Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
KPHRNXIFUJLFNL 8.5 Ki 5
SHVHFZCMOBFTPO 8.5 Ki 2
VASDDDNKICCHAA 8.5 Ki 2
WHWGPUNVTOQEIM 8.5 Ki 2
PMLHYFDQPIWSKJ 8.5 Ki 4
BHFQBHBXODOWRO 8.5 Ki 5
HBRLNTBOOKFZCC 8.5 Ki 5
JRAZMHFHZFKHQJ 8.5 Ki 7
OPAZJRBBVVHUKF 8.5 Ki 2
USVAHAACEDZWOK 8.5 IC50 2
ZAJOQFQUHOWCFD 8.5 Ki 2
NZWLHYJVHGBBSI 8.5 Ki 2
PXJGFTOIRXIPQQ 8.5 Ki 2
OURWEQSYKPJJJA 8.5 Ki 2
AGJCEEAUUACOSG 8.5 Ki 2
FEOISNNNAYEFKH 8.5 Ki 2
WQVOCWHVRYZKFN 8.5 Ki 2
SLXGVSHQIUXHQI 8.4 Ki 2
YTKDGWHLDZNCMB 8.4 Ki 2
JQSHBVHOMNKWFT 8.4 Ki 3
LJEPPQATHWQMBV 8.4 Ki 5
ZTSSUVKQGBVRTE 8.4 Ki 2
HFALPZZGNQXIMP 8.4 Ki 5
HFIMLFRJUJSWHZ 8.4 Ki 4
HSTBEKFBYFHTES 8.4 Ki 2
OEWOQZPDLZUIGU 8.4 Ki 5
USXYDBGSWSSTGE 8.4 Ki 2
IGRBOGLDQXBDPE 8.4 IC50 2
OIPILFWXSMYKGL 8.4 Ki 6
XSOAGDBGBRRJLR 8.4 Ki 2
SOEBPVQMXRKIOZ 8.4 Ki 3
DRZJLSBEDUUOBI 8.4 Ki 2
VUROYLWVIMGNBJ 8.3 IC50 2
RKMOIOORHCEDOW 8.3 Ki 2
NTFKOQBZSNCLLA 8.3 Ki 4
SNICXCGAKADSCV 8.3 Ki 8
DWHQCXVYIKBENZ 8.3 IC50 2
MOMRLMDRIJFWPM 8.3 IC50 5
MOMRLMDRIJFWPM 8.3 IC50 3
MXYUKLILVYORSK 8.3 Ki 3
MXYUKLILVYORSK 8.3 Ki 2
SCQZRFDFSKEVKQ 8.3 Ki 4
WJSJLTQPBJXQOW 8.3 Ki 4
JFPXLNSBLNDHFH 8.3 Ki 3
UBBGAHHMACAFKM 8.3 Ki 2
CCEBJZRLEVFTNS 8.3 Ki 3
FAEVMLINNNVLLK 8.3 Ki 3
ROMQYXADXASYDV 8.3 Ki 4
AQYPBNGIIYVIBQ 8.3 Ki 5
HCVVQYDWEUQYOH 8.3 IC50 4
2D structure