 3
PYSCVJMLJRHJGJ 8.2 Ki 2
SHVHFZCMOBFTPO 8.2 Ki 2
ITPXKRKCDRCWLZ 8.2 IC50 2
WESGVHHRAFNWER 8.2 Ki 7
OHYANMWFAIMESB 8.2 Ki 4
OWYJMZSLCXNXPU 8.2 IC50 2
HFALPZZGNQXIMP 8.2 Ki 5
INYNWEUTASDACG 8.2 Ki 5
MPHNMTSXVNYBBU 8.2 Ki 4
NUQOQQYEHCYTBU 8.2 Ki 2
FAEVMLINNNVLLK 8.1 Ki 5
QDTDIHUMTXWBEH 8.1 Ki 2
IKBFUAJBNDCGFQ 8.1 Ki 7
NLPRAJRHRHZCQQ 8.1 Ki 2
WONBUILDJNKYCB 8.1 IC50 5
PREYWAJYVTVVPE 8.1 IC50 10
FHIJCASAUMRSAS 8.1 Ki 4
MLPOWHAMUPIMTC 8.1 IC50 4
RPPABJHZNYUIDN 8.1 Ki 2
RSJYAQNYOKPXLY 8.1 Ki 2
RUJFIXHHAWJMRM 8.1 Ki 5
VTZZSDWXGJOEAU 8.1 Ki 2
VZXFAFSZALKXPY 8.1 Ki 2
FDYKMNCWHGRGGQ 8.1 IC50 2
ILRKKMGSYJDPCB 8.1 Ki 2
PGTPXIBBHIHMQS 8.1 IC50 10
KPCBJGYPNGGQFN 8.1 Ki 2
WJSJLTQPBJXQOW 8.1 Ki 5
ABPSWEJOHYDZDP 8.0 IC50 11
SNICXCGAKADSCV 8.0 Ki 5
ACPHUHSYZGYUCK 8.0 Ki 5
FQIJPHXWIONJLF 8.0 IC50 2
PWXQAVZNBKKQOF 8.0 Ki 6
KISYGAAWAUCCJZ 8.0 Ki 2
MQVPACXYSJDEHQ 8.0 IC50 5
SPTQZFUOJBUHQA 8.0 Ki 3
2D structure